Search results for "TERPENES"

showing 10 items of 470 documents

Selecting Microbial Strains from Pine Tree Resin: Biotechnological Applications from a Terpene World

2014

Resin is a chemical and physical defensive barrier secreted by many plants, especially coniferous trees, with insecticidal and antimicrobial properties. The degradation of terpenes, the main components accounting for the toxicity of resin, is highly relevant for a vast range of biotechnological processes, including bioremediation. In the present work, we used a resin-based selective medium in order to study the resin-tolerant microbial communities associated with the galls formed by the moth Retinia resinella; as well as resin from Pinus sylvestris forests, one of the largest ecosystems on Earth and a yet-unexplored source of terpene-degrading microorganisms. The taxonomic and functional di…

DNA BacterialAntifungal AgentsApplied MicrobiologyMicroorganismlcsh:MedicineMothsBiologyMicrobiologyTerpeneEnvironmental BiotechnologyBioremediationPhylogeneticsMicrobial PhysiologyPlant TumorsPseudomonasBotanyGeneticsRNA Ribosomal 18SAnimalsEcosystemlcsh:SciencePhylogenyMicrobial MetabolismMultidisciplinaryTerpeneslcsh:RPseudomonasFungitechnology industry and agricultureFungal geneticsBiology and Life SciencesGenomicsSequence Analysis DNAPinusbiology.organism_classificationAntimicrobiallcsh:QTranscriptomeBioremediationResins PlantResearch ArticleBiotechnologyPLoS ONE
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T-DNA insertion alters the terpenoid content composition and bioactivity of transgenic Artemisia annua.

2014

In this study, the interference of T-DNA insertion upon Agrobacterium-mediated transformation on the biochemical expression of the host genome is discussed. Plant extracts of transgenic Artemisia annua L. with or without an overexpressed farnesyl pyrophosphate synthase gene have been investigated for their bioactivity and metabolic profile in comparison with wild type A. annua. The highest antimicrobial activity against Staphylococcus aureus, Bacillus subtilis and Candida albicans was observed in the T253 transgenic lines. Moreover, the crude extract from T253 showed higher antimalarial activity against the Plasmodium faciparum K1 strain than those of the others. The terpenoid constituents…

DNA BacterialTransgeneArtemisia annuaPlant ScienceBacillus subtilisMicrobial Sensitivity TestsArtemisia annuaSqualenechemistry.chemical_compoundDrug DiscoveryBotanyPharmacologybiologyTerpenesfungiWild typeGeranyltranstransferaseGeneral Medicinebiology.organism_classificationAntimicrobialPlants Genetically ModifiedTerpenoidTransformation (genetics)Complementary and alternative medicinechemistryBiochemistryNatural product communications
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Inhibition of pro-inflammatory enzymes by inuviscolide, a sesquiterpene lactone from Inula viscosa

2006

Abstract This work concerns the pharmacological activity of inuviscolide, a sesquiterpenoid from Inula viscosa. It exerts inhibitory effects on elastase, cyclooxygenase 1 and secretory phospholipase A2. Furthermore, it reduces the skin leukocyte infiltration in a murine model of dermatitis induced by repeated application of 12-O-tetradecanoylphorbol 13-acetate.

DermatitisBiologyPharmacognosyPharmacologySesquiterpene lactoneSesquiterpeneLactonesMicechemistry.chemical_compoundDrug DiscoveryLeukocytesAnimalsHumansEnzyme InhibitorsPharmacologychemistry.chemical_classificationPancreatic Elastaseintegumentary systemPlant ExtractsAnti-Inflammatory Agents Non-SteroidalElastaseBiological activityGeneral MedicineEnzymechemistryBiochemistrybiology.proteinTetradecanoylphorbol AcetateInulaCyclooxygenaseSesquiterpenesLactonePhytotherapyFitoterapia
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Synthesis and comparison of the antiinflammatory activity of manoalide and cacospongionolide B analogues.

1998

We have synthesized analogues of two naturally occurring antiinflammatory marine compounds, manoalide and cacospongionolide B, containing a pyranofuranone moiety which is considered the pharmacophoric group. The two compounds, and hence their analogues, differ in the presence or absence in the dihydropyran ring of an hemiacetal function which was considered essential to irreversibly inactivate phospholipase A 2 (PLA 2 ). The two series of compounds were tested for their inhibitory effects on secretory PLA 2 belonging to the groups I, II, and III, and the activities were found to be similar in both series, irrespective of the presence or absence of the additional hemiacetal function. In addi…

