ChemInform Abstract: Synthesis, Benzodiazepine Receptor Binding and Molecular Modelling of Isochromeno[4,3-c]pyrazol-5(1H)-one Derivatives.

6533b86dfe1ef96bd12ca79c

RESEARCH PRODUCT

ChemInform Abstract: Synthesis, Benzodiazepine Receptor Binding and Molecular Modelling of Isochromeno[4,3-c]pyrazol-5(1H)-one Derivatives.

Livia Basile Salvatore Guccione Benedetta Maggio Fabiana Plescia Claudia Martini Maria Valeria Raimondi Maria Letizia Trincavelli Demetrio Raffa Fiorella Meneghetti Giuseppe Daidone

subject

Membrane Bovine brain Chemistry Stereochemistry medicine General Medicine Flunitrazepam Benzodiazepine receptor binding medicine.drug

description

A series of isochromeno[4,3-c]pyrazol-5(1H)-one derivatives (III) is prepared and tested for their ability to displace specific [3H]flunitrazepam from bovine brain membranes.

year	journal	country	edition	language
2012-11-29	ChemInform

https://doi.org/10.1002/chin.201250143

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