Synthesis of Fluorinated and Nonfluorinated Tebufenpyrad Analogues for the Study of Anti-angiogenesis MOA

6533b828fe1ef96bd1288675

RESEARCH PRODUCT

Synthesis of Fluorinated and Nonfluorinated Tebufenpyrad Analogues for the Study of Anti-angiogenesis MOA

Saba Husain Maria Alvim-gaston Antonio Simón-fuentes Santos Fustero Dariusz Wodka Antonio Navarro Natalie Franklin Raquel Román

subject

Tebufenpyrad chemistry.chemical_compound Chemistry Anti angiogenesis Stereochemistry Drug discovery Phenotypic screening Organic Chemistry Physical and Theoretical Chemistry Combinatorial chemistry

description

In this contribution we report the synthesis of fluorinated and nonfluorinated tebufenpyrad analogues to explore potential druglike properties through the phenotypic screening as part of the Lilly Open Innovation Drug Discovery (OIDD) program.

year	journal	country	edition	language
2014-06-17

https://fundanet.cipf.es/Publicaciones/ProdCientif/PublicacionFrw.aspx?id=2379

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