Search results for " Farm"

showing 10 items of 2009 documents

Inhalable Formulation Based on Lipid–Polymer Hybrid Nanoparticles for the Macrophage Targeted Delivery of Roflumilast

2022

Here, novel lipid-polymer hybrid nanoparticles (LPHNPs), targeted to lung macrophages, were realized as potential carriers for Roflumilast administration in the management of chronic obstructive pulmonary disease (COPD). To achieve this, Roflumilast-loaded fluorescent polymeric nanoparticles, based on a polyaspartamide-polycaprolactone graft copolymer, and lipid vesicles, made from 1,2-dipalmitoyl-sn-glycero-3-phosphocholine and 1,2-distearoyl-sn-glycero-phosphoethanolamine-N-(polyethylene glycol)-mannose, were properly combined using a two-step method, successfully obtaining Roflumilast-loaded hybrid fluorescent nanoparticles (Man-LPHFNPs@Roflumilast). These exhibit colloidal size and a ne…

CyclopropanesPolymers and PlasticsPolymersMacrophagesPhosphatidylethanolaminesAminopyridinesBioengineeringPolyethylene GlycolsBiomaterialsSettore CHIM/09 - Farmaceutico Tecnologico ApplicativoBenzamidesMaterials ChemistryHumansNanoparticlesParticle SizeMannoseBiomacromolecules
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Inhalable nano into micro dry powders for ivacaftor delivery: The role of mannitol and cysteamine as mucus-active agents.

2020

In this paper the innovative approach of Nano into micro (NiM9 was developed to produce Nanoparticles loaded Ivacaftor to incorporate into mannitol or mannitol/cysteamine micromatrices for drug pulmonary administration in CF. Nanoparticles composed by a mixture of two polyhydrohydroxyethtylaspartamide copolymers containing a loading of Ivacaftor of 15.5 % w/w were produced. These Nanoparticles were incorporated into microparticles to obtain NiM that were characterized in terms of size and size distribution, interaction with CF-AM by rheological and turbidimetric studies as well as by aerodynamic diameter measurements. Finally the activity of Ivacaftor into these NiM was evaluated by in vitr…

Cystic Fibrosisαβ-poly-(N-2-hydroxyethyl)-DL-aspartamide (PHEA) copolymer PHEA ivacaftor mucus-penetrating nanoparticle cell penetrating peptide nano into micro strategy. CysteamineDrug CompoundingPharmaceutical ScienceNanoparticleCystic Fibrosis Transmembrane Conductance Regulator02 engineering and technologyQuinolonesAminophenols030226 pharmacology & pharmacyIvacaftor03 medical and health scienceschemistry.chemical_compound0302 clinical medicineNano-Administration InhalationMucus-penetrating nanoparticlemedicineCopolymerAnimalsMannitolChloride Channel AgonistsCells CulturedExpectorantsCell penetrating peptideNano into micro strategyChemistry021001 nanoscience & nanotechnologyMucusRats Inbred F344IvacaftorCopolymer PHEADrug LiberationSettore CHIM/09 - Farmaceutico Tecnologico ApplicativoMutationNanoparticlesCysteamineMannitolPowders0210 nano-technologyPeptidesαβ-poly-(N-2-hydroxyethyl)-DL-aspartamide (PHEA)medicine.drugNuclear chemistryInternational journal of pharmaceutics
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HETEROCYCLIC COMPOUNDS AND MEDICAL USE THEREOF

2019

The present invention relates to heterocyclic nitrogen compounds, use thereof as a medicament and pharmaceutical compositions thereof. Furthermore, the invention provides combinations of compounds of general formula (I) with therapeutic agents, such as correctors, potentiators and amplifiers of dysfunctional proteins.

Cystic fibrosiCFTR correctorCystic fibrosis transmembrane conductance regulatorCFTRSettore CHIM/08 - Chimica FarmaceuticaF508del-CFTR
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Using Y-chromosome capture enrichment to resolve haplogroup H2 shows new evidence for a two-path Neolithic expansion to Western Europe

2021

Uniparentally-inherited markers on mitochondrial DNA (mtDNA) and the non-recombining regions of the Y chromosome (NRY), have been used for the past 30 years to investigate the history of humans from a maternal and paternal perspective. Researchers have preferred mtDNA due to its abundance in the cells, and comparatively high substitution rate. Conversely, the NRY is less susceptible to back mutations and saturation, and is potentially more informative than mtDNA owing to its longer sequence length. However, due to comparatively poor NRY coverage via shotgun sequencing, and the relatively low and biased representation of Y-chromosome variants on capture assays such as the 1240 k, ancient DNA…

