Search results for " P.A.E.S."

showing 10 items of 309 documents

PEG 400/Cerium Ammonium Nitrate Combined with Microwave-Assisted Synthesis for Rapid Access to Beta-Amino Ketones. An Easy-to-Use Protocol for Discov…

2018

Compound libraries are important requirement in target-based drug discovery. In the present work, a small focused compound library based on β-aminoketone scaffold has been prepared combining microwave-assisted organic synthesis (MAOS) with polymer-assisted solution phase synthesis (PASPS) and replacing reaction workup standard purification procedures with solid phase extraction (SPE). Specifically, the effects of solvent, such as dioxane, dimethylformamide (DMF), polyethylene glycol 400 (PEG 400), temperature, irradiation time, stoichiometric ratio of reagents, and catalysts (HCl, acetic acid, cerium ammonium nitrate (CAN)) were investigated to maximize both conversion and yield. The optimi…

3003Transcription FactorPharmaceutical ScienceNitratePolyethylene Glycol01 natural sciencesPolyethylene GlycolsPolymer-assisted solution phase synthesiAnalytical Chemistrychemistry.chemical_compoundDrug DiscoveryMannich reactionSolid phase extractionMicrowavesβ-aminoketonesCeriumKetonesKetoneDNA-Binding ProteinsSolventCeriumChemistry (miscellaneous)Molecular MedicineDimethylformamideMicrowave-assisted organic synthesiMannich reaction; β-aminoketones; microwave-assisted organic synthesis; polymer-assisted solution phase synthesis; solid phase extraction; drug discoveryDNA-Binding ProteinBacterial Proteinchemistry.chemical_elementPolyethylene glycol010402 general chemistryArticlelcsh:QD241-441Bacterial Proteinslcsh:Organic chemistryΒ-aminoketonePhysical and Theoretical ChemistrySolid phase extractionpolymer-assisted solution phase synthesisPEG 400Nitrates010405 organic chemistryDrug Discovery3003 Pharmaceutical ScienceOrganic ChemistrySettore CHIM/08 - Chimica FarmaceuticaCombinatorial chemistry0104 chemical scienceschemistryYield (chemistry)microwave-assisted organic synthesisOrganic synthesisMicrowaveTranscription FactorsMolecules
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PLLA scaffolds with controlled architecture as potential microenvironment for in vitro tumor model

2019

Abstract The "microenvironment" where a tumor develops plays a fundamental role in determining its progression, the onset of metastasis and, eventually, its resistance to therapies. Tumor cells can be considered more or less invasive depending both on the nature of the cells and on the site where they are located. Commonly adopted laboratory culture protocols for the investigation of tumor cells take usually place on standard two-dimensional supports. However, such cultures do not allow for reproduction of the biophysical properties of the tumor’s microenvironment, thus causing the cells to lose most of their relevant characteristics. In this work MDA-MB 231 breast cancer cells were cultiva…

3D tumor modelPolyestersCellBreast Neoplasms02 engineering and technologyBiologyModels BiologicalMetastasis03 medical and health scienceschemistry.chemical_compoundCell Line TumorTumor MicroenvironmentmedicineHumansViability assayDAPICell adhesion030304 developmental biologySettore ING-IND/24 - Principi Di Ingegneria Chimica0303 health sciencesTissue ScaffoldsSettore ING-IND/34 - Bioingegneria IndustrialeBreast cancer cellCell BiologyGeneral Medicine021001 nanoscience & nanotechnologymedicine.diseaseIn vitroLactic acidStainingmedicine.anatomical_structurechemistryBiophysicsFemaleThermally induced phase separation0210 nano-technologyPoly-L-Lactic acidDevelopmental BiologyTissue and Cell
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Specific muscle-tendon architecture in elite Kenyan distance runners

2013

The Achilles tendon moment arm (MA_AT) and foot lever ratio (FLR) can play important roles for force production and movement economy during locomotion. This notion has become more relevant, and suggestion has been given that the Kenyan runners belonging to the world elite would have specific anatomical, mechanical, and functional properties in their lower limbs and that this feature could be responsible for their high running economy. The present study aimed to characterize the AT of elite Kenyan distance runners as compared with Japanese ones, and to examine the potential relationship with their running performance. Ultrasonography was used to measure AT cross-sectional area and AT soleus …

