Search results for "COPP"

showing 10 items of 3147 documents

Synthesis, Crystal Structure, Magnetic Properties, and Theoretical Studies of [{Cu(mepirizole)Br}2(μ-OH)(μ-pz)] (Mepirizole = 4-Methoxy-2-(5-methoxy-…

2003

A novel mu-pyrazolato-mu-hydroxo-dibridged copper(II) complex has been synthesized and structurally characterized: [(Cu(mepirizole)Br)2(mu-OH)(mu-pz)] (mepirizole=4-methoxy-2-(5-methoxy-3-methyl-1H-pyrazol-1-yl)-6-methylpyrimidine; pz=pyrazolate). The title compound crystallizes in the monoclinic system, space group P2(1)/c, with a=15.618(2) A, b=15.369(3) A, c=16.071(3) A, and beta=112.250(1) degrees. The structure is built up of dinuclear [(Cu(mepirizole)Br)2(mu-OH)(mu-pz)] units with five-coordinated copper(II) ions (CuBrN3O chromophores) linked by mu2-OH and mu2-pyrazolato bridges that are well separated from each others. The intramolecular copper-copper distance is 3.378(3) A. Magnetic…

Models MolecularChemical PhenomenaChemistry PhysicalBand gapStereochemistryIronchemistry.chemical_elementCrystal structureChromophoreCrystallography X-RayLigandsCopperMagnetic susceptibilityIonInorganic ChemistryMagneticsCrystallographychemistryIntramolecular forceIndicators and ReagentsEpirizolePhysical and Theoretical ChemistryMonoclinic crystal systemInorganic Chemistry
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Metamorphosis of a butterfly: synthesis, structural, thermal, magnetic and DFT characterisation of a ferromagnetically coupled tetranuclear copper(ii…

2007

The reaction in water of Cu(OH)(2) with 2,2'-bipyridine (bipy) and (NH(4))(2)HPO(4) in a 4 : 4 : 2 molar ratio under an inert atmosphere leads to the formation of a tetranuclear copper(II) complex of formula {[(H(2)O)(2)Cu(4)(bipy)(4)(mu(4)-PO(4))(2)(mu(2)-OH)] x 0.5 HPO(4) x 15.5 H(2)O}, 1, with butterfly topology. The structure of the tetranuclear core in 1 consists of four crystallographically unique copper(II) ions in approximate square-pyramidal geometry with each coordinated to a bipy ligand and interacting through two mu(4)-O,O',O''-phosphate bridges. Additional bridging between Cu(3) and Cu(4) is provided by a hydroxide ligand, whereas two water molecules cap the Cu(1) and Cu(2) squ…

Models MolecularChemistryLigandInorganic chemistryTemperaturechemistry.chemical_elementChromophoreCrystallography X-RayCopperMagnetic susceptibilityIonInorganic ChemistryMagneticsCrystallographychemistry.chemical_compoundModels ChemicalIntramolecular forceOrganometallic CompoundsMoleculeHydroxideCopperDalton Transactions
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Ferromagnetic Cu(II)4, Co(II)4, and Ni(II)6 azido complexes derived from metal-assisted methanolysis of di-2,6-(2-pyridylcarbonyl)pyridine.

2009

Reaction of copper(II) perchlorate with di-2,6-(2-pyridylcarbonyl)pyridine (pyCOpyCOpy, dpcp) in the presence of sodium azide yields complex [Cu(4)(N(3))(2){pyC(OMe)(O)pyC(OMe)(O)py}(2)(MeOH)(2)](ClO(4)) x 2 MeOH (1 x 2 MeOH), which crystallizes in the monoclinic P2(1)/c space group. Similar reaction of cobalt(II) nitrate yields complex [Co(4)(N(3))(2)(NO(3))(2){pyC(OMe)(O)pyC(OMe)(O)py}(2)] x 0.5 MeOH (2 x 0.5 MeOH) which crystallizes in the monoclinic I2/m space group. Reaction of nickel(II) perchlorate yields complex [Ni(6)(CO(3))(N(3))(6){pyCOpyC(O)(OMe)py}(3)(MeOH)(2)(H(2)O)][Ni(6)(CO(3))(N(3))(6){pyCOpyC(O)(OMe)py}(3) (MeOH)(3)](ClO(4))(2) x 1.8 MeOH (3 x 1.8 MeOH), which crystallizes…

