Search results for "DRY"

showing 10 items of 980 documents

The Effects of Sulphydryl Reagents on the Binding and Mixed Function Oxidation of Hexobarbital in Rat Hepatic Microsomes

1975

1. The effects of the sulphydryl reagents p-chloromercuribenzoate, N-ethylmaleimide and iodoacetamide on the binding spectrum, oxygen consumption and formation of a suspected substrate-cytochrome P-450-oxygen complex for hexobarbital in rat liver microsomes were investigated. 2. The oxygen consumption caused by hexobarbital oxidation was inhibited non-competitively by all three agents, with 50% inhibition at 4 times 10(-5) M for p-chloromercuribenzoate, 3-7 times 10(-4) M for N-ethylmaleimide and 1-9 times 10(-3) M for iodoacetamide. Cysteamine protected and at least partially reversed this inhibition. 3. p-chloromercuribenzoate inhibited the formation of the cytochrome P-450-substrate-oxyg…

MaleCytochromeCysteamineHealth Toxicology and Mutagenesischemistry.chemical_elementHexobarbitalToxicologyBiochemistryOxygenIodoacetamidechemistry.chemical_compoundOxygen ConsumptionCytochrome P-450 Enzyme SystemmedicineAnimalsPharmacologybiologySulfhydryl ReagentsGeneral MedicineRatsHexobarbitalchemistryBiochemistryEthylmaleimideSpectrophotometryReagentMicrosomes LiverIodoacetamidebiology.proteinCysteamineHepatic microsomeChloromercuribenzoatesOxidation-ReductionNADPFunction (biology)medicine.drugXenobiotica
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Beneficial effects of dithiothreitol on relative levels of glutathione S-transferase activity and thiols in oocytes, and cell number, DNA fragmentati…

2006

We analyzed the effect of in vitro aging of mouse oocytes in the presence of dithiothreitol (DTT) on relative levels of glutathione S-transferase (GST) activity and thiols in oocytes, and cell number, DNA fragmentation and cellular allocation to the inner cell mass (ICM) and trophectoderm (TE) lineage at the blastocyst stage. Ovulated oocytes from gonadotropin primed hybrid female mice of 6-8 weeks of age were aged in vitro in the presence of 0, 5, 50, or 500 microM DTT for 6 hr prior to insemination. Relative levels of GST activity and thiols in oocytes were determined by confocal laser scanning microscopy, DNA fragmentation using a single-step TUNEL method, and cell allocation to the ICM …

MaleDNA FragmentationFertilization in VitroBiologyDithiothreitolchemistry.chemical_compoundMiceGeneticsmedicineInner cell massAnimalsPropidium iodideBlastocystSulfhydryl Compoundsreproductive and urinary physiologyGlutathione TransferaseTUNEL assayCell BiologyGlutathioneMolecular biologyIn vitroMice Inbred C57BLDithiothreitolmedicine.anatomical_structureBlastocystchemistryembryonic structuresMice Inbred CBAOocytesDNA fragmentationFemaleDevelopmental BiologyMolecular reproduction and development
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Effectiveness of dapagliflozin versus comparators on renal endpoints in the real world: A multicentre retrospective study.

2019

Aim: To evaluate the changes in renal endpoints in type 2 diabetes patients treated with dapagliflozin versus other glucose-lowering medications in routine clinical practice. Materials and Methods: DARWIN-T2D was a retrospective study conducted at 46 outpatient diabetes clinics in Italy. An automated software collected data on 17 285 patients who received dapagliflozin, glucagon-like peptide-1 receptor agonists, dipeptidyl peptidase-4 inhibitors, or gliclazide, 6751 of whom had a follow-up visit. We analysed changes in albumin excretion rate (AER) and estimated glomerular filtration rate (eGFR). Results: Patients who received dapagliflozin (n = 473) were younger, more obese, and had a poore…

MaleEndocrinology Diabetes and MetabolismType 2 diabetes030204 cardiovascular system & hematologyKidneychemistry.chemical_compound0302 clinical medicineEndocrinologyGlucosidesRetrospective StudieInterquartile rangeMedicineGliclazideDiabetic NephropathiesDapagliflozinPractice Patterns Physicians'Benzhydryl CompoundAged 80 and overdatabase researchMiddle AgedDiabetes and MetabolismTreatment OutcomeItalyFemaleOriginal Articletype 2 diabetesHumanmedicine.drugGlomerular Filtration Ratemedicine.medical_specialtyGlucosideDrug-Related Side Effects and Adverse ReactionsUrologyRenal function030209 endocrinology & metabolism03 medical and health sciencesDiabetes mellitusantidiabetic drug; dapagliflozin; database research; diabetic nephropathy; type 2 diabetes; Internal Medicine; Endocrinology Diabetes and Metabolism; EndocrinologyInternal MedicineHumansHypoglycemic AgentsBenzhydryl CompoundsAgedRetrospective Studiesantidiabetic drugtype 2 diabeteCreatinineHypoglycemic Agentbusiness.industrydiabetic nephropathyRetrospective cohort studyBiomarkerOriginal Articlesdapagliflozinmedicine.diseasechemistryDiabetes Mellitus Type 2Diabetic NephropathieDrug-Related Side Effects and Adverse ReactionbusinessBiomarkersDiabetes, obesitymetabolism
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Fullerenes(nC60) affect the growth and development of the sediment-dwelling invertebrate Chironomus riparius larvae

