Search results for " solution"

showing 10 items of 3084 documents

MAST-RT0 solution of 3D Navier Stokes equations in very irregular domains. Preliminary results in the laminar case

2021

A new numerical methodology to solve the 3D Navier-Stokes equations for incompressible fluids within complex boundaries and unstructured body-fitted tetrahedral mesh is presented and validated with three literature and one real-case tests. We apply a fractional time step procedure where a predictor and a corrector problem are sequentially solved. The predictor step is solved applying the MAST (Marching in Space and Time) procedure, which explicitly handles the non-linear terms in the momentum equations, allowing numerical stability for Courant number greater than one. Correction steps are solved by a Mixed Hybrid Finite Elements discretization that assumes positive distances among tetrahedr…

A new numerical solver for the 3D Navier Stokes incompressible laminar problems is proposedThe proposed model is suitable for the solution of laminar flows in irregular domainsSettore ICAR/01 - Idraulica
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Polyoxypregnanes as safe, potent, and specific ABCB1-inhibitory pro-drugs to overcome multidrug resistance in cancer chemotherapy in vitro and in vivo

2021

Multidrug resistance (MDR) mediated by ATP binding cassette subfamily B member 1 (ABCB1) is significantly hindering effective cancer chemotherapy. However, currently, no ABCB1-inhibitory drugs have been approved to treat MDR cancer clinically, mainly due to the inhibitor specificity, toxicity, and drug interactions. Here, we reported that three polyoxypregnanes (POPs) as the most abundant constituents of Marsdenia tenacissima (M. tenacissima) were novel ABCB1-modulatory pro-drugs, which underwent intestinal microbiota-mediated biotransformation in vivo to generate active metabolites. The metabolites at non-toxic concentrations restored chemosensitivity in ABCB1-overexpressing cancer cells v…

ABCC1 ATP binding cassette subfamily C member 1IC50 half maximal inhibitory concentrationMultidrug resistancePharmacologyNADPH reduced nicotinamide adenine dinucleotide phosphateF bioavailabilitychemistry.chemical_compoundPCR polymerase chain reaction0302 clinical medicineMDR multidrug resistanceECL electrochemiluminescencet1/2 elimination half-lifeLC–MS liquid chromatography coupled with mass spectrometryN.D. not detectedGeneral Pharmacology Toxicology and PharmaceuticsBBB blood–brain barriermedia_commonATF3 activating transcription factor 30303 health sciencesChemistryABC ATP-binding cassetteNMPA National Medical Products AdministrationPXR pregnane X receptorSDS-PAGE sodium dodecyl sulfate-polyacrylamide gel electrophoresisHBSS Hankʹs balanced salt solutionABCB1Combination chemotherapyProdrugMarsdenia tenacissimaCmax peak concentrationPaclitaxelGAPDH glyceraldehyde-3-phosphate dehydrogenase030220 oncology & carcinogenesisBHI brain heart infusionOriginal ArticleAUC0–∞ area under plasma concentration vs. time curveMRT mean residence timeDrugmedia_common.quotation_subjectRM1-950Vd volume of distributionABCB1 ATP binding cassette subfamily B member 1UIC-2 mouse monoclonal ABCB1 antibodyABCG2 ATP binding cassette subfamily G member 2Combination chemotherapyCYP cytochrome P450 isozymePI propidium iodideTEER transepithelial electrical resistance03 medical and health sciencesPBS phosphate buffer salineFBS fetal bovine serumDox doxorubicinIn vivoPOP polyoxypregnanemedicine030304 developmental biologyEVOM epithelial tissue voltohmmeterTmax time for peak concentrationCancerLBE lowest binding energyPE phycoerythrinmedicine.diseaseMultiple drug resistancePolyoxypregnanePapp apparent permeabilityN.A. not applicableCancer cellH&E hematoxylin and eosinMDR1a multidrug resistance protein 1aTherapeutics. PharmacologyqPCR quantitative PCRM. tenacissima Marsdenia tenacissimaCL clearanceSD standard derivationActa Pharmaceutica Sinica B
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Isocratic and gradient elution in micellar liquid chromatography with Brij-35

