6533b7dafe1ef96bd126f6d7

RESEARCH PRODUCT

‘Interrupted’ diazotization of 3-aminoindoles and 3-aminopyrroles

Péter MátyusBarbara ParrinoAnna CarboneVirginia SpanòPaola BarrajaPatrizia DianaAlessandra MontalbanoGirolamo Cirrincione

subject

chemistry.chemical_classificationQuenching (fluorescence)Organic ChemistryInorganic chemistryPhotochemistryBiochemistrySettore CHIM/08 - Chimica Farmaceuticachemistry.chemical_compoundchemistryNitrateDrug DiscoveryAmino pyrroles Aminoindoles Diazoindoles Diazo pyrrolesNitriteCounterion

description

Abstract ‘Interrupted’ diazotization of 3-aminoindoles and 3-aminopyrroles, achieved by quenching with cold water immediately after the addition of nitrite, led, in good yields, to stable compounds whose structures were identified to be the diazonium species with nitrate as the counter ion, which show no saline character.

10.1016/j.tet.2014.07.051http://hdl.handle.net/10447/97018