Search results for " Sor"

showing 10 items of 408 documents

1,2,4-Oxadiazole topsentin analogs as staphylococcal biofilm inhibitors targeting the bacterial transpeptidase sortase A

2020

The inhibition or prevention of biofilm formation represents an emerging strategy in the war against antibiotic resistance, interfering with key players in bacterial virulence. This approach includes the inhibition of the catalytic activity of transpeptidase sortase A (Srt A), a membrane enzyme responsible for covalently attaching a wide variety of adhesive matrix molecules to the peptidoglycan cell wall in Gram-positive strains. A new series of seventeen 1,2,4-oxadiazole derivatives was efficiently synthesized and screened as potential new anti-virulence agents. The ability of inhibiting biofilm formation was evaluated against both Gram-positive and Gram-negative pathogens. Remarkably, all…

Indoles124-Oxadiazoles Antibiofilm activity Sortase A inhibitors Anti-virulence agents Marine alkaloids Topsentin analogs01 natural scienceslaw.inventionchemistry.chemical_compoundMarine alkaloidslawDrug DiscoveryPathogenchemistry.chemical_classificationOxadiazoles0303 health sciencesChemistry4-OxadiazolesImidazolesGeneral MedicineStaphylococcal InfectionsAminoacyltransferasesAnti-Bacterial AgentsCysteine EndopeptidasesAnti-virulence agentsBiochemistrySortase AAntibiofilm activityPseudomonas aeruginosaTopsentin analogsRecombinant DNA124-Oxadiazoles; Anti-virulence agents; Antibiofilm activity; Marine alkaloids; Sortase A inhibitors; Topsentin analogsStaphylococcus aureus12Sortase A inhibitorsCell LineCell wall03 medical and health sciencesAntibiotic resistanceBacterial Proteins124-OxadiazolesHumansPseudomonas Infections030304 developmental biologyPharmacology010405 organic chemistryOrganic ChemistryBiofilmSettore CHIM/08 - Chimica Farmaceutica0104 chemical sciencesEnzymeBiofilmsPeptidoglycan
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Nota a 1) Cass. 23 gennaio 2012, n.11621; 2) Cass. 16 dicembre 2011, n. 9907; 3)Cass. 5 dicembre 2011, n. 15026.

2013

Nota a tre sentenze della Cassazione in materia di ingiuria e minacce. Più in particolare, sub 1) rilevanza penale dell'espressione "lei non sa chi sono io"; sub 2) presupposti e limiti dell'esimente della provocazione; sub 3) rilevanza dell'ingiuria da parte del soggetto sordomuto.

Ingiuria - Minacce - "Lei non sa chi sono io" - Provocazione - Soggetto sordomuto.Settore IUS/17 - Diritto Penale
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Chiral Self‐Sorting of trans ‐Chelating Chiral Ligands upon Formation of Pd II Complexes (Eur. J. Inorg. Chem. 15/2014)

2014

Inorganic ChemistrySelf sortingchemistryStereochemistryPolymer chemistrySupramolecular chemistrychemistry.chemical_elementChelationSelf-assemblyPlanar chiralityPalladiumEuropean Journal of Inorganic Chemistry
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Chiral Self-Sorting of trans-Chelating Chiral Ligands upon Formation of PdII Complexes

2014

Invited for the cover of this issue is the group of Arne Lutzen at the University of Bonn, Germany. The cover image shows two dissymmetric bis(3-pyridyl) ligands based on a planar chiral pseudo-ortho-disubstituted [2.2]paracyclophane scaffold. Upon forming a mononuclear [ML2] complex with palladium(II) ions, these ligands act in a trans-chelating manner and undergo complete chiral self-sorting.

Inorganic ChemistrySelf sortingchemistryStereochemistrySupramolecular chemistrychemistry.chemical_elementChelationSelf-assemblyta116PalladiumEuropean Journal of Inorganic Chemistry
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Cholesterol Dependence of Collagen and Echovirus 1 Trafficking along the Novel α2β1 Integrin Internalization Pathway

2013

We have previously shown that soluble collagen and a human pathogen, echovirus 1 (EV1) cluster α2β1 integrin on the plasma membrane and cause their internalization into cytoplasmic endosomes. Here we show that cholesterol plays a major role not only in the uptake of α2β1 integrin and its ligands but also in the formation of α2 integrin-specific multivesicular bodies (α2-MVBs) and virus infection. EV1 infection and α2β1 integrin internalization were totally halted by low amounts of the cholesterol-aggregating drugs filipin or nystatin. Inhibition of cholesterol synthesis and accumulation of lanosterol after ketoconazole treatment inhibited uptake of collagen, virus and clustered integrin, an…