2015

Abstract The possible toxicity of nanoparticles (NPs) to aquatic organisms needs to be investigated for chronic effects at low concentrations. Chronic effects of carbon NPs, fullerenesC60, on the midges of Chironomus riparius at different life stages on larvae and adult midges were investigated. Sediment associated fullerenesC60 were studied by 10-day growth and 42-day emergence tests with artificial sediment at nominal concentration ranges 0.0004–80 mg/kg dry weight. The body length decreased in the lower tested concentrations (0.0025–20 mg/kg), but the effect vanished with higher concentrations. Delayed emergence rate observed at 0.5 mg/kg. The observed effects correlated with analyzed se…

MaleGeologic SedimentshiiliHealth Toxicology and Mutagenesista1172ved/biology.organism_classification_rank.speciesPopulationmyrkyllisyysToxicologycarbon nanoparticleChironomidaeToxicologyDry weightAnimalssurviaissääsketeducationta116nanoecotoxicologyInvertebrateChironomus ripariusLarvaeducation.field_of_studyChironomus ripariusved/biologyChemistrySedimentGeneral MedicinePollutionekotoksikologiafullereenitBenthic zonenanotoxicityLarvaEnvironmental chemistryToxicitynanohiukkasetFemaleFullerenesWater Pollutants ChemicalEnvironmental Pollution
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Efficacy and safety of dapagliflozin in patients with inadequately controlled type 1 diabetes (DEPICT-1): 24 week results from a multicentre, double-…

2017

Background Dapagliflozin is a sodium-glucose cotransporter-2 inhibitor approved for the treatment of type 2 diabetes. We aimed to assess the efficacy and safety of dapagliflozin as an add-on to adjustable insulin in patients with inadequately controlled type 1 diabetes. Methods DEPICT-1 was a double-blind, randomised, parallel-controlled, three-arm, phase 3, multicentre study done at 143 sites in 17 countries. Eligible patients were aged 18–75 years and had inadequately controlled type 1 diabetes (HbA1c between ≥7·7% and ≤11·0% [≥61·0 mmol/mol and ≤97·0 mmol/mol]) and had been prescribed insulin for at least 12 months before enrolment. After an 8 week lead-in period to optimise diabetes man…

MaleGlycated Hemoglobin AEndocrinology Diabetes and MetabolismType 2 diabetes030204 cardiovascular system & hematologySettore MED/13 - Endocrinologialaw.inventionchemistry.chemical_compound0302 clinical medicineEndocrinologydiabetes dapaglifozinGlucosidesRandomized controlled triallawInsulin03.02. Klinikai orvostanDapagliflozinMiddle AgedDiabetes and MetabolismTreatment OutcomeCombinationDrug Therapy CombinationFemaleType 1Adultmedicine.medical_specialtyDiabetic ketoacidosis030209 endocrinology & metabolismPlacebo03 medical and health sciencesDrug TherapyDiabetes managementDiabetes mellitusInternal medicineDiabetes MellitusInternal MedicinemedicineHumansHypoglycemic AgentsBenzhydryl CompoundsAdult; Benzhydryl Compounds; Body Weight; Diabetes Mellitus Type 1; Drug Therapy Combination; Female; Glucosides; Glycated Hemoglobin A; Humans; Hypoglycemia; Hypoglycemic Agents; Insulin; Male; Middle Aged; Treatment OutcomeAdult; Benzhydryl Compounds; Body Weight; Diabetes Mellitus Type 1; Drug Therapy Combination; Female; Glucosides; Glycated Hemoglobin A; Humans; Hypoglycemia; Hypoglycemic Agents; Insulin; Male; Middle Aged; Treatment Outcome; Internal Medicine; Endocrinology Diabetes and Metabolism; EndocrinologyGlycated HemoglobinType 1 diabetesbusiness.industryBody Weightmedicine.diseaseHypoglycemiaSurgeryDiabetes Mellitus Type 1chemistrybusinessThe Lancet Diabetes & Endocrinology
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Genetic evidence confirms polygamous mating system in a crustacean parasite with multiple hosts.

