Search results for "BLAST"

showing 10 items of 2136 documents

Lead-time and overdiagnosis estimation in neuroblastoma screening.

2003

In Germany, neuroblastoma is the most frequent extracranial solid childhood tumour. Its properties made it seem an ideal candidate for screening. A German trial assessed the effect of screening at one year of age from 1995-2001 in a nationwide project. We present here the methods developed for the estimation of lead-time and overdiagnosis in this project. Follow up on 1.5 million screened children and 2.1 million control children is currently available until June 2002. Ascertainment of control cohort cases and false negative cases is complete up to this date. A method for determining an empirical lead-time distribution and overdiagnosis estimate from comparing the age specific incidences in…

Statistics and ProbabilityPediatricsmedicine.medical_specialtyEpidemiologySensitivity and SpecificityCohort StudiesNeuroblastomaAge DistributionGermanyNeuroblastoma screeningBiomarkers TumorMedicineHumansMass ScreeningFalse Positive ReactionsOverdiagnosisMass screeningEstimationbusiness.industryIncidence (epidemiology)IncidenceInfantPopulation SurveillanceCohortbusinessLead timeDemographyCohort studyStatistics in medicine
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Paracrine effect of membrane vesicles released by mouse mesoangioblast stem cells on non correlated cell types

2016

Introduction Mouse mesoangioblasts are vessel-associated multipotent progenitor stem cells, which are able to differentiate into different mesodermal cell types. In our previous paper we have demonstrated that these cells are able to shed in the extracellular environment membrane vesicles (EV), which contain both structural proteins and biological factors such as FGF2 and the two gelatinases MMP2/9. EV represent an important mediator of cell-to-cell communication and are involved in both autocrine and paracrine signalling. Interestingly, there is a bidirectional signalling exchange between stem cell EV and damaged cells. In particular, EV from injured cells can reprogram stem cells to acqui…

Stem cells mesoangioblasts membrane vesicles migration. macrophages endothelial cells.
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Inhibition of Cancer Derived Cell Lines Proliferation by Synthesized Hydroxylated Stilbenes and New Ferrocenyl-Stilbene Analogs. Comparison with Resv…

2014

Further advances in understanding the mechanism of action of resveratrol and its application require new analogs to identify the structural determinants for the cell proliferation inhibition potency. Therefore, we synthesized new trans-resveratrol derivatives by using the Wittig and Heck methods, thus modifying the hydroxylation and methoxylation patterns of the parent molecule. Moreover, we also synthesized new ferrocenylstilbene analogs by using an original protective group in the Wittig procedure. By performing cell proliferation assays we observed that the resveratrol derivatives show inhibition on the human colorectal tumor SW480 cell line. On the other hand, cell viability/cytotoxicit…

StereochemistryCell SurvivalPharmaceutical ScienceResveratrolresveratrolArticleAnalytical Chemistrylcsh:QD241-441chemistry.chemical_compoundlcsh:Organic chemistryIntestinal mucosaCell Line TumorDrug DiscoveryStilbenesresveratrol; methoxystilbenes; ferrocenylstilbene analogs; colon cancer; hepatoblastomaHumansViability assayFerrous CompoundsPhysical and Theoretical ChemistrymethoxystilbenesIntestinal MucosaCytotoxicityCell ProliferationCell growthferrocenylstilbene analogsOrganic ChemistryCell CycleEpithelial CellsHep G2 CellsCell cyclehepatoblastomaBiochemistrychemistrycolon cancerChemistry (miscellaneous)Cell cultureCancer cellMolecular MedicineColorectal NeoplasmsMolecules
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Antiproliferative agents that interfere with the cell cycle at the G(1)-->S transition: further development and characterization of a small library o…

2008

In this continuation of our research on derivatives containing the stilbene privileged structure or that are derived from it, we report the results of further studies carried out on the previously initiated collection of compounds. We used a parallel synthetic approach to rapidly obtain small sets of compounds and started the annotation of the library in progress by calculating some physicochemical properties to be eventually correlated with biological activities. A pharmacophore for the antiproliferative activity was also built to summarize the features of the library. We evaluated the antiproliferative and pro-apoptotic activities of all compounds as well as the cell-cycle effects of some…