Models MolecularChemistryStereochemistryPyridinesCyclohexane conformationTemperaturechemistry.chemical_elementCobaltCrystallography X-RayMagnetic susceptibilityInorganic ChemistryPerchloratechemistry.chemical_compoundNickelCrystallographyMagneticsDeprotonationCubaneNickelPyridineOrganometallic CompoundsPhysical and Theoretical ChemistryCopperMonoclinic crystal systemInorganic chemistry
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Synthesis, characterization, cellular uptake and interaction with native DNA of a bis(pyridyl)-1,2,4-oxadiazole copper(II) complex

2010

The copper(II) complex of 3,5-bis(2'-pyridyl)-1,2,4-oxadiazole was synthesized and characterized. X-Ray crystallography revealed that the complex consists of a discrete [Cu(3,5-bis(2'-pyridyl)-1,2,4-oxadiazole)(2)(H(2)O)(2)](2+) cation and two ClO(4)(-) anions. The Cu(II) coordination sphere has a distorted octahedral geometry and each ligand chelates the copper ion through the N(4) nitrogen of the oxadiazole ring and the nitrogen of one pyridine moiety. The coordinated water molecules are in cis position and each of them is H-bonded to the 5-pyridyl nitrogen of the oxadiazole ligand and to an oxygen of the perchlorate anion. Biological assays showed that, despite the free ligand not being …

Models MolecularCircular dichroismCoordination sphereheterocylces metal complex DNA binders anti-tumoralsCell SurvivalPyridinesStereochemistrychemistry.chemical_elementOxadiazoleLigandsInorganic Chemistrychemistry.chemical_compoundPerchlorateCell Line TumorOctahedral molecular geometryOrganometallic CompoundsHumansOxadiazolesChemistryLigandDNASettore CHIM/06 - Chimica OrganicaCopperBinding constantCrystallographySettore CHIM/03 - Chimica Generale E InorganicaCopper
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DNA binding and antiproliferative activity toward human carcinoma cells of copper(ii) and zinc(ii) complexes of a 2,5-diphenyl[1,3,4]oxadiazole deriv…

2012

The interaction of calf thymus DNA with [CuL(ClO(4))]ClO(4)·H(2)O (1) and [ZnLBr]Br·H(2)O (2) (L = 9,12,15,18,27,28-hexaaza-29-oxatetracyclo[24.2.1.0(2,7).0(20,25)]enneicosa-2,4,6,20,22,24,26,28(1)-octaene) dicationic complexes in aqueous solution at neutral pH, was investigated by variable-temperature UV-vis absorption, circular dichroism and fluorescence spectroscopy. The values of the DNA-binding constants of these complexes, determined by competitive binding spectrofluorimetric titrations of ethidium bromide (EB)-DNA solutions, are (6.7 ± 0.5) × 10(6) M(-1) for CuL(2+) and (4.7 ± 0.5) × 10(5) M(-1) for ZnL(2+). These data together with a through analysis of the spectroscopic behaviour c…

Models MolecularCircular dichroismDNA binding antiproliferative activity 25-diphenyl[134]oxadiazole derivativeStereochemistryCell SurvivalOxadiazoleAntineoplastic AgentsBreast NeoplasmsNucleic Acid DenaturationFluorescence spectroscopyInorganic Chemistrychemistry.chemical_compoundCoordination ComplexesCell Line TumorHumansOxazolesAqueous solutionDNAIn vitroZincchemistrySettore CHIM/03 - Chimica Generale E InorganicaTitrationFemaleEthidium bromideDNACopper
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Copper(II)-Induced Restructuring of ZnuD, a Zinc(II) Transporter from Neisseria meningitidis.

2019

Cluster 2 (288HDDDNAHAHTH298) from Neisseria meningitidis ZnuD is a flexible loop that captures zinc(II) ions, acting as a "fishing net". We describe its Zn(II) and Cu(II) binding capabilities, focusing on the thermodynamics of such interactions and comparing them with the complexes of the 1MAHHHHHHL9-NH2 region. Copper(II) complexes with the studied ZnuD regions are thermodynamically more stable than the zinc(II) ones-Cu(II) complexes dominate in solution even in close to physiological ratios of the studied metal ions (a 10-fold excess of Zn(II) over Cu(II)). While the binding of native Zn(II) has no significant impact on the structure of its transporter, Cu(II) binding induces a conformat…

Models MolecularConformational changeMetal ions in aqueous solutionchemistry.chemical_elementZincNeisseria meningitidis010402 general chemistry01 natural sciencesInorganic ChemistryBacterial ProteinsHumansProlineAmino Acid SequencePhysical and Theoretical ChemistryCation Transport ProteinsPolyproline helix010405 organic chemistryTransporterCopper0104 chemical sciencesMeningococcal InfectionsCrystallographyZincchemistryHelixThermodynamicsCopperProtein BindingInorganic chemistry
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Cupredoxin-like domains in haemocyanins