IntegrinsNystatinFluorescent Antibody TechniqueBiochemistryCollagen receptorchemistry.chemical_compoundBINDINGMolecular Cell BiologyInternalizationLipid raftREQUIRESmedia_common0303 health sciencesMicroscopy ConfocalMultidisciplinarybiologyQRIMMUNODEFICIENCY-VIRUS TYPE-1RNA REPLICATIONCellular StructuresExtracellular MatrixEnterovirus B Human3. Good healthCell biologyProtein TransportCholesterolENTRYCytochemistryMedicineMembranes and Sortinglipids (amino acids peptides and proteins)CollagenIntegrin alpha2beta1Research ArticleSignal TransductionViral EntryEndosomeSciencemedia_common.quotation_subjecteducationIntegrinLOW-DENSITY-LIPOPROTEINMicrobiologyFilipinClathrinGPI-ANCHORED PROTEINS03 medical and health sciencesVirologyCell Line TumorCell AdhesionHumansFilipinBiology030304 developmental biology030306 microbiologyCell MembraneVirus Uncoatingta1182TRANSPORTLIPID RAFTSMicroscopy ElectronSubcellular Organelleschemistrybiology.protein3111 BiomedicineChromatography Thin LayerCELL-MEMBRANESViral Transmission and InfectionPLoS ONE
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UN IRRADIATORE NEUTRONICO MODULARE CON SORGENTI DI 241Am-Be PER IL TEST DI DOSIMETRI NEUTRONICI PERSONALI

2010

Irradiatori neutronici basati su sorgenti radionuclidiche sono impiegati in diversi paesi per l’analisi per attivazione di vari campioni, per studiare le caratteristiche dei materiali sottoposti a irradiazione, ma anche per studiare la risposta di rivelatori e/o dosimetri personali sensibili alla componente neutronica. Per quest’ultima applicazione, l’uso di un irradiatore con sorgenti risulta molto vantaggioso per la stabilità nel tempo del flusso neutronico, mentre è relativamente poco importante il valore assoluto del flusso neutronico, di qualche ordine di grandezza inferiore a quello di reattori o di acceleratori di particelle. Per l’effettuazione di test su rivelatori e/o dosimetri pe…

Irradiatore neutronico sorgenti Am-Be Dosimetri neutroniciSettore ING-IND/20 - Misure E Strumentazione Nucleari
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José Capuz Mamano (1884-1964), maestro de Helena Sorolla García (1895-1975)

2014

Isabel 253 265UNESCO::CIENCIAS DE LAS ARTES Y LAS LETRAS0211-5808 9678 Archivo de arte valenciano 385455 2014 95 4940223 José Capuz Mamano (1884-1964):CIENCIAS DE LAS ARTES Y LAS LETRAS [UNESCO]maestro de Helena Sorolla García (1895-1975) Justo
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The comparison of seven different methods to quantify the amorphous content of spray dried lactose

2006

The purpose of this work was to verify the usefulness, advantages and disadvantages of seven methods that are widely used to detect, and quantify the amorphous contents in pharmaceutical solids. Here, StepScan DSC, a type of modulated temperature calorimetry method, was applied for the first time to quantify amorphicity. The comparison of the analytical methods was undertaken with real (non-artificial) test samples, i.e. spray-dried lactose samples with various degrees of crystallinity. In these samples, it was essential that the amorphous and the crystalline portions are not present as separate particles, which is the case when physical (artificial) mixtures of totally amorphous and totall…

Isothermal microcalorimetryRecrystallization (geology)Chemistryrecrystallizationspectroscopic methodsGeneral Chemical Engineeringx-ray powder diffractionAnalytical chemistryCalorimetrycalorimetric methodsAmorphous solidlactosemoisture sorptionCrystallinityDifferential scanning calorimetryGravimetric analysisamorphicitypharmaceutical compoundsGlass transitionPowder Technology
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Responses of Prunus ferganensis, Prunus persica and two interspecific hybrids to moderate drought stress

2003

Prunus ferganensis (Kost. & Riab) Kov. & Kost, a close relative of the cultivated peach (Prunus persica (L.) Batsch.), is native to arid regions of central Asia and may possess traits valuable for improving drought tolerance of commercial peach varieties. One distinguishing feature of P. ferganensis is its prominent, elongated, unbranched leaf venation pattern, which behaves as a simple recessive trait in segregating populations of P. ferganensis x P. persica hybrids. To understand whether this trait could be used as a marker in breeding for drought tolerance, we investigated the association between leaf morphological and physiological parameters related to drought response in P. ferganensi…

L-Iditol 2-DehydrogenaseSpecific leaf areaPhysiologyClimatic adaptationDrought tolerancePlant ScienceBiologyTreesPrunusDry weightSorbitolLeaf sizePhotosynthesisgas exchange non-hydraulic signals peach photosynthesis sorbitol water potentialHybridDehydrationfungiWaterfood and beveragesPlant TranspirationPlant LeavesSettore AGR/03 - Arboricoltura Generale E Coltivazioni ArboreeAgronomyPrunusRootstockSugar Alcohol DehydrogenasesTree Physiology
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Segnare, parlare, intendersi: modalità e forme

2012

LINGUE DEI SEGNI LINGUE VERBALI PEDAGOGIA LINGUISTICA GESTI E SEGNI SCRITTURA IN SEGNI CULTURA SORDA IDENTITA' E DIFFERENZE INTERCULTURA FORMAZIONE SCUOLA ASSISTENTI ALLA COMUNICAZIONESettore M-PED/01 - Pedagogia Generale E Sociale
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