DihydropyranStereochemistrySwineCarrageenanChemical synthesisPhospholipases ACell Linechemistry.chemical_compoundManoalideMiceStructure-Activity RelationshipCytosol4-ButyrolactoneDrug DiscoveryMoietyAnimalsEdemaHumansEnzyme InhibitorsPancreasPyranschemistry.chemical_classificationElapid VenomsPhospholipase AbiologyMolecular StructureTerpenesAnti-Inflammatory Agents Non-SteroidalSynovial MembraneBee VenomsKineticsPhospholipases A2chemistryEnzyme inhibitorDrug Designbiology.proteinMolecular MedicineHemiacetalFemaleLactoneJournal of medicinal chemistry
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The ethnobotany, phytochemistry, and biological properties of Nigella damascena – A review

2022

This review is a systematic scientific work on medicinal and traditional use, on the chemical composition of specialized metabolites, volatile and non-volatile, on aspects related to toxicology and phytotherapy of Nigella damascena L. The genus Nigella (Ranunculaceae) is distributed throughout the Mediterranean basin, extending to northern India, and has been divided into three sections. Nigella damanscena L. is traditionally used as an ingredient in food, for example, as flavouring agents in bread and cheese, but is also known in folk medicine, used to regulate menstruation; for catarrhal affections and amenorrhea; as a diuretic and sternutatory; as an analgesic, anti-oedematous, and antip…

Dolabellane diterpenesAntipyreticsβ-elemenePlant ExtractsPhytochemicalsEthnobotanyPlant ScienceGeneral MedicineSettore CHIM/06 - Chimica OrganicaHorticultureAnticancer propertiesBiochemistryNigella damascenaAnti-inflammatory aspectsFixed oilsEthnopharmacologySettore BIO/03 - Botanica Ambientale E ApplicataMedicine TraditionalSettore BIO/15 - Biologia FarmaceuticaMolecular BiologyRanunculaceaePhytotherapy
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Herbicidal Activity of Peumus boldus and Drimys winterii Essential Oils from Chile

2011

[EN] The essential oil composition of Peumus boldus and Drimys winterii was analyzed by means of capillary GC-FID and GC-MS. More than 96% of the total oil components (43 and 54 compounds, respectively) were identified, with ascaridole (51.17 ± 9.51), p-cymene (16.31 ± 2.52) and 1,8-cineole (14.45 ± 2.99) as the main compounds in P. boldus and ¿-eudesmol (21.65 ± 0.41), followed of elemol (12.03 ± 0.34) and terpinen-4-ol (11.56 ± 1.06) in D. winterii. The herbicidal activity was tested against Amaranthus hybridus and Portulaca oleracea. P. boldus essential oil was the most phytotoxic against both weeds, inhibiting seed germination and seedling growth at all concentrations assayed (0.125-1 ¿…

DrimysChromatography GasAmaranthus hybridusBOTANICAPharmaceutical ScienceGerminationPortulacaEssential oilArticleAnalytical Chemistrylaw.inventionlcsh:QD241-441chemistry.chemical_compoundlcsh:Organic chemistrylawDrug DiscoveryBotanyOils VolatilePhysical and Theoretical ChemistryChileSeedling growthEssential oilBIOLOGIA VEGETALGas chromatographybiologyMass spectrometryHerbicidesOrganic Chemistrybiology.organism_classificationDrimysChemistrychemistryIsolation and purificationChemistry (miscellaneous)GerminationSeedlingEssential oilsPhytotoxicityPeumusMonoterpenesMolecular MedicinePhytotoxicityHerbicideAscaridoleessential oils; phytotoxicity; germination; seedling growth; monoterpenesPeumus boldus
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Chemical composition and antimicrobial activity of the essential oils of some species of Anthemis sect. Anthemis (Asteraceae) from Sicily

2017

The chemical composition of the essential oils isolated from the aerial parts of Anthemis arvensis L. subsp. arvensis, Anthemis cretica subsp. messanensis (Brullo) Giardina & Raimondo and from flowers and leaves of Anthemis cretica subsp. columnae (Ten.) Frezén were determinated by GC–FID and GC–MS analyses. Torreyol (85.4%) was recognised as the main constituent of the Anthemis arvensis subsp. arvensis essential oil, while in the essential oils of Anthemis cretica subsp. messanensis, collected on the rock and cultivated in Hortus Botanicus Panormitanus, (E)-chrysanthenyl acetate (28.8 and 24.2% resp.), 14-hydroxy-α-humulene (8.1 and 5.3% resp.), santolina triene (8 and 5.8% resp.) and …

