Search results for "Anti-inflammatory drug"

showing 4 items of 14 documents

The Effect of Acetylsalicylic Acid, as a Representative Non-Steroidal Anti-Inflammatory Drug, on the Activity of Myeloperoxidase

2023

Background: Acetylsalicylic acid (ASA or aspirin) is one of the world’s most widely used non-steroidal anti-inflammatory drug (NSAID). Numerous studies have shown that the long-term use of aspirin may contribute to longer survival among patients with various types of cancer, including ovarian cancer. Aim: The aim of this study was to investigate the effect of ASA on myeloperoxidase (MPO), which is found at an elevated level in women with ovarian cancer, among others. Methods: The influence of different concentrations of ASA on the chlorinating and peroxidase activity of MPO was analysed. The relationship between the concentration of ASA and the degree of inhibition of MPO activity was deter…

myeloperoxidasenon-steroidal anti-inflammatory drugsacetylsalicylic acidPharmaceuticals
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Nesteroīdo pretiekaisuma līdzekļu aprite aptiekā

2020

Nesteroīdie pretiekaisuma līdzekļi (NPL) ir vispieprasītākā medikamentu grupa pasaulē. Galvenie iemesli NPL lietošanai ir sāpes, iekaisums un drudzis. Darba mērķis bija salīdzināt NPL pieprasījumu par 2017., 2018. un 2019. gadu, kā arī noskaidrot, kādas ir biežākās blakusparādības, ar kurām šo medikamentu lietošanas laikā sastopas respondenti. Darba uzdevumi bija izanalizēt NPL apgrozījumu vienā no SIA “Euro aptieka” tīkla aptiekām, kura atrodas Rīgā, Ziepniekkalna rajonā par 2017., 2018. un 2019. gadu, noskaidrot, kuri NPL medikamenti ir vispieprasītākie, noskaidrot, kādas ir visbiežākās blakusparādības respondentiem, noskaidrot, kādas sāpes biežāk piemeklē respondentus. Iegūtie dati lieci…

nesteroīdie pretiekaisuma līdzekļinon-steroidal anti-inflammatory drugsFarmācijaparacetamolsibuprofēnssāpes
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Synthesis, characterization, and cellular investigations of porphyrin– and chlorin–indomethacin conjugates for photodynamic therapy of cancer

2021

Indomethacin is a potent non-steroidal anti-inflammatory drug (NSAID) with a strong selective inhibitor activity towards cyclooxygenase-2 (COX-2), an enzyme that is highly overexpressed in various tumour cells, being involved in tumourigenesis. Concomitantly, porphyrins have gained much attention as promising photosensitizers (PSs) for the non-invasive photodynamic therapy (PDT) of cancer. Herein, we report the design, and determine the singlet oxygen generation capacity and in vitro cellular toxicity of porphyrin- and chlorin-indomethacin conjugates (P2-Ind and C2-Ind). Both the conjugates were obtained in high yields and were characterized by 1H, 19F and 13C NMR as well as by high resolut…

photosensitizermedicine.medical_treatmentPhotodynamic therapyDFT calculations010402 general chemistryPhotochemistry01 natural sciencesBiochemistrychemistry.chemical_compoundnon-steroidal anti-inflammatory drugpolycyclic compoundsmedicinePhysical and Theoretical ChemistryTriplet stateCytotoxicity010405 organic chemistrySinglet oxygenOrganic Chemistrysinglet oxygen generationPorphyrin0104 chemical sciencesPhotochemotherapychemistrySettore CHIM/03 - Chimica Generale E InorganicaChlorincytotoxicityPhototoxicityporphyrinConjugateOrganic & Biomolecular Chemistry
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Isolement et caractérisation de saponosides extraits de deux plantes médicinales : Cyclamen africanum, Zygophyllum cornutum et évalution de leur acti…

2014

The appearance of several diseases, such as cancer, diabetes, high blood pressure and spread of infections mutagenic virus type can be linked to the quality and lifestyle that we lead today. Indeed, several studies on the factors triggering these so-called "morbid" long-or short-term illnesses are related to stress and quality of food consumed, whether of plant and animal origin. These diseases are becoming a common occurrence, they affect different races and all classes of society. According ethnobotanical research, naturally occurring substances, allowed civilizations to survive deadly diseases. For example, we thus find references to periods of malarial fever in China and one of the symp…

protéines réponse inflammatoire (PRI)[SDV.MHEP] Life Sciences [q-bio]/Human health and pathologyMass spectrometry1D and 2D NMRZygophyllum cornutumMédiateurs pro-inflammatoire (COX-2)Anti-inflammatoires (AINS)INOSPro-inflammatory mediatorsProtein inflammatory response (PRI)Activité anti inflammatoireAnti inflammatory activitySaponins triterpeneCyclamen africanumCOX-2Spectrométrie de masseRMN 1DRMN 2DSaponines triterpéniques[SDV.SP.PHARMA] Life Sciences [q-bio]/Pharmaceutical sciences/Pharmacology[SDV.SP.PHARMA]Life Sciences [q-bio]/Pharmaceutical sciences/PharmacologyAnti-inflammatory drugs (NSAIDs)TNF -αPGE2[SDV.MHEP]Life Sciences [q-bio]/Human health and pathology
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