Search results for " 50"

showing 10 items of 2715 documents

Fusta de les serres ibériques (1750-1790) : L'impacte de la demanda per a la construcció fluvial a Cartagena

2014

0210-086X 364 Cuadernos de geografía 396981 2014 95-96 5076880 Fusta de les serres ibériques (1750-1790) L'impacte de la demanda per a la construcció fluvial a Cartagena Piqueras Haba:GEOGRAFÍA [UNESCO]JuanSanchís DeusaMaría del Carmen 67 99UNESCO::GEOGRAFÍA
researchProduct

La inserción de las ciudades en las redes globales a través de las relaciones financieras : El caso de la ciudad de Valencia

2014

0210-086X 364 Cuadernos de geografía 396981 2014 95-96 5076881 La inserción de las ciudades en las redes globales a través de las relaciones financieras El caso de la ciudad de Valencia Salom Carrasco:GEOGRAFÍA [UNESCO]Julia 101 123UNESCO::GEOGRAFÍA
researchProduct

Las almadrabas del Reino de Valencia entre finales del siglo XVI e inicios del XVII

2018

0210-9093 553 Estudis: Revista de historia moderna 500918 2018 44 6623952 Las almadrabas del Reino de Valencia entre finales del siglo XVI e inicios del XVII Vidal BonavilaUNESCO::HISTORIAJudit 107 133:HISTORIA [UNESCO]Revista de historia moderna 500918 2018 44 6623952 Las almadrabas del Reino de Valencia entre finales del siglo XVI e inicios del XVII Vidal Bonavila [0210-9093 553 Estudis]
researchProduct

Creiximent de la població, mortalitat, natalitat i migracions a les comarques de Tarragona (1700-1860)

2018

0210-9093 553 Estudis: Revista de historia moderna 500918 2018 44 6623956 Creiximent de la poblacióUNESCO::HISTORIAmortalitat:HISTORIA [UNESCO]natalitat i migracions a les comarques de Tarragona (1700-1860) Ferrer i AlòsRevista de historia moderna 500918 2018 44 6623956 Creiximent de la població [0210-9093 553 Estudis]Llorenç 197 223
researchProduct

Damage identification of a jacket support structure for offshore wind turbines

2020

Offshore jacket structures are regarded as a suitable type of support structure for offshore wind turbines in immediate water depths. Because of the welded tubular members used and environmental conditions, offshore jackets are often subjected to fatigue damages during their service life. Underwater sensors can provide measurements of the structural vibration signals and provide an efficient way to detect damages at early stages. In this work, simplified forms of the damages are assumed, random damages are imposed on the jacket structure, and damaged indicators are established from combination of modal shapes. Then, a response surface is constructed mapping the damage indicators and damages…

0211 other engineering and technologiesComputingMilieux_LEGALASPECTSOFCOMPUTING020101 civil engineering02 engineering and technology0201 civil engineeringVDP::Teknologi: 500Identification (information)Offshore wind powerStructural vibrationService lifeDamagesEnvironmental scienceSubmarine pipeline021108 energySensitivity (control systems)UnderwaterMarine engineering
researchProduct

The regression Tsetlin machine: a novel approach to interpretable nonlinear regression

2019

Relying simply on bitwise operators, the recently introduced Tsetlin machine (TM) has provided competitive pattern classification accuracy in several benchmarks, including text understanding. In this paper, we introduce the regression Tsetlin machine (RTM), a new class of TMs designed for continuous input and output, targeting nonlinear regression problems. In all brevity, we convert continuous input into a binary representation based on thresholding, and transform the propositional formula formed by the TM into an aggregated continuous output. Our empirical comparison of the RTM with state-of-the-art regression techniques reveals either superior or on par performance on five datasets. Thi…

021110 strategic defence & security studiesTheoretical computer scienceEmpirical comparisonComputer scienceGeneral Mathematics0211 other engineering and technologiesGeneral EngineeringGeneral Physics and AstronomyBinary number02 engineering and technologyThresholdingRegressionPropositional formula0202 electrical engineering electronic engineering information engineering020201 artificial intelligence & image processingBitwise operationTheme (computing)Nonlinear regressionVDP::Teknologi: 500::Informasjons- og kommunikasjonsteknologi: 550
researchProduct

