Search results for "Classification"

showing 10 items of 29475 documents

Synthesis, antiproliferative activity, and in silico insights of new 3-benzoylamino-benzo[ b ]thiophene derivatives

2014

A new series of 3-benzoylamino-5-imidazol-5-yl-benzo[b]thiophenes and the parent amino derivatives were synthesized and screened as antitumor agents. All tested compounds showed concentration-dependent antiproliferative activity profile against HeLa cell line, exhibiting GI50 values in the low micromolar range. The most active compounds were tested in cell cycle perturbation experiments. A rapid accumulation of cells in the G2/M phase, with a concomitant reduction of cells in both the S and G0/G1 phases, was observed, suggesting that cell exposure to selected derivatives produces mitotic failure. To rationalize the biological results, the 3-benzoylamino-benzo[b]thiophenes were analyzed thro…

thiopheneVLAK protocolStereochemistryIn silicoCellAntineoplastic AgentsMechanism of actionHeLa CellHeLaAntineoplastic AgentStructure-Activity Relationship3-Benzoylamino-5-imidazol-4-yl-benzo[b]Settore BIO/10 - BiochimicaDrug DiscoverymedicineHumansMoietyComputer SimulationMitosisCell ProliferationPharmacologyAntitumor agentsbiologyDose-Response Relationship DrugMolecular StructureChemistryDrug Discovery3003 Pharmaceutical ScienceMedicine (all)Cell CycleOrganic ChemistryAntitumor agentG2/M phaseGeneral MedicineSettore CHIM/06 - Chimica OrganicaHeLa cell linebiology.organism_classificationSettore CHIM/08 - Chimica Farmaceuticamedicine.anatomical_structureCell cultureSettore CHIM/03 - Chimica Generale E InorganicathiophenesAntimitotic AgentTopoisomerase-II InhibitorDrug Screening Assays AntitumorHeLa CellsHuman
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Improving statistical classification methods and ecological status assessment for river macroinvertebrates

2016

Aquatic ecosystems are facing a growing number of human-induced stressors and the need to implement more biomonitoring to assess the ecological status of water bodies is eminent. This dissertation aims at providing tools to reduce the costs and improve the accuracy of freshwater benthic macroinvertebrate biomonitoring. To improve the cost-e ciency, we consider automated classi cation and develop a novel classi er suitable for complex macroinvertebrate image data. To enhance the accuracy of macroinvertebrate biomonitoring, we study the statistical properties of the Percent Model A nity index crucial to current Finnish biomonitoring and the factors a ecting these statistics. Finally, we perfo…

tieteellinen luokitteluindeksitbayesilainen menetelmätilastomenetelmätvesiekosysteemitmonitorointiselkärangattomatcurse of dimensionalitydimensioiden kirouspohjaeläimistöautomaatioclassificationbiomonitoringvirheetlajinmääritysekologinen tilabiomonitorointibiological indicesvirheanalyysierror propagationbenthic macroinvertebratesaquatic ecosysytems
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Calcium mediated polyelectrolyte adsorption on like-charged surfaces.

2011

International audience; Monte Carlo simulations within the primitive model of calcium-mediated adsorption of linear and comb polyelectrolytes onto like-charged surfaces are described, focusing on the effect of calcium and polyion concentrations as well as on the ion pairing between polymers and calcium ions. We use a combination of Monte Carlo simulations and experimental data from titration and calcium binding to quantify the ion pairing. The polymer adsorption is shown to occur as a result of surface overcharging by Ca2+ and ion pairing between charged monomers and Ca2+. In agreement with experimental observations, the simulations predict that the polymer adsorption isotherm goes through …

titrationInorganic chemistrychemistry.chemical_element02 engineering and technologyCalcium010402 general chemistry01 natural sciencesIonQuantitative Biology::Cell BehaviorQuantitative Biology::Subcellular ProcessesinterfacesAdsorptionElectrochemistryGeneral Materials ScienceSpectroscopypolyelectrolytechemistry.chemical_classificationQuantitative Biology::BiomoleculesQuantitative Biology::Neurons and CognitionSurface Chemistry and ColloidsSurfaces and InterfacesPolymerPolymer adsorption021001 nanoscience & nanotechnologyCondensed Matter PhysicsPolyelectrolyte0104 chemical sciencesCondensed Matter::Soft Condensed Matter[ PHYS.PHYS.PHYS-CHEM-PH ] Physics [physics]/Physics [physics]/Chemical Physics [physics.chem-ph]chemistryPolyelectrolyte adsorptionChemical physicsadsorptionMonte Carlo SimulationsTitration[PHYS.PHYS.PHYS-CHEM-PH]Physics [physics]/Physics [physics]/Chemical Physics [physics.chem-ph]0210 nano-technologyLangmuir : the ACS journal of surfaces and colloids
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Predicting Individual Differences from Brain Responses to Music using Functional Network Centrality

