The formation of pyrazolo[1,5-a]pyrimidines by the reaction of 3-(4-chlorophenyl)pyrazol-5-amine with chalcones

6533b823fe1ef96bd127e3ae

RESEARCH PRODUCT

The formation of pyrazolo[1,5-a]pyrimidines by the reaction of 3-(4-chlorophenyl)pyrazol-5-amine with chalcones

Herbert Meier Norbert Hanold Jairo Quiroga Marina Larrahondo Braulio Insuasty Ricardo Rincon

subject

Chemistry Yield (chemistry)Organic Chemistry Amine gas treating Medicinal chemistry

description

Cyclocondensation reactions of the pyrazol-5-amine 1 and the 1-aryl-3-phenyl-2-propen-1-ones 2a-d yield the 6,7-dihydropyrazolo[1,5-a]pyrimidines 7a-d. Whereas 7a-c can be isolated in pure state, 7d is subjected to a spontaneous oxidation.

year	journal	country	edition	language
1994-11-01

http://www.scopus.com/inward/record.url?eid=2-s2.0-0028569599&partnerID=MN8TOARS

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