Kick Detection and Influx Size Estimation during Offshore Drilling Operations using Deep Learning

2019

An uncontrolled or unobserved influx or kick during drilling has the potential to induce a well blowout, one of the most harmful incidences during drilling both in regards to economic and environmental cost. Since kicks during drilling are serious risks, it is important to improve kick and loss detection performance and capabilities and to develop automatic flux detection methodology. There are clear patterns during a influx incident. However, due to complex processes and sparse instrumentation it is difficult to predict the behaviour of kicks or losses based on sensor data combined with physical models alone. Emerging technologies within Deep Learning are however quite adapt at picking up …

021110 strategic defence & security studiesgeographygeography.geographical_feature_categoryArtificial neural networkComputer sciencebusiness.industryDeep learning0211 other engineering and technologiesDrilling0102 computer and information sciences02 engineering and technology01 natural sciencesWellboreVDP::Teknologi: 500Drilling machines010201 computation theory & mathematicsInstrumentation (computer programming)Artificial intelligencebusinessOffshore drillingMarine engineeringWater well2019 14th IEEE Conference on Industrial Electronics and Applications (ICIEA)
researchProduct

2,3-Dihydrobenzofuran privileged structures as new bioinspired lead compounds for the design of mPGES-1 inhibitors

2016

International audience; 2,3-Dihydrobenzofurans are proposed as privileged structures and used as chemical platform to design small compound libraries. By combining molecular docking calculations and experimental verification of biochemical interference, we selected some potential inhibitors of microsomal prostaglandin E2 synthase (mPGES)-1. Starting from low affinity natural product 1, by our combined approach we identified the compounds 19 and 20 with biological activity in the low micromolar range. Our data suggest that the 2,3-dihydrobenzofuran derivatives might be suitable bioinspired lead compounds for development of new generation mPGES-1 inhibitors with increased affinity.

0301 basic medicine300323-Dihydrobenzofuran privileged structure; Cancer; Inflammation; Molecular docking; mPGES-1 inhibitors; Biochemistry; Clinical Biochemistry; Molecular Biology; Molecular Medicine; Organic Chemistry; Drug Discovery3003 Pharmaceutical Science; 3003Amino Acid MotifsClinical BiochemistryGene ExpressionPharmaceutical Science01 natural sciencesClinical biochemistryBiochemistry[ CHIM ] Chemical SciencesProtein Structure Secondary[ SDV.CAN ] Life Sciences [q-bio]/Cancerchemistry.chemical_compoundLow affinityDrug DiscoveryEnzyme Inhibitors23-Dihydrobenzofuran privileged structure; Molecular docking; mPGES-1 inhibitors; Cancer; InflammationProstaglandin-E SynthasesCancerAnti-Inflammatory Agents Non-SteroidalBiological activityProto-Oncogene Proteins c-metIntramolecular OxidoreductasesMolecular Docking SimulationMolecular dockingMolecular Medicinelipids (amino acids peptides and proteins)Cell SurvivalStereochemistryMolecular Sequence Data2Antineoplastic Agents[SDV.CAN]Life Sciences [q-bio]/Cancer3-Dihydrobenzofuran privileged structureInhibitory Concentration 50Structure-Activity Relationship03 medical and health sciencesCell Line TumorMicrosomesHumans[CHIM]Chemical SciencesMolecular BiologyBenzofuransInflammationNatural product010405 organic chemistryDrug Discovery3003 Pharmaceutical ScienceOrganic ChemistryEpithelial CellsmPGES-1 inhibitorsCombinatorial chemistryCombined approach0104 chemical sciences030104 developmental biologychemistryDrug DesignDrug Screening Assays Antitumor
researchProduct

Cytotoxic effects induced by patulin, deoxynivalenol and toxin T2 individually and in combination in hepatic cells (HepG2).

