Search results for "3b"

showing 10 items of 143 documents

CCDC 1047646: Experimental Crystal Structure Determination

2017

Related Article: Michael Mirion, Lars Andernach, Caroline Stobe, Joaquin Barjau, Dieter Schollmeyer, Till Opatz, Arne Lützen, Siegfried R. Waldvogel|2015|Eur.J.Org.Chem.|2015|4876|doi:10.1002/ejoc.201500600

Space GroupCrystallographyCrystal SystemCrystal StructureCell Parametersrac-(5aRS7RS8aSR8cSR13bRS)-7-Ethyl-24101213b15-hexamethyl-568-trioxa-(benzo[h]-(benzo[b]furo)[23-b]-[4.3.3]propellan)-14-eneExperimental 3D Coordinates
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CCDC 1484252: Experimental Crystal Structure Determination

2016

Related Article: Stefan Pusch, Dieter Schollmeyer, Till Opatz|2016|Org.Lett.|18|3043|doi:10.1021/acs.orglett.6b01449

Space GroupCrystallographyCrystal SystemCrystal StructureCell Parametersrel-(3bR*7aR*)-11-acetyl-10-methyl-3b5677a9-hexahydrobenzo[56]furo[2'3':34]cyclohepta[12-b]pyrrol-8(4H)-oneExperimental 3D Coordinates
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CCDC 1484251: Experimental Crystal Structure Determination

2016

Related Article: Stefan Pusch, Dieter Schollmeyer, Till Opatz|2016|Org.Lett.|18|3043|doi:10.1021/acs.orglett.6b01449

Space GroupCrystallographyCrystal Systemrel-(3bR*7aS*)-11-acetyl-10-methyl-3b5677a9-hexahydrobenzo[56]furo[2'3':34]cyclohepta[12-b]pyrrol-8(4H)-oneCrystal StructureCell ParametersExperimental 3D Coordinates
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CCDC 652753: Experimental Crystal Structure Determination

2009

Related Article: A.Valkonen, M.Lahtinen, J.Tamminen, E.Kolehmainen|2008|J.Mol.Struct.|886|197|doi:10.1016/j.molstruc.2007.11.018

Space GroupCrystallographyMethyl 3beta-azido-5beta-cholan-24-oateCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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CCDC 652754: Experimental Crystal Structure Determination

2009

Related Article: A.Valkonen, M.Lahtinen, J.Tamminen, E.Kolehmainen|2008|J.Mol.Struct.|886|197|doi:10.1016/j.molstruc.2007.11.018

Space GroupCrystallographyMethyl 3beta-formyloxy-5beta-cholan-24-oateCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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Investigating the Molecular Mechanism of H3B-8800: A Splicing Modulator Inducing Preferential Lethality in Spliceosome-Mutant Cancers.

2021

The SF3B1 protein, part of the SF3b complex, recognizes the intron branch point sequence of precursor messenger RNA (pre-mRNA), thus contributing to splicing fidelity. SF3B1 is frequently mutated in cancer and is the target of distinct families of splicing modulators (SMs). Among these, H3B-8800 is of particular interest, as it induces preferential lethality in cancer cells bearing the frequent and highly pathogenic K700E SF3B1 mutation. Despite the potential of H3B-8800 to treat myeloid leukemia and other cancer types hallmarked by SF3B1 mutations, the molecular mechanism underlying its preferential lethality towards spliceosome-mutant cancer cells remains elusive. Here, microsecond-long a…

SpliceosomeQH301-705.5Protein ConformationPyridinesRNA SplicingMutantDruggabilityH3B-8800Molecular Dynamics Simulationmedicine.disease_causeCatalysisPiperazinesArticleInorganic ChemistryNeoplasmsspliceosome-mutant cancermedicineHumansPhysical and Theoretical ChemistryBiology (General)Molecular BiologyQD1-999SpectroscopyMutationsplicing modulatorsChemistryOrganic ChemistryWild typeIntronleukemiaGeneral MedicinePhosphoproteinsH3B‐8800molecular dynamicsComputer Science ApplicationsCell biologyChemistryPhenotypeCancer cellRNA splicingMutationRNA Splicing FactorsSpliceosome‐mutant cancerInternational journal of molecular sciences
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Synthesis of new derivatives of Nortopsentin with potential inhibitory activity against GSK-3b

Synthesis of new derivatives of Nortopsentin with potential inhibitory activity against GSK-3b
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Suppressive effects of C3b on monocyte-dependent T cell proliferation.

1987

The effect of C3b treatment of human monocytes on secondary antigen-dependent T cell response was studied. When antigen-specific T cell blasts were cultivated together with C3b-treated monocytes the proliferative response was inhibited in a dose-dependent fashion. This suppressive effect was specific for C3b because heat-inactivated C3b or buffer alone had no influence on T cell proliferation. In part, this suppressive effect is mediated through a C3b-induced decreased expression of class II antigens on the surface of treated monocytes, but another suppressive mechanism exists because the C3b pretreatment of monocytes also led to an inhibition of the proliferative response in a class II ant…

T cellT-LymphocytesImmunologyIndomethacinchemical and pharmacologic phenomenaBiologyIn Vitro TechniquesInhibitory postsynaptic potentialT cell responseLymphocyte ActivationMonocytesmedicineImmune ToleranceImmunology and AllergyHumansCells CulturedMonocyteComplement C3Molecular biologyProliferative responsemedicine.anatomical_structureComplement C3dComplement C3bImmunologic MemoryClass II Antigenscirculatory and respiratory physiologyEuropean journal of immunology
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Underlying Simple Graphs

2019

Summary In this article the notion of the underlying simple graph of a graph (as defined in [8]) is formalized in the Mizar system [5], along with some convenient variants. The property of a graph to be without decorators (as introduced in [7]) is formalized as well to serve as the base of graph enumerations in the future.

Theoretical computer scienceApplied Mathematics020207 software engineering0102 computer and information sciences02 engineering and technology68t9901 natural sciencesComputational Mathematics03b35010201 computation theory & mathematicsSimple (abstract algebra)underlying simple graphQA1-9390202 electrical engineering electronic engineering information engineering05c76Graph operationsgraph operationsMathematicsMathematicsofComputing_DISCRETEMATHEMATICSMathematicsFormalized Mathematics
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Caracterización molecular de la anemia refractaria con sideroblastos en anillo mediante un panel de secuenciación de segunda generación

2019

Los síndromes mielodisplásicos (SMD) son un grupo heterogéneo de neoplasias hematológicas que presentan citopenias, mielodisplasia, hematopoyesis ineficaz y un riesgo variable de transformación a leucemia mieloide aguda (t-LMA). Los SMD con sideroblastos en anillo (SMD-SA) constituyen aproximadamente el 10-12% de todos los SMD y en médula ósea muestran SA, eritroblastos con depósitos anormales de ferritina, en porcentaje igual o superior al 5%. El objetivo terapéutico en los SMD-SA es mejorar las citopenias y su sintomatología, en especial el síndrome anémico. La administración de eritropoyetina y el soporte transfusional con concentrados de hematíes son las opciones terpéuticas de primera …

UNESCO::CIENCIAS DE LA VIDA::Biología molecularazacitidina:CIENCIAS MÉDICAS ::Medicina interna::Hematología [UNESCO]SF3B1DNMT3Asecuenciaciónsíndromes mielodisplásicossideroblastos en anillo:CIENCIAS DE LA VIDA::Biología molecular [UNESCO]UNESCO::CIENCIAS MÉDICAS ::Medicina interna::Hematología
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