2022

Individual differences are known to modulate brain responses to music. Recent neuroscience research suggests that each individual has unique and fundamentally stable functional brain connections irrespective of the task they perform. 77 participants’ functional Magnetic Resonance Imaging (fMRI) responses were measured while continuously listening to music. Using a graph-theory-based approach, we modeled whole-brain functional connectivity. We then calculate voxel-wise eigenvector centrality and subsequently use it to classify gender and musical expertise using binary Support Vector Machine (SVM). We achieved a cross-validated classification accuracy of 97% and 96% for gender and musical exp…

toiminnallinen magneettikuvausclassificationfMRIfunctional connectivitynaturalistic paradigmmusiikkipsykologiacentralitykognitiivinen neurotiedeerotyksilöllisyysindividual differenceskuunteleminen2022 Conference on Cognitive Computational Neuroscience
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The link of a finitely determined map germ from R 2 to R 2

2010

Let f: (R2, 0) → (R2, 0) be a finitely determined map germ. The link of f is obtained by taking a small enough representative f: U ⊂ R2 → R2 and the intersection of its image with a small enough sphere Sε1 centered at the origin in R2. We will describe the topology of f in terms of the Gauss word associated to its link.

topological classificationGeneral MathematicsImage (category theory)GaussTopological classificationlink58K4058K65Gauss wordCombinatorics58K15IntersectionTheoryofComputation_ANALYSISOFALGORITHMSANDPROBLEMCOMPLEXITYGermLink (knot theory)Word (group theory)Mathematics
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Honey Bee Pollen in Meagre (Argyrosomus regius) Juvenile Diets: Effects on Growth, Diet Digestibility, Intestinal Traits, and Biochemical Markers Rel…

2020

This research aimed to evaluate the effects of the inclusion of honey bee pollen (HBP) in meagre (Argyrosoumus regius) juveniles&rsquo

total serum proteingrowth trialtrace elementsArgyrosomus regiusmedicine.disease_causemeagre honey bee pollen growth trial digestibility trial TNF-α HSP70 intestinal immunohistochemistry toxic elements trace elements total serum proteinArticleintestinal immunohistochemistry03 medical and health sciencesAnimal sciencePredatory fishIntestinal mucosaSettore AGR/20 - ZoocolturePollenlcsh:Zoologymedicinelcsh:QL1-991toxic elementKeywords: meagreDigestibility trial; Growth trial; Honey bee pollen; HSP70; Intestinal immunohistochemistry; Meagre; TNF-α; Total serum protein; Toxic elements; Trace elementsHSP70030304 developmental biology2. Zero hungertoxic elements0303 health sciencesLamina proprialcsh:Veterinary medicineGeneral Veterinarybiologydigestibility trialfood and beveragestrace elementHistology04 agricultural and veterinary sciencesHoney beebiology.organism_classificationmeagre3. Good healthmedicine.anatomical_structureBee pollenTNF-α040102 fisherieslcsh:SF600-11000401 agriculture forestry and fisheriesAnimal Science and Zoologyhoney bee pollenAnimals
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Evolutionary advantage conferred by an eukaryote-to-eukaryote gene transfer event in wine yeasts