2015

Polyoxyethylene(23)lauryl ether (known as Brij-35) is a nonionic surfactant, which has been considered as an alternative to the extensively used in micellar liquid chromatography anionic surfactant sodium lauryl (dodecyl) sulfate, for the analysis of drugs and other types of compounds. Brij-35 is the most suitable nonionic surfactant for micellar liquid chromatography, owing to its commercial availability, low cost, low toxicity, high cloud temperature, and low background absorbance. However, it has had minor use. In this work, we gather and discuss some results obtained in our laboratory with several β-blockers, sulfonamides, and flavonoids, concerning the use of Brij-35 as mobile phase mo…

Absorbancechemistry.chemical_compoundChromatographyAqueous solutionPulmonary surfactantchemistryMicellar liquid chromatographyPhase (matter)Filtration and SeparationEtherAcetonitrileMicellar electrokinetic chromatographyAnalytical ChemistryJournal of Separation Science
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Lanthanide–saccharide chemistry: synthesis and characterisation of Ce(III)–saccharide complexes

2000

A series of nine Ce(III) complexes has been synthesised with seven different monosaccharides (D-glucose, D-fructose, D-galactose, D-mannose, L-sorbose, D-ribose and D-xylose) and two different disaccharides (D-maltose and L-lactose), and these have been characterised with various analytical, spectral, magnetic and electrochemical techniques. The NMR studies have highlighted some interesting features about the metal-ion-binding pattern of the saccharides. Some additional coordination has been proposed along with the chelating groups in the saccharide molecules, based on the shifts in 13C NMR spectra. On the other hand, solution absorption studies and solid-state magnetic susceptibilities hav…

Absorption SpectraLanthanideMagnetic Resonance SpectroscopyStereochemistryMetal ions in aqueous solutionMannoseDisaccharidesBiochemistryAnalytical Chemistrychemistry.chemical_compoundSpectroscopy Fourier Transform InfraredElectrochemistryMonosaccharideOrganic chemistryMoleculeChelating Agentschemistry.chemical_classificationMolecular StructureSpectrometersCircular DichroismMetal IonsMonosaccharidesOrganic ChemistryElectric ConductivityElectron Spin Resonance SpectroscopyFructoseCeriumGeneral MedicineCarbon-13 NMRSorbosechemistrySpectrophotometryMetals Rare EarthElectrochemical AnalysisCarbohydrate Research
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Recognition of oxovanadium(V) species and its separation from other metal species through selective complexation by some acyclic ligands

1998

Acyclic molecules possessing –OH (phenoxo and alkoxo type) groups and imine or amine moieties have been developed to sense the specific preference for VO3+ species. These molecules also showed a capability to quantitatively separate oxovanadium(V) species from a reaction mixture containing metal species of V, Mo, U, Fe, and Mn ions in solution. A cascade quantitative separation of VO3+ followed by cis–MoO2+2 followed by trans –UO2+2 species is demonstrated from their mixture. Synthesis and structural details of oxo-species of vanadium molybdenum and uranium are also discussed. Factors influencing the complexation of these molecules towards oxo metal species of V, Mo and U are also addressed.

Absorption SpectraPolyanilineStereochemistryMetal ions in aqueous solutionImineCis-Dioxome(Vi)Vanadiumchemistry.chemical_elementTrans-Dioxoo(Iv)Medicinal chemistryInorganic ChemistryMetalSynthesisTransmetalationchemistry.chemical_compoundOxidationElectronicMaterials ChemistryPolythiophenesMoleculeSelective ComplexationPhysical and Theoretical ChemistryConducting PolymerCis-Dioxov(V)TransmetallationChemistryReactivityChemistryRecognitionMolybdenumvisual_artvisual_art.visual_art_mediumAmine gas treatingCrystallographicPolyhedron
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Structural, magnetic and electronic characterization of an isostructural series of dinuclear complexes of 3d metal ions bridged by tpbd

2013

Abstract Dinuclear complexes of the type [{M(H2O)(phen)}2(μ-tpbd)](ClO4)4 with N,N,N′,N′-Tetrakis-(2-pyridylmethyl)-benzene-1,4-diamine (tpbd) as bridging ligand and M = Mn(II) (1), Fe(II) (2), Co(II) (3), Ni(II) (4), Cu(II) (5), Zn(II) (6) were synthesized, structurally analyzed and their magnetic as well as their electrochemical properties are determined. A ligand-centered one-electron oxidation leads to radical complexes for which the lifetimes are strongly dependent on the coordinated metal ion as followed from time-resolved UV–Vis absorption spectroscopy. In addition to the six homometallic dinuclear complexes, one analog heterometallic Mn(II)/Ni(II) compound (7) of the same constituti…

