Targeting the Class A Carbapenemase GES-5 via Virtual Screening

6533b832fe1ef96bd129a4a9

RESEARCH PRODUCT

Targeting the Class A Carbapenemase GES-5 via Virtual Screening

Martina Montanari Donatella Tondi Raphael Klein Pierangelo Bellio Giuseppe Celenza Laura Cendron Ruth Brenk Lorenzo Maso

subject

Models Molecular Drug antibiotic resistance GES-5 Antibiotic resistance media_common.quotation_subject In silico Drug Evaluation Preclinical lcsh:QR1-502 Guyana extended-spectrum-β-lactamase Microbial Sensitivity Tests Computational biology Biology Biochemistry beta-Lactamases Article lcsh:Microbiology guyana extended-spectrum-β-lactamase carbapenemase 03 medical and health sciences Antibiotic resistance Bacterial Proteins Drug Resistance Bacterial Humans Antibiotic resistance; GES-5; Guyana extended-spectrum-β-lactamase; carbapenemase; virtual screening; docking; noncovalent inhibition ges-5 noncovalent inhibition Molecular Biology 030304 developmental biology media_common 0303 health sciences Virtual screening 030306 microbiology Antibiotic resistance; Carbapenemase; Docking; GES-5; Guyana extended-spectrum-β-lactamase; Noncovalent inhibition; Virtual screening Hit to lead virtual screening Antimicrobial Anti-Bacterial Agents Carbapenems docking

description

The worldwide spread of &beta

year	journal	country	edition	language
2020-02-01	Biomolecules

https://doi.org/10.3390/biom10020304

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