2015

Although an increasing number of horizontal gene transfers have been reported in eukaryotes, experimental evidence for their adaptive value is lacking. Here, we report the recent transfer of a 158-kb genomic region between Torulaspora microellipsoides and Saccharomyces cerevisiae wine yeasts or closely related strains. This genomic region has undergone several rearrangements in S. cerevisiae strains, including gene loss and gene conversion between two tandemly duplicated FOT genes encoding oligopeptide transporters. We show that FOT genes confer a strong competitive advantage during grape must fermentation by increasing the number and diversity of oligopeptides that yeast can utilize as a s…

transfert de gènes[SDV.SA]Life Sciences [q-bio]/Agricultural sciencesBiologiaAliments BiotecnologiaSaccharomycesnitrogensaccharomycesvinVitisBiomassAmino AcidsHomologous Recombinationgene transferFermentation in winemakingGeneticsazote0303 health sciencesVegetal Biologybiologyfot genesfood and beverageseucaryoteBiological EvolutionGlutathioneAgricultural sciencesPhenotypeEukaryotehgt;domestication;competition;nitrogen;oligopeptides;fot genesoligopeptidescompetitionGene Transfer HorizontalGenes FungalSaccharomyces cerevisiaehgtSaccharomyces cerevisiae03 medical and health sciencesdomesticationalcoholic fermentationGenetics[SDV.BV]Life Sciences [q-bio]/Vegetal BiologyFermentacióGene conversionwineMolecular BiologyGeneDiscoveriesEcology Evolution Behavior and Systematics030304 developmental biologyWinefermentation alcooliqueBase Sequence030306 microbiologybiology.organism_classificationYeastFermentationrégion génomiqueBiologie végétaleSciences agricoles
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Aeolian Remobilisation of the 2011-Cordón Caulle Tephra-Fallout Deposit: Example of an Important Process in the Life Cycle of Volcanic Ash

2020

Although volcanic eruptions represent short periods in the whole history of a volcano, the large amount of loose pyroclastic material produced, combined with aeolian processes, can lead to continuous, long-lasting reworking of volcanic products. Driven by wind, these processes significantly influence the geomorphology and prolong the impacts of eruptions on exposed communities and ecosystems. Since such phenomena are of interest to scientists from a range of disciplines (e.g., volcanology, atmospheric and soil sciences), a well-defined, common nomenclature is necessary to optimise the multidisciplinary characterisation of both processes and deposits. We, therefore, first describe ash wind-r…

transport and deposition processestephra falloutlcsh:Qlcsh:Sciencewind remobilisationlithometeor classificationvolcanic ash life cycleFrontiers in Earth Science
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Double copies of blaKPC-3::Tn4401a on an IncX3 plasmid in Klebsiella pneumoniae successful clone ST512 from Italy

2015

ABSTRACT A carbapenem-resistant sequence type 512 (ST512) Klebsiella pneumoniae carbapenemase 3 (KPC-3)-producing K. pneumoniae strain showing a novel variant plasmid content was isolated in Palermo, Italy, in 2014. ST512 is a worldwide successful clone associated with the spread of bla KPC genes located on the IncFIIk pKpQIL plasmid. In our ST512 strain, the bla KPC-3 gene was unusually located on an IncX3 plasmid, whose complete sequence was determined. Two copies of bla KPC-3 ::Tn 4401a caused by intramolecular transposition events were detected in the plasmid.

