Search results for "2D-NMR"

showing 3 items of 3 documents

A new ecdysteroid and other constituents from two Dioscorea species

2008

Phytochemical investigation of the rhizome of Dioscorea dumetorum has led to the isolation by several chromatographic steps on normal and reversed phase silica gel of a new ecdysteroid, (20R)-5β,11α,20-trihydroxyecdysone (1), and two known ecdysteroids, ajugasterone C (2) and herkesterone (3). Their structures were determined by spectroscopic methods including 1D- and 2D-NMR (COSY, TOCSY, HSQC and HMBC). This is the first report on the occurrence of phytoecdysteroids in the Dioscoreaceae family. These compounds were devoid of antifungal activity against three Candida species (Candida albicans, Candida glabrata and Candida tropicalis, MIC > 200 μg/ml).

Dioscoreaceae01 natural sciencesBiochemistryCandida tropicalischemistry.chemical_compoundDioscoreaceaeCandida albicansDioscorea schimperianaDioscorea dumetorumEcology Evolution Behavior and SystematicsEcdysteroidChromatographybiologyCandida glabrata010405 organic chemistryEcdysteroidsbiology.organism_classification0104 chemical sciences3. Good healthRhizome010404 medicinal & biomolecular chemistrychemistryPhytochemicalBiochemistry[SDV.SP.PHARMA]Life Sciences [q-bio]/Pharmaceutical sciences/PharmacologyDioscorea2D-NMR
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Activation of a Sweet Taste Receptor by Oleanane-Type Glycosides from Wisteria sinensis

2022

The phytochemical study of Wisteria sinensis (Sims) DC. (Fabaceae), commonly known as the Chinese Wisteria, led to the isolation of seven oleanane-type glycosides from an aqueous-ethanolic extract of the roots. After successive purifications by various chromatographic methods, like solid/liquid chromatographic methods, vacuum liquid chromatography (VLC), medium pressure liquid chromatography (MPLC), on normal and reverse phase (RP-18 silica gel), and size exclusion chromatography on Sephadex L, their structures were elucidated by an extensive 600 MHz NMR analysis including 1D and 2D NMR experiments as well as ESI-MS. Among the seven isolated saponins, two have never been reported before : 3…

Organic ChemistryPharmaceutical ScienceFabaceaeSweet taste receptorsWisteria sinensisTAS1R2/TAS1R3Analytical ChemistryChemistry (miscellaneous)Drug Discovery[SDV.BBM] Life Sciences [q-bio]/Biochemistry Molecular BiologyMolecular Medicine<i>Wisteria sinensis</i>; Fabaceae; triterpene glycosides; sweet taste; TAS1R2/TAS1R3Physical and Theoretical Chemistry2D-NMRMolecules
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Interaction between flavour compounds and beta-lactoglobulin: approach by NMR and 2D/3D-QSAR studies of ligands

2004

 author cannot archive publisher's version/PDF; International audience; Interactions between flavour compounds and beta-lactoglobulin (BLG) have been the subject of several studies, but there are no unanimous binding site explanations. In our laboratory, interactions between BLG, and two flavour compounds, beta-ionone and gamma-decalactone, were studied by 2D-NMR spectroscopy. It appears that several amino acids affected by binding of gamma-decalactone are buried in the central cavity, whereas binding of beta-ionone affects amino acids located in a groove near the outer surface of the protein. 2D/3D-QSAR studies were performed using QSAR+ module of Cerius2 and Catalyst. The QSAR equation pr…

Quantitative structure–activity relationshipAROMAMolecular modelStereochemistry01 natural sciences03 medical and health sciencesComputational chemistryMolecular descriptor[SDV.IDA]Life Sciences [q-bio]/Food engineeringFLAVOURBinding site030304 developmental biology3D-QSAR0303 health sciencesChemistryHydrogen bondLigand[ SDV.IDA ] Life Sciences [q-bio]/Food engineeringGeneral Chemistry[SDV.IDA] Life Sciences [q-bio]/Food engineeringAffinitiesBETA-LACTOGLOBULIN0104 chemical sciences010404 medicinal & biomolecular chemistry2D-QSAR2D-NMRTwo-dimensional nuclear magnetic resonance spectroscopyFood Science
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