ChemInform Abstract: Leaving Group and Regioselectivity Switches in the Aminoalkylation Reaction of Indoles and Related Heterocycles with α-Amido Sulfones.

6533b854fe1ef96bd12ae80c

RESEARCH PRODUCT

ChemInform Abstract: Leaving Group and Regioselectivity Switches in the Aminoalkylation Reaction of Indoles and Related Heterocycles with α-Amido Sulfones.

José R. Pedro Gonzalo Blay Marc Montesinos-magraner Rosa M. Giron

subject

Chemistry Leaving group Regioselectivity General Medicine Medicinal chemistry Pyrrole derivatives

description

Two methods are presented which allow the regioselective C- or N-aminoalkylation of indoles, pyrroles or azaindoles.

year	journal	country	edition	language
2013-10-14	ChemInform

https://doi.org/10.1002/chin.201345111

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