transposonsequence analysispolymerase chain reactionDrug ResistanceGene DosageSettore MED/42 - Igiene Generale E Applicatabacterial proteinbeta-Lactamaseopen reading framecarbapenemasePlasmidminocyclineplasmid DNAmeropenemPharmacology (medical)geneticscolistincefpodoximeceftazidime610 Medicine & healthCarbapenemBacterialpolymyxin Btimentingene expression regulationbacteriumKlebsiella pneumoniae carbapenemase 3 producing Klebsiella pneumoniae3. Good healthantiinfective agentmicrobial sensitivity testKlebsiella pneumoniaeItalypriority journaltigecyclineMultipleclone (Java method)cefotaxime030106 microbiologyKlebsiella pneumoniae carbapenemase 3tobramycinMicrobial Sensitivity Testsgentamicinpiperacillin plus tazobactamchemistryGene dosageArticleMicrobiology03 medical and health sciencesComplete sequenceClone CellOpen Reading FramesertapenemBacterial Proteinsmultidrug resistanceextensively drug resistant bacteriumAnti-Bacterial AgentcefepimePharmacologylevofloxacinmicrobiologycefoxitinbiochemical phenomena metabolism and nutritionbacterial infections and mycosesVirologyAnti-Bacterial Agents; Bacterial Proteins; Carbapenems; Clone Cells; Drug Resistance Multiple Bacterial; Gene Dosage; Italy; Klebsiella Infections; Klebsiella pneumoniae; Microbial Sensitivity Tests; Open Reading Frames; Plasmids; beta-Lactamases; DNA Transposable Elements; Gene Expression Regulation Bacterial; Pharmacology (medical); Pharmacology; Infectious Diseasesantibiotic sensitivityClone CellsKlebsiella InfectionsceftriaxoneCarbapenemsbacterial genetics0301 basic medicinemolecular cloningSettore MED/07 - Microbiologia E Microbiologia ClinicaKlebsiella pneumoniaeTransposition (music)Drug Resistance Multiple Bacterialpolycyclic compoundsgenetic screeningcell clonecarbapenem derivativeKlebsiella infectionunclassified drugAnti-Bacterial AgentsInfectious Diseasesbacterial genePlasmidsenzymologydoripenemBiologyminimum inhibitory concentrationbeta-Lactamasesbeta lactamaseMechanisms of ResistanceciprofloxacinAmikacin; aztreonam; carbapenemase; cefepime; cefotaxime; cefoxitin; cefpodoxime; ceftazidime; ceftriaxone; ciprofloxacin; colistin; cotrimoxazole; doripenem; doxycycline; ertapenem; gentamicin; imipenem; Klebsiella pneumoniae carbapenemase 3; levofloxacin; meropenem; minocycline; piperacillin plus tazobactam; plasmid DNA; polymyxin B; tigecycline; timentin; tobramycin; unclassified drug; antiinfective agent; bacterial protein; beta lactamase; carbapenem derivative; transposon antibiotic sensitivity; Article; bacterial gene; bacterial genetics; bacterial strain; bacterium; bacterium detection; bacterium isolation; Escherichia coli; extensively drug resistant bacterium; gene dosage; genetic screening; Italy; Klebsiella pneumoniae; Klebsiella pneumoniae carbapenemase 3 producing Klebsiella pneumoniae; minimum inhibitory concentration; molecular cloning; nonhuman; polymerase chain reaction; priority journal; sequence analysis; cell clone; chemistry; drug effects; enzymology; gene expression regulation; genetics; isolation and purification; Klebsiella infection; Klebsiella pneumoniae; metabolism; microbial sensitivity test; microbiology; multidrug resistance; open reading frame; plasmid; transposon Anti-Bacterial Agents; Bacterial Proteins; beta-Lactamases; Carbapenems; Clone Cells; DNA Transposable Elements; Drug Resistance Multiple Bacterial; Gene Dosage; Gene Expression Regulation Bacterial; Italy; Klebsiella Infections; Klebsiella pneumoniae; Microbial Sensitivity Tests; Open Reading Frames; Plasmidsplasmidbacterium isolationEscherichia coliGeneAmikacinbacterium detectionnonhumandoxycyclineisolation and purificationGene Expression Regulation Bacterialbiology.organism_classificationbacterial straincotrimoxazoleOpen reading frameDNA Transposable Elementdrug effectsDNA Transposable Elementsmetabolismaztreonamimipenem
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Helminth Infection of the Loggerhead Sea Turtle Caretta caretta along the Coasts of Sicily and the North West Adriatic Sea

2021

We provide new data on the presence of helminth parasites in 64 individual loggerhead sea turtles Caretta caretta stranded along the coasts of Sicily and the northwest Adriatic Sea between June 2014 and August 2016. The necropsy examination revealed 31 individuals (48.4%) positive for endoparasites, showing a greater prevalence of trematodes than nematodes. In particular, seven species and a single genus of Trematoda (Hapalotrema) and a single species and genus of Nematoda (Kathlania) were identified. Among the Digenea flukes the species with the highest prevalence of infection were Rhytidodes gelatinosus (34.6%) and Hapalotrema sp. (33.3%), while among the Nematoda they were Kathlania sp. …

trematoda; nematoda; loggerhead sea turtle; <i>Caretta caretta</i>; Mediterranean seaVeterinary medicineSettore BIO/05 - ZoologiaZoologyLoggerhead sea turtleDigeneaMediterranean seaSingle speciesGenustrematodaSF600-1100HelminthsnematodaCaretta carettaGeneral Veterinarybiologybiology.organism_classificationbody regionsloggerhead sea turtleQL1-991North westMediterranean seaAnimal Science and ZoologyTrematodaZoology<i>Caretta caretta</i>Animals
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