CzechSELECTIONPopulation geneticsMITOCHONDRIAL-DNAearly farmersDIVERSITYmitochondrial DNAshotgun sequencingPrehistòriaHaplogroupGerman0302 clinical medicineMedicine and Health SciencesDNA sequencingScience and technologymedia_common0303 health sciencesMultidisciplinaryHorizon (archaeology)Critical eventShotgun sequencingchromosomal haplogroupsEuropean researchQRSTEPPEWestern europelanguageMedicineGenetic MarkersMitochondrial DNA[SHS.ARCHEO]Humanities and Social Sciences/Archaeology and Prehistoryuniparentally-inherited markersScienceLibrary scienceBiologyY chromosomeDNA MitochondrialPolymorphism Single NucleotideTarget enrichmentArticle03 medical and health sciencesPolitical scienceHumansmedia_common.cataloged_instanceANCIENT DNAGenetic TestingEuropean unionAlleles030304 developmental biologyMUTATION-RATEChromosomes Human YY chromosomeSaturation (genetic)History and ArchaeologyY-mappable capture assayAncient DNA; Neanderthals; Anatomically modern humanslanguage.human_languageNeolithic transitionGenetics PopulationAncient DNAHaplotypesEvolutionary biologyGENOMIC HISTORY030217 neurology & neurosurgery
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Resistencia frente a la infección por Penicillium digitatum durante la postcosecha de los frutos cítricos. Bases moleculares y metabolismo de fenilpr…

2007

Tesis Doctoral. Facultad de Farmacia, Universidad de Valencia y Grupo de Postcosecha, Instituto de Agroquímica y Tecnología de Alimentos (CSIC)

Cítricosnone632FenilpropanoidesF. FarmaciaPenicillium digitatumPodredumbre de los cítricos
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PHARMACOLOGICAL MODULATION OF OPERANT BEHAVIOUR FOR ACETALDEHYDE. INVOLVEMENT OF D2 AND CB1 RECEPTORS.

2013

Acetaldehyde (ACD), the first metabolite of ethanol, has rewarding and motivational properties, as shown by behavioural studies specifically tailored for studying addictive-like behaviour (1, 2). The rewarding and incentive effects of alcohol and others addictive substances, result from their capability to enhance mesolimbic dopamine (DA) transmission, as well as to affect the cannabinoid system, which is able to fine-tune the activity of DA neurons (3). ACD directly increases DA neurotransmission (4), but the neural underpinning the operant behaviour for oral-self administered ACD still remains poorly understood. Since D2 and CB1 receptors are involved in alcohol addiction (3), as well as …

D2-receptorSettore BIO/14 - FarmacologiaAcetaldehydeCB1-receptorsoperant self-administration
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Virulence and Molecular Typing of Vibrio harveyi Strains Isolated from Cultured Dentex, Gilthead Sea Bream and European Sea Bass

2003

Vibrio harveyi was isolated from internal organs or ulcers of diseased and apparently healthy gilthead sea bream (Sparus aurata) and European sea bass (Dicentrarchus labrax) cultured in several fish farms located on the Spanish Mediterranean coast. The prevalence of the bacterium was significantly higher in European sea bass than in gilthead sea bream, and was closely related to the season in both fish species, occurring almost exclusively on warm months (June to November). After phenotypic characterization, a selection of forty five isolates from gilthead sea bream, sea bass, and several isolates previously obtained from common dentex (Dentex dentex) of the same area, were molecularly type…

DNA BacterialFish farmingFisheriesVirulenceZoologyMediterranean aquacultureRibotypingApplied Microbiology and BiotechnologyMicrobiologyFish DiseasesRibotypingRAPDSparus aurataAnimalsDicentrarchus labraxSea bassFish pathogensEcology Evolution Behavior and SystematicsVibrioVirulencebiologyVibrio harveyiLD50Dentex dentexbiology.organism_classificationVibrio harveyiSea BreamBacterial Typing TechniquesPerciformesRandom Amplified Polymorphic DNA TechniqueRAPDFisheryPhenotypeVibrio InfectionsCarrier StateBassDicentrarchussense organsDentex dentexSystematic and Applied Microbiology
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Assessment of Salmonella spp. in feces, cloacal swabs, and eggs (eggshell and content separately) from a laying hen farm.

2011

Microbial pathogens of the genus Salmonella are among the leading causes of foodborne illness in the world. The present study was done on a laying hen farm with a Salmonella enterica serovar Enteritidis-positive result according to the testing specified by European regulation 2160/2003. The aim of this study was to compare the Salmonella contamination on a laying hen farm with the Salmonella presence in the hen eggs. The strains were isolated by ISO method 6579:2002 (standard method for the detection of Salmonella spp. in the European regulation for food and animal feeding stuffs, animal feces, and environmental samples from the primary production stage, including poultry farms) and were co…

DNA BacterialVeterinary medicineSalmonellaSalmonella enteritidisEggsmedicine.disease_causeEgg ShellFecesAnimal scienceCloacamedicinemedia_common.cataloged_instanceFood microbiologyAnimalsEuropean UnionEuropean unionEggshellDeoxyribonucleases Type II Site-SpecificFecesPoultry Diseasesmedia_commonSalmonella Infections AnimalChi-Square Distributionbiologybusiness.industryGeneral MedicinePoultry farmingbiology.organism_classificationElectrophoresis Gel Pulsed-FieldSalmonella enteritidisSalmonella entericaFood MicrobiologyAnimal Science and ZoologyFemalebusinessChickensPoultry science
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Transition Metal Complexes as DNA-intercalators

2008

DNA Intercalators metal complex oxadiazoleSettore CHIM/03 - Chimica Generale E InorganicaSettore CHIM/08 - Chimica Farmaceutica
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DNA Binding and Biological Activity of Transition Metal Complexes

2011

DNA Transition Metal complexesSettore CHIM/03 - Chimica Generale E InorganicaSettore CHIM/08 - Chimica Farmaceutica
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