2010

Haemocyanins are multimeric oxygen transport proteins, which bind oxygen to type 3 copper sites. Arthropod haemocyanins contain 75-kDa subunits, whereas molluscan haemocyanins contain 350–400-kDa subunits comprising seven or eight different 50 kDa FUs (functional units) designated FU-a to FU-h, each with an active site. FU-h possesses a tail of 100 amino acids not present in the other FUs. In the present study we show by X-ray crystallography that in FU-h of KLH1 (keyhole-limpet-haemocyanin isoform 1) the structure of the tail domain is cupredoxin-like but contains no copper. The copper-free domain 3 in arthropod haemocyanin subunits has also recently been reinterpreted as being cupredoxin-…

Models MolecularCopper proteinmedicine.medical_treatmentGastropodaMolecular Sequence DataBiologyCrystallography X-RayBiochemistryAzurinmedicineAnimalsAmino Acid SequenceBinding siteMolecular BiologyPeptide sequencePhylogenychemistry.chemical_classificationBinding SitesSequence Homology Amino AcidOxygen transportActive siteHemocyaninCell BiologyAnatomyProtein Structure TertiaryAmino acidMolecular WeightBiochemistrychemistryHemocyaninsbiology.proteinAzurinCopper
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Similar enzyme activation and catalysis in hemocyanins and tyrosinases

2006

This review presents the common features and differences of the type 3 copper proteins with respect to their structure and function. In spite of these differences a common mechanism of activation and catalysis seems to have been preserved throughout evolution. In all cases the inactive proenzymes such as tyrosinase and catecholoxidase are activated by removal of an amino acid blocking the entrance channel to the active site. No other modification at the active site seems to be necessary to enable catalytic activity. Hemocyanins, the oxygen carriers in many invertebrates, also behave as silent inactive enzymes and can be activated in the same way. The molecular basis of the catalytic process…

Models MolecularCopper proteinmedicine.medical_treatmentTyrosinaseCatalysisEnzyme activatorProtein structureGeneticsmedicineAnimalsHumanschemistry.chemical_classificationbiologyMonophenol MonooxygenaseActive siteHemocyaninGeneral MedicineProtein Structure TertiaryAmino acidEnzyme ActivationOxygenEnzymeBiochemistrychemistryHemocyaninsbiology.proteinProtein BindingGene
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Cu(II) complexes with a sulfonamide derived from benzoguanamine. Oxidative cleavage of DNA in the presence of H2O2 and ascorbate

2004

Reaction between benzoguanamine (2,4-diamino-6-phenyl-1,3,5-triazine) and 2-mesitylenesulfonyl chloride leads to formation of a sulfonamide able to form two mononuclear Cu(II) complexes with a CuL(2) stoichiometry. The local environment of the metal cation is a distorted octahedron, with two ligands and two solvent molecules; both complexes crystallize in the monoclinic structure, space group P2(1), with Z=2. In the presence of ascorbate/H(2)O(2,) the two complexes significantly cleavage double-strand pUC18 DNA plasmid. Both complexes exhibit more nuclease efficiency that the copper phenantroline complex. From scavenging reactive oxygen studies we conclude that the hydroxyl radical and a si…

Models MolecularDNA damagechemistry.chemical_elementAscorbic AcidCrystallography X-RayCleavage (embryo)PhotochemistryGuanidinesBiochemistryPeroxideMedicinal chemistryInorganic ChemistryMetalchemistry.chemical_compoundOrganometallic CompoundsMoleculechemistry.chemical_classificationSulfonamidesMolecular StructureTriazinesDNAHydrogen PeroxideCopperSulfonamidechemistryvisual_artvisual_art.visual_art_mediumHydroxyl radicalOxidation-ReductionCopperJournal of Inorganic Biochemistry
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Synergy between quantum dots and 1,10-phenanthroline–copper(ii) complex towards cleaving DNA

2011

We have found that the DNA cleaving activity of quantum dots and 1,10-phenanthroline-Cu(II) complex is significantly enhanced when they are combined.

Models MolecularDNA SuperhelicalPhenanthrolineMetals and Alloyschemistry.chemical_elementDrug SynergismNanotechnologyDNAGeneral ChemistryCopperhumanitiesCatalysisSurfaces Coatings and FilmsElectronic Optical and Magnetic Materialschemistry.chemical_compoundchemistryQuantum dotQuantum DotsOrganometallic CompoundsMaterials ChemistryCeramics and CompositesNucleic Acid ConformationDNA CleavageDNAPhenanthrolinesChemical Communications
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