Search results for "YAP"

showing 8 items of 268 documents

Anti-inflammatory activity of flavonoids from Cayaponia tayuya roots.

2008

Taiuiá or tayuya (Cayaponia tayuya, Cucurbitaceae) is a climbing, lignified plant with a large swollen root that has traditionally been used as an anti-inflammatory and anti-rheumatic agent in the folk medicine of Brazil, Peru, and Colombia.We have assayed the pharmacological properties of a flavonoid fraction obtained from the butanol extract of Cayaponia tayuya roots using two models of topical mouse ear oedema, paying special attention to its influence on the induction on pro-inflammatory enzymes and peptidic mediators.The in vivo experiments involved both the acute oedema induced by a single application of TPA and the subchronic inflammation brought on by repeated applications of TPA. T…

medicine.drug_classFlavonoidIsovitexinAnti-Inflammatory AgentsNitric Oxide Synthase Type IIPharmacologyPharmacognosyColombiaPlant RootsAnti-inflammatoryCell Linechemistry.chemical_compoundMiceWestern blotIn vivoDrug DiscoveryPerumedicineAnimalsPharmacologychemistry.chemical_classificationFlavonoidsInflammationbiologymedicine.diagnostic_testbusiness.industryPlant ExtractsMacrophagesbiology.organism_classificationCayaponia tayuyaCucurbitaceaeDisease Models AnimalchemistryBiochemistryCyclooxygenase 2biology.proteinFemaleCyclooxygenaseMedicine TraditionalbusinessBrazilJournal of ethnopharmacology
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Anti-inflammatory activity of two cucurbitacins isolated from Cayaponia tayuya roots.

2004

Fractionation of an anti-inflammatory extract from Cayaponia tayuya roots yielded two active compounds, identified as 23,24-dihydrocucurbitacin B (1) and cucurbitacin R (2). Both were evaluated for their anti-inflammatory activity on several experimental models of pain and inflammation. In addition, their cytotoxicity and effects on leukotriene B 4 (LTB 4 ) formation were evaluated in rat polymorphonuclear leukocytes. Both compounds showed activity in the following models: carrageenan-induced mouse paw oedema (1, 4 mg/kg p.o., 46% inhibition at 3 h), phospholipase A 2 -induced mouse paw oedema (2, 3 mg/kg i.p., 61% inhibition at 60 min), serotonin-induced mouse paw oedema (1 and 2, 0.5 mg/k…

medicine.drug_classLeukotriene B4Pharmaceutical ScienceAdministration OralPainPharmacologyAdministration CutaneousCarrageenanLeukotriene B4Plant RootsAnti-inflammatoryPhospholipases AAnalytical Chemistrychemistry.chemical_compoundMicePhospholipase A2Drug DiscoverymedicineLeukocytesAnimalsEdemaRats WistarPharmacologyPhospholipase AbiologyDose-Response Relationship DrugPlant ExtractsAntiglucocorticoidOrganic ChemistryAnti-Inflammatory Agents Non-SteroidalCucurbitacinsbiology.organism_classificationCayaponia tayuyaTriterpenesCarrageenanRatsCucurbitaceaePhospholipases A2Complementary and alternative medicinechemistryBiochemistryEicosanoidbiology.proteinMolecular MedicineTetradecanoylphorbol AcetateFemalePhytotherapyPlanta medica
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Dihydrocucurbitacin B, isolated from Cayaponia tayuya, reduces damage in adjuvant-induced arthritis

2005

23,24-Dihydrocucurbitacin B, from the anti-rheumatic plant Cayaponia tayuya, was tested on arthritis induced by adjuvant to corroborate the anti-inflammatory properties of this plant. Arthritis was induced in Lewis rats; the resulting arthritic rats were then treated with dihydrocucurbitacin B (1 mg/kg orally, daily, 1 week). The effect of dihydrocucurbitacin B on the synthesis, release, and activity of pro-inflammatory enzymes (elastase, cyclooxygenase-2, and nitric oxide synthase-2) as well as its effect on different mediators (tumor necrosis factor-alpha and interleukin-1beta) were determined. Dihydrocucurbitacin B modified the evolution of the clinical symptoms, reducing the swelling an…