Drug Evaluation PreclinicalRaimondoAnthemis arvensisFlowersMicrobial Sensitivity TestsPlant Science01 natural sciencesBiochemistryGas Chromatography-Mass Spectrometryessential oillaw.inventionAnalytical Chemistrychemistry.chemical_compoundBridged Bicyclo CompoundsAnti-Infective Agentsantibacterial activitylawSantolinaBotanyOils VolatileAnthemisSettore BIO/15 - Biologia FarmaceuticaChemical compositionSicilyAnthemis arvensis L. subsp. arvensiEssential oiltorreyolBicyclic MonoterpenesPolycyclic Sesquiterpenesalpha-PineneEucalyptolbiology010405 organic chemistryOrganic ChemistryAnthemis cretica subsp. columnae (Ten.) FrezénAsteraceaebiology.organism_classificationCyclohexanols0104 chemical sciencesPlant Leaves010404 medicinal & biomolecular chemistryEucalyptolchemistryMonoterpenesAnthemis cretica subsp. messanensis (Brullo) Giardina &ampAnthemisSesquiterpenes
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Coscinolactams A and B: new nitrogen-containing sesterterpenoids from the marine sponge Coscinoderma mathewsi exerting anti-inflammatory properties

2009

Abstract Investigation of the marine sponge Coscinoderma mathewsi led to the isolation of two novel nitrogen-containing cheilanthane sesterterpenoids, coscinolactams A and B, together with known suvanine. The structures were elucidated by extensive spectroscopic measurements including NOE experiments to deduce the stereochemistry. The natural compounds, as well as a semisynthetic derivative, showed moderate anti-inflammatory activity measured as their capability to inhibit PGE2 and NO production. The suvanine aldehyde derivative 4 inhibited inducible nitric oxide protein expression with an IC50 value of 7.3 μM.

EXTRACTIONmedicine.drug_classStereochemistrySesterterpenoidsBiochemistryAldehydeAnti-inflammatorySesterterpenesNitric oxidechemistry.chemical_compoundAnti-inflammatory activityEPONGESpongeDrug DiscoverymedicineOrganic chemistryIC50ACTIVITE ANTIINFLAMMATOIREchemistry.chemical_classificationTESTACTIVITE BIOLOGIQUEbiologyOrganic ChemistryINVERTEBRE AQUATIQUEbiology.organism_classificationTerpenoidSpongechemistrySUBSTANCE NATURELLEDerivative (chemistry)
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Terpenoid treatment in osteoporosis: this is where we have come in research.

2021

Lower bone resistance to load is due to the imbalance of bone homeostasis, where excessive bone resorption, compared with bone formation, determines a progressive osteopenia, leading to a high risk of fractures and consequent pain and functional limitations. Terpenoids, with their activities against bone resorption, have recently received increased attention from researchers. They are potentially more suitable for long-term use compared with traditional therapeutics. In this review of the literature of the past 5 years, we provide comprehensive information on terpenoids, with their anti-osteoporotic effects, highlighting molecular mechanisms that are often in epigenetic key and a possible p…

Endocrinology Diabetes and MetabolismOsteoporosisBioinformaticsBone resorptionBone and BonesFractures BoneEndocrinologyOsteoclastterpenoidsSettore BIO/13 - Biologia ApplicataSettore BIO/10 - Biochimicamedicinebone erosive diseasesHumansBone formationBone ResorptionProgressive osteopeniaepigeneticsbusiness.industryTerpenesOsteoporosis preventionOsteoblastmedicine.diseaseSettore BIO/18 - Geneticamedicine.anatomical_structureosteoclastosteoblastOsteoporosisbusinessTrends in endocrinology and metabolism: TEM
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Biological effects and photodegradation by TiO(2) of terpenes present in industrial wastewater.

2010

Abstract The aim of this work was to study the biological effects of four monoterpenes, i.e. α-pinene, β-pinene, 3-carene and d -limonene present in the wastewater of a citrus transformation factory. The study was carried out by exposing V79 Chinese hamster cells to single terpene or to the mixture of four terpenes at concentrations corresponding to those in the wastewater evaluated by head space solid phase micro extraction and gas chromatography (HS-SPME-GC) analyses. Treatments with single or combined terpenes similarly affected cell vitality, but only the combined treatments induced the 6-thioguanine resistant mutants. Moreover the photocatalytic degradation of the four terpenes was suc…

Environmental EngineeringChromatography GasSettore CHIM/10 - Chimica Degli AlimentiHealth Toxicology and MutagenesisIndustrial WasteCatalysisCell LineTerpeneIndustrial wastewater treatmentchemistry.chemical_compoundCricetulusCricetinaeEnvironmental ChemistryAnimalsWater PollutantsPhotodegradationWaste Management and DisposalEffluentSolid Phase MicroextractionTitaniumLimoneneChromatographyPhotolysisTerpenesTerpenes clonogenicassay Terpenes mutationassay TiO2 photocatalysisPollutionSettore BIO/18 - GeneticaWastewaterchemistryEnvironmental chemistryPhotocatalysisSettore CHIM/07 - Fondamenti Chimici Delle TecnologieGas chromatographyJournal of hazardous materials
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