StereochemistryCellular differentiationAntineoplastic AgentsApoptosisHL-60 CellsBiochemistryS PhaseSmall Molecule Librarieschemistry.chemical_compoundInhibitory Concentration 50Biological profileCell Line TumorDrug DiscoveryStilbenespharmacophoresHumansGeneral Pharmacology Toxicology and PharmaceuticsPhosphorylationPharmacologyChemistryOrganic ChemistryG1 PhaseRetinoblastomaSmall Molecule LibrariesG1/S transitionCell DifferentiationCell cycleFlow CytometryCombinatorial chemistryantitumor agentAntiproliferative AgentsMolecular MedicineTriolcell cyclePharmacophoreC-C couplingK562 Cells
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[68Ga]Ga-DO2A-(OBu-l-tyr)2: Synthesis, 68Ga-radiolabeling and in vitro studies of a novel 68Ga-DO2A-tyrosine conjugate as potential tumor tracer for …

2009

The synthesis, (68)Ga-labeling and in vitro study of the novel tyrosine chelate derivative [(68)Ga]Ga-1,4,7,10-tetraazacyclododecane-1,7-diacetic acid-4,10-di-(O-butyl)-l-tyrosine ([(68)Ga]Ga-DO(2)A-(OBu-l-tyr)(2)) as a potential tracer for imaging tumor metabolism by positron emission tomography (PET) is presented. This approach combines the biological amino acid transporter targeting properties of l-tyrosine with the outstanding availability of (68)Ga(III) via the (68)Ge/(68)Ga generator. In vitro studies utilizing the F98-glioblastoma cell line revealed specific uptake of [(68)Ga]Ga-DO2A-(OBu-l-tyr)(2) that was comparable to that of the reference O-(2-[(18)F]fluoroethyl)-l-tyrosine (FET)…

StereochemistryClinical BiochemistryPharmaceutical ScienceBiochemistryChemical synthesisCell Line TumorDrug DiscoveryOrganometallic CompoundsAnimalsChelationAmino acid transporterTyrosineMolecular BiologyGallium IsotopesFluoroethylBrain NeoplasmsChemistryOrganic ChemistryLigand (biochemistry)In vitroRatsPositron-Emission TomographyMolecular MedicineRadiopharmaceuticalsGlioblastomaConjugateBioorganic & Medicinal Chemistry Letters
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Polysaccharide/polyaminoacid composite scaffolds for modified DNA release.

2009

Abstract In this work composite polymeric films or sponges, based on hyaluronic acid (HA) covalently crosslinked with α,β-poly(N-2-hydroxyethyl)(2-aminoethylcarbamate)- d , l -aspartamide (PE), have been prepared and characterized as local gene delivery systems. In particular, HA/PE scaffolds have been loaded with PE/DNA interpolyelectrolyte complexes, employing PE as a macromolecular crosslinker for HA and as a non-viral vector for DNA. In vitro studies showed that HA/PE films and sponges have high compatibility with human dermal fibroblasts and they give a sustained DNA release, whose trend can be easily tailored by varying the crosslinking ratio between HA and PE. Electrophoresis analysi…

StereochemistryMelanoma ExperimentalPharmaceutical ScienceHyaluronoglucosaminidaseElectrophoretic Mobility Shift Assaymacromolecular substancesBiologyGene deliveryTransfectionchemistry.chemical_compoundMiceTissue engineeringHyaluronic acidPolyaminesCOMPOSITE SCAFFOLD SCAFFOLD AMINOACID DNA RELEASE.AnimalsHumansHyaluronic AcidAspartameCells CulturedMolecular StructureGenetic transfertechnology industry and agricultureBiological TransportTransfectionDNAFibroblastsIn vitroKineticsCross-Linking ReagentschemistrySolubilitySettore CHIM/09 - Farmaceutico Tecnologico ApplicativoNucleic Acid ConformationDNAMacromoleculeNuclear chemistryInternational journal of pharmaceutics
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Effects of Hypericum Extract on the Expression of Serotonin Receptors

1994

The influence of hypericum extract LI 160 on the expression of serotonin receptors was investigated using a neuroblastoma cell line to establish a model for the regulation of neurotransmitters by immunologically active compounds such as cytokines. The cells were incubated with hypericum extract LI 160 in kinetic form for 2, 4, 6, 8, and 10 hours, then washed. The serotonin receptor expression analysis was compared to that of a placebo control solution. The neuroblastoma cells showed a clearly reduced expression of the serotonin receptors under treatment with hypericum extract. First stimulation experiments with interleukin-1 (IL-1) and hypericum extract suggest that a further reduction of …

StimulationPharmacologyPharmacognosyNeuroblastoma cellNeuroblastoma03 medical and health sciences0302 clinical medicineTumor Cells CulturedAnimalsHypericum extractPerylene5-HT receptorPlants Medicinal030214 geriatricsPlant ExtractsChemistryHypericum perforatumBiological activityAntidepressive AgentsIn vitroRatsPsychiatry and Mental healthXanthenesReceptors SerotoninQuercetinSerotonin AntagonistsNeurology (clinical)Geriatrics and GerontologyHypericum030217 neurology & neurosurgeryInterleukin-1Journal of Geriatric Psychiatry and Neurology
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Streptavidin-coated TiO2 surfaces are biologically inert: Protein adsorption and osteoblast adhesion studies

