Search results for "Analytical"

showing 10 items of 9586 documents

The Potential Use of Resveratrol for Cancer Prevention.

2019

In addition to the traditional treatments of cancer and cancer prevention, the use of natural compounds, especially those found in food, should be considered. To clarify if resveratrol has the potential for cancer prevention and the possibility of use in therapy, the following must be taken into account: data from epidemiology, clinical protocol (case and control), preclinical studies (lab animals), use of established cell lines as models of cancer cells, test tube assays (enzymes activities), and requirements of nanotechnologies in order to discover new drugs to fight cancer. From this perspective and future expected advances, more information is needed such as improved efficacy, methods o…

medicine.medical_treatmentDrug Evaluation PreclinicalPharmaceutical ScienceReviewResveratrolresveratrolBioinformaticsChemopreventionAnalytical Chemistry03 medical and health scienceschemistry.chemical_compound0302 clinical medicinepreventionNeoplasmsDrug DiscoverymedicineAnimalsHumanscancerPhysical and Theoretical ChemistrySensitization030304 developmental biology0303 health sciencesmechanismsCancer preventionbusiness.industryOrganic ChemistryClinical Studies as TopicCancerDisease Managementmedicine.diseaseAntineoplastic Agents PhytogenicBioavailabilitymedicine.anatomical_structurechemistryChemistry (miscellaneous)030220 oncology & carcinogenesisapproach strategiesCancer cellMolecular MedicineDisease Susceptibilitybusinessinnovative formulationsAdjuvantSignal TransductionMolecules (Basel, Switzerland)
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Evaluation of Flavonoid Derivative and Doxorubicin Effects in Lung Cancer Cells (A549) Using Differential Pulse Voltammetry Method.

2018

Purpose: Electrochemical measurements have prompted the progress as a consequence of their affectability, cost-affectivity and comparatively short examination time. The aim of this study was the fast evaluation of the effect of chemotherapy compounds on the viability of lung cancer cells (A549) via electrochemical methods. Methods: Cyclic voltammetry (CV) was used as a primary method to distinguish between electrochemical behavior of normal and lung cancer cells. Differential pulse voltammetry (DPV) was employed as a complementary analyses method for the impact of doxorubicin (DOX) and Flavonoid modified drug (FMD) (US patent Application number: 62548886) on Lung cancer cells. Results: Only…

medicine.medical_treatmentFlavonoidPharmaceutical SciencePharmacology01 natural sciences0404 agricultural biotechnologyLung neoplasmsElectrochemistrymedicineDoxorubicinGeneral Pharmacology Toxicology and PharmaceuticsLung cancerVoltammetrychemistry.chemical_classificationChemotherapylcsh:RM1-950010401 analytical chemistry04 agricultural and veterinary sciencesmedicine.disease040401 food science0104 chemical scienceslcsh:Therapeutics. PharmacologychemistryDoxorubicinCancer cellVoltammetryDifferential pulse voltammetryCyclic voltammetryResearch Articlemedicine.drugAdvanced pharmaceutical bulletin
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2021

Severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) is the causative agent for the COVID-19 pandemic, which generated more than 1.82 million deaths in 2020 alone, in addition to 83.8 million infections. Currently, there is no antiviral medication to treat COVID-19. In the search for drug leads, marine-derived metabolites are reported here as prospective SARS-CoV-2 inhibitors. Two hundred and twenty-seven terpene natural products isolated from the biodiverse Red-Sea ecosystem were screened for inhibitor activity against the SARS-CoV-2 main protease (Mpro) using molecular docking and molecular dynamics (MD) simulations combined with molecular mechanics/generalized Born surface area b…

medicine.medical_treatmentMetaboliteIn silicoPharmaceutical SciencePharmacology01 natural sciencesMolecular mechanicsAnalytical Chemistry03 medical and health scienceschemistry.chemical_compoundDrug DiscoverymedicineProtease inhibitor (pharmacology)Physical and Theoretical ChemistryBinding site030304 developmental biology0303 health sciencesProteaseDrug discoveryOrganic ChemistryLopinavir0104 chemical sciences010404 medicinal & biomolecular chemistrychemistryChemistry (miscellaneous)Molecular Medicinemedicine.drugMolecules
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Characterization of the synthetic cannabinoid MDMB-CHMCZCA

2016

The synthetic cannabinoid MDMB-CHMCZCA was characterized by various spectroscopic techniques including NMR spectroscopy and tandem mass spectrometry. The synthetic sample was found to be of S-configuration by VCD spectroscopy and comparison of the data with DFT calculations, while ECD spectroscopy was found to be inconclusive in this case. The enantiomeric purity of samples from test purchases and police seizures was assessed by a self-developed chiral HPLC method.

