ChemInform Abstract: Gold-Catalyzed Tandem Hydroamination/Formal Aza-Diels-Alder Reaction of Homopropargyl Amino Esters: A Combined Computational and Experimental Mechanistic Study.

6533b7d8fe1ef96bd126a124

RESEARCH PRODUCT

ChemInform Abstract: Gold-Catalyzed Tandem Hydroamination/Formal Aza-Diels-Alder Reaction of Homopropargyl Amino Esters: A Combined Computational and Experimental Mechanistic Study.

Javier Miró Javier Gonzalez Santos Fustero María Sánchez-roselló Carlos Del Pozo

subject

Amino esters Tandem Chemistry Aza-Diels–Alder reaction General Medicine Hydroamination Combinatorial chemistry Catalysis Stereocenter

description

Under optimized conditions, the title reaction leads to formation of a tetracyclic nitrogen-containing framework with generation of 4 bonds and 5 stereocenters.

year	journal	country	edition	language
2015-08-01	ChemInform

https://doi.org/10.1002/chin.201534196

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