2011

Non-fouling TiO2 surfaces are attractive for a wide range of applications such as biosensors and medical devices, where biologically inert surfaces are needed. Typically, this is achieved by controlled surface modifications which prevent protein adsorption. For example, polyethylene glycol (PEG) or PEG-derived polymers have been widely applied to render TiO2 surfaces biologically inert. These surfaces have been further modified in order to achieve specific bio-activation. Therefore, there have been efforts to specifically functionalize TiO2 surfaces with polymers with embedded biotin motives, which can be used to couple streptavidin for further functionalization. As an alternative, here a s…

StreptavidinMaterials scienceSurface PropertiesBiomedical EngineeringNanotechnologyMicroscopy Atomic ForceCell LineBiomaterialschemistry.chemical_compoundCell AdhesionHumansBiotinylationTitaniumchemistry.chemical_classificationOsteoblaststechnology industry and agricultureMetals and AlloysPolymerSilanesFibronectinsKineticsSurface coatingchemistryBiotinylationCeramics and CompositesSurface modificationMuramidaseAdsorptionStreptavidinBiosensorLayer (electronics)Protein adsorptionJournal of Biomedical Materials Research Part A
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The Marine Sponge-Derived Inorganic Polymers, Biosilica and Polyphosphate, as Morphogenetically Active Matrices/Scaffolds for the Differentiation of …

2014

The two marine inorganic polymers, biosilica (BS), enzymatically synthesized from ortho-silicate, and polyphosphate (polyP), a likewise enzymatically synthesized polymer consisting of 10 to >100 phosphate residues linked by high-energy phosphoanhydride bonds, have previously been shown to display a morphogenetic effect on osteoblasts. In the present study, the effect of these polymers on the differential differentiation of human multipotent stromal cells (hMSC), mesenchymal stem cells, that had been encapsulated into beads of the biocompatible plant polymer alginate, was studied. The differentiation of the hMSCs in the alginate beads was directed either to the osteogenic cell lineage by …

Stromal cellAlginatesPolymersCellular differentiationOsteogenesis DistractionPharmaceutical ScienceBone Morphogenetic Protein 2biosilica; polyphosphate; multipotent stromal cells; mesenchymal stem cells; alkaline phosphatase; 3D cell/tissue printing; distraction osteogenesisBone morphogenetic protein 2ChondrocyteArticleCollagen Type IGlucuronic AcidPolyphosphatesDrug Discoverymedicinemultipotent stromal cellsAnimalsHumansbiosilicaPharmacology Toxicology and Pharmaceutics (miscellaneous)lcsh:QH301-705.5Collagen Type IImesenchymal stem cells3D cell/tissue printingOsteoblastsTissue ScaffoldsChemistryHexuronic AcidsMesenchymal stem cellBiomaterialpolyphosphateCell DifferentiationAnatomyChondrogenesisAlkaline PhosphataseSilicon DioxideCell biologyPoriferamedicine.anatomical_structuredistraction osteogenesislcsh:Biology (General)Alkaline phosphataseMarine Drugs
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The influence of bone allograft processing on osteoblast attachment and function

2004

In order to assess the influence of eight different sterilisation and disinfection methods for bone allografts on adhesion, proliferation, and differentiation of human bone marrow stromal cells (BMSC), cells were grown in culture and then plated onto pieces of human bone allografts. Following processing methods were tested: autoclavation (AUT), low-temperature-plasma sterilisation of demineralised allografts (D-LTP), ethylene oxide sterilisation (EtO), fresh frozen bone (FFB), 80 degrees C-thermodisinfection (80 degrees C), gamma-irradiation (Gamma), chemical solvent disinfection (CSD), and Barrycidal-disinfection (BAR). The seeding efficiency was determined after one hour to detect the num…

Stromal cellCell Survivalmedicine.medical_treatmentOsteocalcinPopulationGene ExpressionBone Marrow CellsIn Vitro TechniquesBone graftingAndrologyCell AdhesionmedicineHumansTransplantation HomologousOrthopedics and Sports MedicineViability assayCell adhesioneducationCells CulturedBone Marrow Transplantationeducation.field_of_studyOsteoblastsbiologyChemistrySterilizationCell DifferentiationOsteoblastAlkaline PhosphataseTransplantationmedicine.anatomical_structureImmunologyOsteocalcinbiology.proteinStromal CellsCell DivisionJournal of Orthopaedic Research
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