Absorption spectroscopyChemistryMetal ions in aqueous solutionInorganic chemistryBridging ligandElectrochemistryCharacterization (materials science)Inorganic ChemistryMetalCrystallographyvisual_artMaterials Chemistryvisual_art.visual_art_mediumPhysical and Theoretical ChemistryIsostructuralGround statePolyhedron
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EXAFS and XANES Studies of CoxMg1−xO Solid Solutions Using a Laboratory EXAFS Spectrometer

1993

Studies of the local electronic structure and the short-range order in solid solutions CoxMg1−xO with x varying from 0.02 to 1.00 are carried out on the CoK-edge X-ray absorption spectra using a laboratory EXAFS spectrometer. A non-monotonous change of the CoO distance in the first coordination shell with a bent at about x = 0.5 is established. The second coordination shell of cobalt is formed by cobalt and magnesium atoms with a distribution close to a statistical one. [Russian Text Ignored.]

Absorption spectroscopySpectrometerExtended X-ray absorption fine structureInorganic chemistryAnalytical chemistrychemistry.chemical_elementElectronic structureCondensed Matter PhysicsXANESElectronic Optical and Magnetic MaterialsBond lengthchemistryCobaltSolid solutionPhysica Status Solidi (a)
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Determination of one compound in the presence of a single interference. Linear absorbances method

1992

The paper exposes the theoretical and experimental principles of an analytical procedure for the determination of one compound in the presence of another with an overlapping absorption spectrum, without the need to use any standard solutions of the latter. The proposed method was applied to the determination of binary mixtures of known composition in order to assess its accuracy and precision.

Accuracy and precisionAbsorption spectroscopyChemistryAnalytical chemistryBinary numberStandard solutionInterference (wave propagation)BiochemistryAnalytical ChemistryFresenius' Journal of Analytical Chemistry
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Comparison of novel and conventional calibration techniques for the analysis of urine samples using plasma source mass spectrometry combined with a n…

2012

The accuracy and precision of the analytical data from the analysis of liquid samples with high matrix load often suffer from a compromised performance of the sample introduction system. This is especially significant in the case of miniaturized, pneumatic low flow nebulizers. Alternative low-flow sampling devices based on different operating principles are imperative to overcome this drawback. The superior performance of such an alternative liquid sample introduction system for ICP-MS, the drop-on-demand (DOD) aerosol generator based on thermal inkjet technology, was recently outlined by the same group for the analysis of aqueous standard solutions. Current improvements of the system now a…

Accuracy and precisionChemistrybusiness.industryPlasma source mass spectrometryDrop (liquid)NozzleAnalytical chemistryStandard solutionAnalytical ChemistryMatrix (chemical analysis)Aerosol generatorOn demandProcess engineeringbusinessSpectroscopyJournal of Analytical Atomic Spectrometry
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Reversed phase liquid chromatography for the enantioseparation of local anaesthetics in polysaccharide-based stationary phases. Application to biodeg…

2020

[EN] A comprehensive study on the chiral separation of bupivacaine, mepivacaine, prilocaine and propanocaine with eight commercial polysaccharide-based chiral stationary phases (CSPs) in reversed phase conditions compatible with MS detection is performed. Methanol and acetonitrile are used as organic modifiers. Retention and resolution values obtained for each compound in the different CSPs and mobile phases are compared. The polysaccharide-based CSPs tested present different enantioselectivity towards the analytes. From the results, the experimental conditions for determining the enantiomers of bupivacaine, mepivacaine, prilocaine and propanocaine in saline aqueous samples using MS detecti…

AcetonitrilesResolution (mass spectrometry)Mepivacaine010402 general chemistry01 natural sciencesBiochemistryAnalytical Chemistrychemistry.chemical_compoundReversed phase conditionsPolysaccharidesPhase (matter)medicineEnantioselective biodegradation studyAnesthetics LocalAcetonitrileLocal anaestheticsChromatography High Pressure LiquidChromatography Reverse-PhaseAqueous solutionChromatographyCellulose and amylose-based chiral stationary phasesMethanol010401 analytical chemistryOrganic ChemistryEnantioselective synthesisWaterStereoisomerismGeneral MedicineReversed-phase chromatography0104 chemical sciencesMolecular WeightBiodegradation EnvironmentalchemistryEnantiomermedicine.drugJournal of chromatography. A
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