medicine.medical_treatmentNPS010402 general chemistryTandem mass spectrometry01 natural sciencesFull Research Paperlcsh:QD241-441lcsh:Organic chemistrymedicinelcsh:Sciencechiral HPLCSpectroscopyChromatographyChemistry010401 analytical chemistryOrganic ChemistryNuclear magnetic resonance spectroscopy0104 chemical sciencesCharacterization (materials science)Chiral column chromatographyChemistryVCD spectroscopyECD spectroscopylcsh:QCannabinoidEnantiomersynthetic cannabinoidsBeilstein Journal of Organic Chemistry
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Encapsulation of Vitamins A and E as Spray-Dried Additives for the Feed Industry

2020

Encapsulated fat-soluble powders containing vitamin A (VA) and E (VE) were prepared as a feasible additive for extruded feed products. The effect of the encapsulating agents (Capsul-CAP&reg

medicine.medical_treatmentPharmaceutical Science02 engineering and technologyAnalytical Chemistrychemistry.chemical_compoundSpectroscopy Fourier Transform InfraredDrug DiscoveryVitamin E03.- Garantizar una vida saludable y promover el bienestar para todos y todas en todas las edadesVitamin ACalorimetry Differential ScanningTemperatureSpray Drying04 agricultural and veterinary sciences021001 nanoscience & nanotechnologyMaltodextrin040401 food science02.- Poner fin al hambre conseguir la seguridad alimentaria y una mejor nutrición y promover la agricultura sostenibleChemistry (miscellaneous)Spray dryingThermogravimetryMAQUINAS Y MOTORES TERMICOSMolecular MedicineEmulsionsExtrusionPowders0210 nano-technologyOxidation-ReductionPorosityMaterials scienceNanoemulsionsDrug CompoundingSodiumChemical structureSpray-dryingchemistry.chemical_elementArticle14.- Conservar y utilizar de forma sostenible los océanos mares y recursos marinos para lograr el desarrollo sosteniblelcsh:QD241-4410404 agricultural biotechnologylcsh:Organic chemistrymedicineThermal stabilityParticle SizePhysical and Theoretical ChemistryPorosityVitamin EOrganic ChemistryHumidityChemical engineeringchemistryDietary SupplementsNanoparticlesEncapsulationMolecules
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Cannabidiol Treatment Might Promote Resilience to Cocaine and Methamphetamine Use Disorders: A Review of Possible Mechanisms

2019

Currently, there are no approved pharmacotherapies for addiction to cocaine and other psychostimulant drugs. Several studies have proposed that cannabidiol (CBD) could be a promising treatment for substance use disorders. In the present work, the authors describe the scarce preclinical and human research about the actions of CBD on the effects of stimulant drugs, mainly cocaine and methamphetamine (METH). Additionally, the possible mechanisms underlying the therapeutic potential of CBD on stimulant use disorders are reviewed. CBD has reversed toxicity and seizures induced by cocaine, behavioural sensitization induced by amphetamines, motivation to self-administer cocaine and METH, context- …

medicine.medical_treatmentPharmaceutical ScienceCravingReviewPharmacologyAnalytical ChemistryHealth Risk Behaviorschemistry.chemical_compoundcannabidiol0302 clinical medicineDrug DiscoveryMedicineratrewardmedia_commonResilience PsychologicalMethamphetamineconditioned place preferenceSubstance Withdrawal SyndromeObservational Studies as TopicChemistry (miscellaneous)Molecular Medicineaddictionmedicine.symptomSelf-administrationself-administrationmedicine.drugmicemedia_common.quotation_subjectAmphetamine-Related DisorderscocaineContext (language use)lcsh:QD241-441Cocaine-Related Disorders03 medical and health scienceslcsh:Organic chemistryAnimalsHumansPhysical and Theoretical Chemistrymethamphetaminebusiness.industryAddictionOrganic ChemistryMeth-Conditioned place preferencedigestive system diseasesreinstatement030227 psychiatryStimulantchemistrybusiness030217 neurology & neurosurgeryMolecules
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Differential regulation of hexameric and dodecameric hemocyanin from A. leptodactylus

