0000000001182738

AUTHOR

Jin Huang

showing 2 related works from this author

Discovery of Natural Products as Novel and Potent FXR Antagonists by Virtual Screening

2018

Farnesoid X receptor (FXR) is a member of nuclear receptor family involved in multiple physiological processes through regulating specific target genes. The critical role of FXR as a transcriptional regulator makes it a promising target for diverse diseases, especially those related to metabolic disorders such as diabetes and cholestasis. However, the underlying activation mechanism of FXR is still a blur owing to the absence of proper FXR modulators. To identify potential FXR modulators, an in-house natural product database (NPD) containing over 4,000 compounds was screened by structure-based virtual screening strategy and subsequent hit-based similarity searching method. After the yeast t…

0301 basic medicinenatural product01 natural scienceslcsh:Chemistry03 medical and health scienceschemistry.chemical_compoundTranscriptional regulationGeneIC50Original ResearchVirtual screeningNatural productantagonistmolecular dockingsimilarity searchingGeneral Chemistryvirtual screening0104 chemical sciencesChemistry010404 medicinal & biomolecular chemistry030104 developmental biologyFXRlcsh:QD1-999Nuclear receptorBiochemistrychemistryFarnesoid X receptorGuggulsteroneFrontiers in Chemistry
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An Adaptive Metamodel-Based Optimization Approach for Vehicle Suspension System Design

2014

Published version of an article in the journal: Mathematical Problems in Engineering. Also available from the publisher at: http://dx.doi.org/10.1155/2014/965157 The performance index of a suspension system is a function of the maximum and minimum values over the parameter interval. Thus metamodel-based techniques can be used for designing suspension system hardpoints locations. In this study, an adaptive metamodel-based optimization approach is used to find the proper locations of the hardpoints, with the objectives considering the kinematic performance of the suspension. The adaptive optimization method helps to find the optimum locations of the hardpoints efficiently as it may be unachie…

Continuous optimizationMathematical optimizationEngineeringArticle SubjectAdaptive optimizationbusiness.industryGeneral MathematicsProbabilistic-based design optimizationlcsh:MathematicsVDP::Technology: 500::Mechanical engineering: 570General EngineeringInterval (mathematics)Kinematicslcsh:QA1-939Multi-objective optimizationEngineering (all)lcsh:TA1-2040Mathematics (all)Multi-swarm optimizationbusinessSuspension (vehicle)lcsh:Engineering (General). Civil engineering (General)Mathematics (all); Engineering (all)Mathematical Problems in Engineering
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