Phosphonium-Boronate Amino Acid Derivatives as Fluoride Pincers for 18F-Labelling

6533b7d1fe1ef96bd125cbbd

RESEARCH PRODUCT

Phosphonium-Boronate Amino Acid Derivatives as Fluoride Pincers for 18F-Labelling

Julie Bernard Benjamin P. Burke Marie-joëlle Eymin Gonçalo S. Clemente Stephen J. Archibald Sylvain Jugé Raluca Malacea-kabbara

subject

inorganic chemicals chemistry.chemical_classification Organic Chemistry digestive system Biochemistry Amino acid Inorganic Chemistry chemistry.chemical_compound chemistry Labelling Organic chemistry heterocyclic compounds Phosphonium Fluoride

description

The synthesis of phosphonium-boronate amino acid derivatives was achieved by quaternization of o-boronatophenylphosphine with iodo-amino acid derivatives. Preliminary radiolabelling studies demonst...

year	journal	country	edition	language
2015-06-03	Phosphorus, Sulfur, and Silicon and the Related Elements

https://doi.org/10.1080/10426507.2014.979991

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