2013

The oxygen binding properties of hemocyanins are regulated on a short time scale by effectors such as l-lactate, urate and protons, and on longer time scales by expression of the different types of subunits. For Astacus leptodactylus it was shown previously that acclimation to higher temperatures leads to increased levels of a 6-meric hemocyanin species, whereas at lower temperatures the 12-meric form prevails. Here we show that the temperature dependence of the two forms supports the idea, that the maintenance of high affinity towards oxygen is the driving force for the differential expression of these hemocyanins. Furthermore, the two different types of hemocyanin differ not only in the a…

medicine.medical_treatmentProtein subunitAllosteric regulationBiophysicschemistry.chemical_elementAstacus leptodactylusBiochemistryOxygenAnalytical ChemistryAllosteric RegulationmedicineAnimalsBinding siteMolecular BiologyBinding SitesbiologyChemistryTemperatureIsothermal titration calorimetryHemocyaninbiology.organism_classificationUric AcidOxygenBiochemistryHemocyaninsLactatesBiophysicsAnuraProtein MultimerizationProtonsOxygen bindingBiochimica et Biophysica Acta (BBA) - Proteins and Proteomics
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Hyperstoichiometric interaction between silver and mercury at the nanoscale.

2012

Breaking through the stoichiometry barrier: As the diameter of silver particles is decreased below a critical size of 32?nm, the molar ratio of aqueous HgII to Ag0 drastically increases beyond the conventional Hg/Ag ratio of 0.5:1, leading to hyperstoichiometry with a maximum ratio of 1.125:1 (see figure). Therein, around 99?% of the initial silver is retained to rapidly form a solid amalgam with reduced mercury.

mercuryAnalytical chemistryNanoparticlechemistry.chemical_element02 engineering and technology010402 general chemistry01 natural sciencesRedoxCatalysisMolar ratioredox chemistryOrganic chemistrysilverSILICANanoscopic scaleSilver particlesComputingMilieux_MISCELLANEOUSAqueous solutionGeneral Chemistry021001 nanoscience & nanotechnologyCOLLOIDSCommunications0104 chemical sciencesMercury (element)REDUCTIONhyperstoichiometrychemistrynanoparticles0210 nano-technologyStoichiometryAngewandte Chemie (International ed. in English)
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Inorganic Mercury Sequestration by a Poly(ethylene imine) Dendrimer in Aqueous Solution

2015

The interaction of the G-2 poly(ethylene imine) dendrimer L, derived from ammonia as initiating core, with Hg(II) and HgCl4 2− was studied in aqueous solution by means of potentiometric (pH-metric) measurements. Speciation of these complex systems showed that L is able to form a wide variety of complexes including 1:1, 2:1, 3:1 and 3:2 metal-to-ligand species, of different protonation states, as well as the anion complexes ((H7L)HgCl4) 5+ and ((H8L)HgCl4) 6+ . The stability of the metal complexes is very high, making L an excellent sequestering agent for Hg(II), over a large pH range, and a promising ligand for the preparation of functionalized activated carbons to be employed in the remedi…

mercuryImineInorganic chemistryPotentiometric titrationPharmaceutical Sciencechemistry.chemical_elementProtonationmercury dendrimers sequestration water contamination environmentArticleAnalytical Chemistrydendrimerspoly(ethylene imine)Metallcsh:QD241-441chemistry.chemical_compoundAmmoniacontaminationlcsh:Organic chemistryDendrimerDrug DiscoveryremediationPhysical and Theoretical ChemistryAqueous solutionMolecular StructureOrganic ChemistryMercury (element)chemistryChemistry (miscellaneous)visual_artPotentiometryvisual_art.visual_art_mediumMolecular MedicineEnvironmental PollutantsIminesPolyethylenesMolecules
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Observation of the rare decay K-S -> pi(0)e(+)e(-)

2003

A search for the decay Ks->pi0e+e- has been made by the NA48/1 experiment at the CERN SPS accelerator. Using data collected during 89 days in 2002 with a high-intensity Ks beam, 7 events were found with a background of 0.15 events. The branching fraction BR(Ks->pi0e+e-, m(ee) > 0.165 GeV/c^2) = (3.0^{+1.5}_{-1.2}(stat) +/-0.2 (syst)) x 10^{-9} has been measured. Using a vector matrix element and a form factor equal to one, the measurement gives BR(Ks->pi0e+e-) = (5.8^{+2.9}_{-2.4}) x 10^{-9}.

mesoni K; decadimenti rariPhysicsNuclear and High Energy Physics010308 nuclear & particles physicsBranching fractionK-LForm factor (quantum field theory)Analytical chemistryKAON DECAYS01 natural sciences3. Good healthHigh Energy Physics - Experimentmesoni Kdecadimenti rariCP VIOLATION; KAON DECAYS; K-L; SEARCHSEARCH0103 physical sciencesMatrix elementCP VIOLATIONAtomic physics010306 general physics
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