Synthesis ofN-Tosylguanidinesby Ring Cleavage of 1,2-Dihydro-2-tosyliminopyrimidines

6533b854fe1ef96bd12addb7

RESEARCH PRODUCT

Synthesis ofN-Tosylguanidinesby Ring Cleavage of 1,2-Dihydro-2-tosyliminopyrimidines

José Sepúlveda-arques Jamal Lasri M. Eugenia González-rosende

subject

Nucleophilic addition Stereochemistry Chemistry Organic Chemistry Amine gas treating Cleavage (embryo)Ring (chemistry)Catalysis

description

The present communication discloses a new synthetic method for the preparation of N-tosylguanidines in high yields by ring cleavage of 1,2-dihydro-2-tosyliminopyrimidines with methyl- amine.

year	journal	country	edition	language
2003-01-01	Synthesis

https://doi.org/10.1055/s-2003-38684

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