Achilles tendonLevermedicine.medical_specialtybusiness.product_categorybusiness.industryPhysical Therapy Sports Therapy and RehabilitationBiologySagittal planeStretch shortening cycleTendonmedicine.anatomical_structurePhysical medicine and rehabilitationElitemedicineRunning economyOrthopedics and Sports MedicineUltrasonographybusinessScandinavian Journal of Medicine & Science in Sports
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Análisis de la distancia recorrida en pádel en función del nivel de juego y el número de puntos por partido (Analysis of distance covered in padel ba…

2020

La distancia que recorren los jugadores por partido supone una forma de cuantificar el volumen de carga externa del juego, y su estudio tiene una gran aplicación en la planificación del entrenamiento deportivo. El objetivo de este estudio fue analizar la distancia recorrida en diferentes fases del partido (activa y pasiva) y su relación con el número de puntos disputados y nivel de juego de los deportistas. La muestra estuvo compuesta por 108 jugadores federados de pádel (edad media = 33.81 ± 6.72 años). Se analizaron, a través de observación sistemática con el sistema SAGIT, un total 4406 puntos correspondientes a 27 partidos de pádel. Los partidos fueron divididos en tres niveles de compe…

Active phaseStatisticsOrthopedics and Sports MedicinePhysical Therapy Sports Therapy and RehabilitationRest timeEducationNumero signMathematicsRetos
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Association between condylar asymmetry and temporo- mandibular disorders using 3D-CT

2011

Objectives: Using reconstructed three-dimensional computed tomography (3D-CT) models, the purpose of this study was to analyze and compare mandibular condyle morphology in patients with and without temporomandibular disorder (TMD). Study Design: Thirty-two patients were divided into two groups: the first comprised those with TMD (n=18), and the second those who did not have TMD (n=14). A CT of each patient was obtained and reconstructed as a 3D model. The 64 resulting 3D condylar models were evaluated for possible TMD-associated length, width and height asymmetries of the condylar process. Descriptive statistics were used to assess the results and student’s t tests applied to compare the tw…

Adult3D-computed tomographyCondilar asymmetryMandibular DisordersDentistryMaxillofacial surgeryComputed tomography3d modelOrthodonticsCondyleImaging Three-Dimensionalstomatognathic systemX ray computedClinical and Experimental DentistrymedicineHumansIn patientGeneral DentistryOrthodonticsmedicine.diagnostic_testbusiness.industryTemporomandibular disorderMandibular CondyleTemporomandibular Joint Disorders:CIENCIAS MÉDICAS [UNESCO]Sagittal planestomatognathic diseasesmedicine.anatomical_structureOtorhinolaryngologyUNESCO::CIENCIAS MÉDICASSurgeryResearch-ArticlebusinessTomography X-Ray ComputedX-ray diagnosishuman activities
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Influence of the structural components of artificial turf systems on impact attenuation in amateur football players

2019

AbstractThe purpose of this research was to evaluate the influence of the structural components of different 3rd generation artificial turf football field systems on the biomechanical response of impact attenuation in amateur football players. A total of 12 amateur football players (24.3 ± 3.7 years, 73.5 ± 5.5 kg, 178.3 ± 4.1 cm and 13.7 ± 4.3 years of sport experience) were evaluated on three third generation artificial turf systems (ATS) with different structural components. ATS were composed of asphalt sub-base and 45 mm of fibre height with (ATS1) and without (ATS2) elastic layer or compacted granular sub-base, 60 mm of fibre height without elastic layer (ATS3). Two triaxial accelerome…

AdultMale0301 basic medicineAccelerationPoison controlSTRIDElcsh:MedicineFútbolArticleLower energyRunningYoung Adult03 medical and health sciences0302 clinical medicineFloors and FloorcoveringsSoccerArtificial turfHumanslcsh:ScienceMathematicsOrthodonticsEsportsFootball playersMultidisciplinaryAttenuationlcsh:RDeporteBone quality and biomechanicsBiomechanical Phenomena030104 developmental biologyRisk factorsAthletesFootball fieldSuperficies deportivas sintéticaslcsh:QEducació físicaAmateur030217 neurology & neurosurgeryInstalación deportiva
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Upper incisor to Soft Tissue Plane (UI-STP) : a new reference for diagnosis and planning in dentofacial deformities

2009

Planning in orthognathic surgery has been and still is an open issue. We have evolved from 2D classical cephalometric hard-tissue planning to 2D soft tissue planning, and finally to 3D and hard and soft tissue evaluation. This, to our knowledge, is the first description of a new Soft Tissue Plane (STP) and its relationship with the anterior position of the upper incisor (UI). Profile photographs of 110 ?attractive individuals? with lips at rest or smiling and with upper incisor shown were used. The photographs used were of 65 professional models from two international agencies and 45 individuals considered most attractive in the internet forums, which included catwalk models and actors. In …