medicine.medical_specialtyCell Survivalmedicine.medical_treatmentAnti-Inflammatory AgentsAdministration OralNitric Oxide Synthase Type IIPainArthritisPlant RootsDinoprostoneCell LineNitric oxidechemistry.chemical_compoundSuperoxidesInternal medicinemedicineAnimalsLymphocytesNitritesPharmacologyDose-Response Relationship DrugPancreatic ElastasebiologyPlant Extractsbusiness.industryMacrophagesElastasemedicine.diseasebiology.organism_classificationArthritis ExperimentalTriterpenesCayaponia tayuyaRatsEnzyme ActivationNitric oxide synthaseCucurbitaceaeEndocrinologyCytokinechemistryCyclooxygenase 2Rats Inbred LewAntirheumatic AgentsToxicitybiology.proteinCytokinesFemaleTumor necrosis factor alphabusinessPhytotherapyEuropean Journal of Pharmacology
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The influence of ossein-hydroxyapatite compound ('Ossopan') on the healing of a bone defect.

1986

A study was undertaken in 60 adult rabbits in order to determine the effects of ossein-hydroxyapatite compound on bone healing. Standardized bony defects were produced in the distal femoral epiphyses, after which animals were randomized into four equal groups. An untreated group served as a control. One group received ossein-hydroxyapatite compound, 830 mg per day, a second group received bone mineral (ossein-hydroxyapatite compound reduced to ash, to remove organic constituents), 510 mg per day, and a third group received calcium carbonate, 650 mg per day. A series of fluorescent vital markers was administered to the animals from the 7th to the 32nd day after production of the defect. A th…

medicine.medical_specialtyDentistryBone healingMineralization (biology)Bone remodelingCalcium Carbonatechemistry.chemical_compoundFractures BoneInternal medicinemedicineAnimalsHydroxyapatitesFemurBone regenerationBone mineralWound Healingbusiness.industryGeneral MedicineCalcium carbonateEndocrinologyDurapatitechemistryMicroscopy FluorescenceDietary mineralDrug EvaluationFemaleHydroxyapatitesRabbitsbusinessCurrent medical research and opinion
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New hydroxyapatite- and selenium-based nanoformulations as potential antimicrobial tools for orthopedic implants

selenium nanoparticles hydroxyapatite inorganic-inorganic complexesSettore CHIM/02 - Chimica Fisica
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MORPHOSTRUCTURAL ANALYSIS OF HUMAN DENTAL FOLLICULAR STEM CELLS ON HIGLY POROUS BONE HYDROXYAPATITE SCAFFOLD

2007

In this study we investigated the in vitro behaviour, morphostructure and extracellular matrix synthesis of human dental follicular stem cells (hDFSCs) isolated from human dental bud, which resulted to be positive for mesenchymal markers (CD29, CD90, CD146 and CD166) by FACS analysis. Cells were analysed by light and electronic microscopy to evaluate their biological response either at week 1, that is before differentiation, or at weeks 3-6, when they had been cultured in osteogenic medium onto a highly porous natural scaffold material (Bio-Oss). Microscopy analysis of primary culture cells showed they had a mesenchymal stem cell-like morphostructure, spindle shaped, similar to the culture …

stem cellporous bone hydroxyapatite (Bio-Oss (R)tissue engineeringdental follicle
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Stability of stochastic nonlinear systems with state-dependent switching

2013

In this paper, the problem of stability on stochastic systems with state-dependent switching is investigated. To analyze properties of the switched system by means of Itô’s formula and Dynkin’s formula, it is critical to show switching instants being stopping times. When the given active-region set can be replaced by its interior, the local solution of the switched system is constructed by defining a series of stopping times as switching instants, and the criteria on global existence and stability of solution are presented by Lyapunov approach. For the case where the active-region set can not be replaced by its interior, the switched systems do not necessarily have solutions, thereby quasi-…

stochastic systemsStability (learning theory)Mathematical proofnonlinear control systemsSet (abstract data type)State-dependent switching; Stochastic systems; Switched systems; Control and Systems Engineering; Computer Science Applications1707 Computer Vision and Pattern Recognition; Electrical and Electronic EngineeringExponential stabilityControl theoryElectrical and Electronic EngineeringSwitched systemsMathematicsLyapunov methodsStochastic systemsSeries (mathematics)Stochastic processApplied MathematicsComputer Science Applications1707 Computer Vision and Pattern Recognitionstate-dependent switchingstabilityComputer Science ApplicationsNonlinear systemControl and Systems EngineeringState dependentswitched systemscontrol system synthesisState-dependent switching
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Efficient zinc incorporation into hydroxyapatite through crystallization of an amorphous phase could extend the properties of zinc apatites

2013

zinc:TECHNOLOGY::Materials science [Research Subject Categories]hydroxyapatiteantimicrobial resistanceamorphous calcium phosphate
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