2014

Mating systems are diverse in animals, notably in crustaceans, but can be inferred from a limited set of parameters. Baeza and Thiel (2007) proposed a model predicting mating systems of symbiotic crustaceans with three host characteristics and the risk of predation. These authors proposed five mating systems, ranging from monogamy to polygynandry (where multiple mating occurs for both genders). Using microsatellite loci, we tested the putatively mating system of the ectoparasite crab Dissodactylus primitivus. We determined the mating frequencies of males and females, parentage assignment (COLONY & GERUD software) as well as the contents of female spermathecae. Our results are globally consi…

MaleGénétique moléculaire[ SDV.MP.PAR ] Life Sciences [q-bio]/Microbiology and Parasitology/Parasitologylcsh:MedicineZoologyMarine BiologyEvolution des espècesBiologyPolygynandryBehavioral EcologySexual Behavior AnimalSpermathecaCrustaceaGenetics[ SDV.EE.IEO ] Life Sciences [q-bio]/Ecology environment/SymbiosisAnimals[SDV.MP.PAR]Life Sciences [q-bio]/Microbiology and Parasitology/ParasitologyMatinglcsh:ScienceSymbiosisBiologySperm competitionreproductive and urinary physiologyGeneticsEvolutionary Biology[ SDE.BE ] Environmental Sciences/Biodiversity and EcologyMultidisciplinaryEcologyAnimal Behaviorlcsh:RMarine EcologyMating systemBrood3. Good healthFemale sperm storagebehavior and behavior mechanismslcsh:QParasitologyFemale[SDE.BE]Environmental Sciences/Biodiversity and EcologyAnimal GeneticsZoologySperm precedenceResearch ArticleMicrosatellite Repeats[SDV.EE.IEO]Life Sciences [q-bio]/Ecology environment/Symbiosis
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4000 years of human dietary evolution in central Germany, from the first farmers to the first elites

2018

Investigation of human diet during the Neolithic has often been limited to a few archaeological cultures or single sites. In order to provide insight into the development of human food consumption and husbandry strategies, our study explores bone collagen carbon and nitrogen isotope data from 466 human and 105 faunal individuals from 26 sites in central Germany. It is the most extensive data set to date from an enclosed geographic microregion, covering 4,000 years of agricultural history from the Early Neolithic to the Early Bronze Age. The animal data show that a variety of pastures and dietary resources were explored, but that these changed remarkably little over time. In the human δ15N h…

MaleHistoryComposite ParticlesPhysiologylcsh:MedicineStone AgeSocial Sciences01 natural sciencesBiochemistryMass SpectrometryIsotopesAnimal ProductsGermanyMedicine and Health Sciences0601 history and archaeologySocioeconomicslcsh:ScienceChildHistory AncientCarbon IsotopesMultidisciplinaryFarmers060102 archaeologyPhysicsEukaryotaGeologyAgriculture06 humanities and the artsAnimal husbandryMiddle AgedBody FluidsGeographyMilkArchaeologyNeolithic PeriodChild PreschoolPhysical SciencesFemaleCollagenAnatomyResearch ArticleAdult010506 paleontologyAtomsMeatAdolescentGeneral Science & TechnologyAnimal TypesRural historyConsumption (sociology)AncientBeveragesAnimal dataYoung AdultBronze AgeBeakerHumansAnimalsDomestic AnimalsPreschoolParticle Physics0105 earth and related environmental sciencesAgedNutritionNitrogen Isotopesbusiness.industrylcsh:RInfant NewbornOrganismsSubsistence agricultureInfantBiology and Life SciencesProteinsGeologic TimeFeeding BehaviorNewbornDietAgricultureFoodEarth Scienceslcsh:QbusinessZoologyCollagens
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Irreversible protein binding of acrylonitrile.