AdultMaleCephalometrymedicine.medical_treatmentOrthognathic surgeryDentistryDentofacial DeformityYoung AdultIncisorReference ValuesMaxillaHumansMedicineAbnormalities MultipleGeneral DentistryOrthodonticsTooth Abnormalitiesbusiness.industrySoft tissue planeSoft tissueMiddle AgedCraniometry:CIENCIAS MÉDICAS [UNESCO]Incisormedicine.anatomical_structureOtorhinolaryngologyFaceMaxillaReference valuesUNESCO::CIENCIAS MÉDICASFemaleSurgerybusiness
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Visuospatial attention lateralization in volleyball players and in rowers.

2011

In the present study, differences in visuospatial attention lateralization were evaluated in athletes engaged in open- compared to closed-skill sports and sedentary nonathletes. 23 volleyball players (open skill; Italian national level and regional level), 10 rowers (closed skill, Italian national level), and 23 sedentary participants responded to a computerized line-length judgment task. Five lines, differing in the length of their right and left segments, were randomly presented; the respondent made a forced-choice decision about the respective length of the two segments. Volleyball players responded significantly faster; those at the higher competitive level were also more accurate, mak…

AdultMalemedicine.medical_specialtyExperimental and Cognitive PsychologyAthletic PerformanceAudiologyChoice BehaviorFunctional LateralityLateralization of brain functionJudgmentYoung AdultOrientationReaction TimemedicineHumansAttentionNational levelSize PerceptionbiologyAthletesvisuospatial attention volley ball players rowersbiology.organism_classificationSensory SystemsVolleyballPattern Recognition VisualSpace PerceptionRespondentPhysical therapyPsychologySports
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VO2max Characteristics of Elite Female Soccer Players, 1989–2007

2013

Purpose:To quantify VO2max among female competitive soccer players as a function of performance level, field position, and age. In addition, the evolution of VO2max among world-class players over an 18-y period was quantified.Methods:Female players (N = 199, 22 ± 4 y, 63 ± 6 kg, height 169 ± 6 cm), including an Olympic winning squad, were tested for VO2max at the Norwegian Olympic Training Center between 1989 and 2007.Results:National-team players had 5% higher VO2max than 1st-division players (P = .042, d = 0.4), 13% higher than 2nd-division players (P < .001, d = 1.2), and 9% higher than junior players (P = .005, d = 1.0). Midfielders had 8% higher VO2max than goalkeepers (P = .048, d …

Adultmaximum oxygen uptakeCompetitive Behaviormedicine.medical_specialtyTime FactorsAdolescentAge categoriesPhysical Therapy Sports Therapy and RehabilitationAthletic PerformanceRunningYoung AdultOxygen ConsumptionSoccerHumansMedicineOrthopedics and Sports Medicinephysical demandsPhysical conditioningNorwaybusiness.industryAge FactorsVO2 maxphysical performancenational team soccer playersaerobic capacityTraining centerMotor SkillsCompetitive behaviorPhysical performanceEliteExercise TestPhysical therapyFemaleVDP::Medical disciplines: 700::Sports medicine: 850businessPhysical Conditioning HumanDemographyInternational Journal of Sports Physiology and Performance
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Practice and play in the development of German top-level professional football players.

2014

This study examined the developmental sporting activities of 52 German football first Bundesliga professionals (including 18 senior national team members) and 50 fourth to sixth league amateur players. They reported their volumes of organised football practice/training, including its "microstructure" (proportions of physical conditioning, skill exercises and playing forms), non-organised leisure football play and engagement in other sports through their career, respectively. Analyses revealed that the Bundesliga professionals performed moderate amounts of organised football practice/training throughout their career. They accumulated 4264 (mean value) hours over ~16 years before debuting in …

Adultmedicine.medical_specialtyeducationPhysical Therapy Sports Therapy and RehabilitationFootballLeagueAthletic PerformanceGerman03 medical and health sciencesYoung Adult0302 clinical medicineGermany0502 economics and businessSoccermedicineHumansOrthopedics and Sports MedicineExerciseMedical educationFootball playersPhysical conditioning05 social sciencesMean value030229 sport sciencesGeneral Medicinelanguage.human_languageTalent developmentAthleteslanguagePhysical therapyPsychologyAmateur050212 sport leisure & tourismEuropean journal of sport science
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