2018

Abstract Patulin (PAT), deoxynivalenol (DON) and toxin T-2 (T-2) are mycotoxins distributed worldwide in food and feed. Cytotoxicity of the three mycotoxins individually or in combination in human hepatocellular carcinoma (HepG2) cells was evaluated by MTT assay over 24, 48 and 72 h of exposure. The concentration ranges used were 0.625–15 μM for DON, 1.25–50 nM for T-2 and 0.45–7.5 μM for PAT. The IC 50 values obtained ranged from 9.30 to 2.53 μM, from 33.69 to 44.37 nM and from 2.66 to 1.17 μM for DON, T-2 and PAT, respectively. The most cytotoxic mycotoxin to HepG2 cells was T-2 followed by PAT and DON. The combination ratios used for the mixtures were 1:3 (DON: T-2), 1:5 (DON: PAT), 1:1.…

0301 basic medicineCell SurvivalComplex MixturesToxicologymedicine.disease_causePatulin03 medical and health scienceschemistry.chemical_compoundInhibitory Concentration 500404 agricultural biotechnologymedicineCytotoxic T cellHumansMTT assayDrug InteractionsCytotoxicityMycotoxinDose-Response Relationship DrugToxin04 agricultural and veterinary sciencesGeneral MedicineHep G2 CellsMycotoxinsmedicine.disease040401 food scienceMolecular biologyDrug CombinationsT-2 Toxin030104 developmental biologyPatulinchemistryLiverHepatocellular carcinomaHepatic stellate cellTrichothecenesFood ScienceFood and chemical toxicology : an international journal published for the British Industrial Biological Research Association
researchProduct

Chemical Composition, In Vitro Antitumor and Pro-Oxidant Activities of Glandora rosmarinifolia (Boraginaceae) Essential Oil

2018

The biological properties of essential oils have been demonstrated in the treatment of several diseases and to enhance the bioavailability of other drugs. In natural habitats the essential oils compounds may play important roles in the protection of the plants as antibacterials, antivirals, antifungals, insecticides and also against herbivores by reducing their appetite for such plants or by repelling undesirable others. We analyzed by gas-chromatography mass spectrometry the chemical composition of the essential oil of aerial parts of Glandora rosmarinifolia (Ten.) D.C. Thomas obtained by hydrodistillation and verified some biological activities on a panel of hepatocellular carcinoma cell …

0301 basic medicineChemical RadicalsAntioxidantmedicine.medical_treatmentMDA-MB-231Cancer Treatmentlcsh:MedicinenaphthoquinoneChemical CompositionBiochemistryPhysical ChemistryditerpeneAntioxidantslaw.invention0302 clinical medicinelawBreast TumorsSUM 149Medicine and Health SciencesBioassaySettore BIO/15 - Biologia FarmaceuticaCytotoxicitylcsh:ScienceMultidisciplinarybiologyTraditional medicineChemistryLiver DiseasesBoraginaceaeBoraginaceaeOxidantsHep3BLipidsChemistryOncology030220 oncology & carcinogenesisPhysical SciencesResearch ArticleHepG2Free RadicalsCell SurvivalGastroenterology and HepatologyCarcinomas03 medical and health sciencesInhibitory Concentration 50Cell Line TumorAromatic HydrocarbonsGastrointestinal TumorsBreast CancermedicineOils VolatileHumansPlant OilsEssential oilcytotoxic activityHA22T/VGH; HepG2; Hep3B; SUM 149; MDA-MB-231; cytotoxic activity; diterpenes; naphthoquinones; plant secondary metabolitesVolatile Organic CompoundsDose-Response Relationship DrugCell growthPlant ExtractsHA22T/VGHlcsh:RChemical CompoundsBiology and Life SciencesCancers and NeoplasmsEpithelial CellsHepatocellular CarcinomaSettore CHIM/06 - Chimica OrganicaPlant Components Aerialbiology.organism_classificationPro-oxidantplant secondary metabolitesAntineoplastic Agents PhytogenicHydrocarbonsBioavailability030104 developmental biologySettore BIO/03 - Botanica Ambientale E ApplicataHepatocytesSettore BIO/14 - Farmacologialcsh:QOils
researchProduct