1981

1. After i.p. injection of [2,3-14C]acrylonitrile to rats, a significant portion of radioactivity becomes irreversibly attached to proteins of liver, lung, spleen and other tissues. 2. When rat liver microsomes were incubated with [2,3-14C]acrylonitrile, a time-dependent irreversible binding of radioactivity occurred to microsomal proteins. This binding was not dependent on NADPH. A high extent of binding to heat-inactivated microsomes indicated that no enzymic metabolic step was involved. 3. The irreversible binding of [2,3-14C]acrylonitrile to rat liver microsomal protein in vitro was inhibited by thiols (cysteine, glutathione, mercaptoethanol). The greatest inhibitory potency was display…

MaleHot TemperatureHealth Toxicology and MutagenesisSpleenPlasma protein bindingToxicologyBiochemistryDithiocarbchemistry.chemical_compoundNitrilesmedicineAnimalsSulfhydryl CompoundsPharmacologyAcrylonitrileChemistryGeneral MedicineGlutathioneIn vitroRatsmedicine.anatomical_structureBiochemistryLiverMicrosomeMicrosomes LiverAcrylonitrileDitiocarbSpleenCysteineProtein BindingXenobiotica; the fate of foreign compounds in biological systems
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The dapagliflozin and prevention of adverse outcomes in chronic kidney disease (DAPA-CKD) trial: baseline characteristics

2020

Abstract Background The Dapagliflozin and Prevention of Adverse outcomes in Chronic Kidney Disease (DAPA-CKD; NCT03036150) trial was designed to assess the effect of the sodium–glucose co-transporter 2 (SGLT2) inhibitor dapagliflozin on kidney and cardiovascular events in participants with CKD with and without type 2 diabetes (T2D). This analysis reports the baseline characteristics of those recruited, comparing them with those enrolled in other trials. Methods In DAPA-CKD, 4304 participants with a urinary albumin:creatinine ratio (UACR) ≥200 mg/g and estimated glomerular filtration rate (eGFR) between 25 and 75 mL/min/1.73 m2 were randomized to dapagliflozin 10 mg once daily or placebo. Me…

MaleIGA NEPHROPATHYRATIONALEPROGRESSIONType 2 diabetesurologic and male genital diseasesDiabetic nephropathychemistry.chemical_compoundGlucosidesDESIGNMedicineFAILUREDiabetic NephropathiesDapagliflozinrandomized controlled clinical trialPrognosisfemale genital diseases and pregnancy complications//purl.org/pe-repo/ocde/ford#3.02.13 [https]Cardiovascular DiseasesNephrologyFemalesodium–glucose co-transporter-2 inhibitormedicine.symptomBENAZEPRILGlomerular Filtration Ratemedicine.medical_specialtyFinerenoneINHIBITIONNephropathy//purl.org/pe-repo/ocde/ford#3.02.20 [https]Double-Blind MethodClinical ResearchInternal medicineDiabetes mellitusEND-POINTSHumansBenzhydryl CompoundsRenal Insufficiency ChronicAcademicSubjects/MED00340Sodium-Glucose Transporter 2 InhibitorsAgedTransplantationDECLINEbusiness.industrysodium-glucose co-transporter-2 inhibitordapagliflozinmedicine.diseaseEFFICACYEditor's ChoiceDiabetes Mellitus Type 2chemistryAlbuminuriaORIGINAL ARTICLESbusinesschronic kidney diseaseKidney disease
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A New Method for Revision of Encapsulated Blebs after Trabeculectomy: Combination of Standard Bleb Needling with Transconjunctival Scleral Flap Sutur…

2016

Purpose A simple needling procedure is the standard method for restoring the function of an encapsulated bleb after trabeculectomy. However, postoperative hypotony represents a possible hazard. This study describes a new surgical approach for treating encapsulated blebs with reduced risk of early postoperative hypotony: bleb needling combined with transconjunctival sutures tightening the scleral flap directly. Methods The study included two groups of 23 patients with failing bleb following trabeculectomy: “Group 1” underwent simple needling revision of the filtering bleb and served as a control group, while “Group 2” received needling revision with additional transconjunctival scleral flap …

MaleIntraocular pressureEye Diseasesgenetic structuresmedicine.medical_treatmentlcsh:MedicineGlaucomaOcular HypotensionPathology and Laboratory MedicineVascular MedicineSurgical FlapsCorneaBlisterPostoperative Complications0302 clinical medicineMedicine and Health SciencesGlaucoma surgeryTrabeculectomylcsh:ScienceDry needlingMultidisciplinaryOphthalmic ProceduresMiddle AgedScleramedicine.anatomical_structureFemaleAnatomyScleraResearch Articlemedicine.medical_specialtyOcular AnatomySurgical and Invasive Medical ProceduresHemorrhageTrabeculectomy03 medical and health sciencesSigns and SymptomsMusculoskeletal System ProceduresAdverse ReactionsOcular SystemDiagnostic MedicineOphthalmologymedicineHumansBleb (cell biology)Intraocular PressureAgedOcular HypotensionPharmacologybusiness.industrylcsh:RBiology and Life SciencesGlaucomamedicine.diseaseeye diseasesSurgeryOphthalmology030221 ophthalmology & optometrylcsh:Qsense organsbusiness030217 neurology & neurosurgeryPLOS ONE
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