Search results for "EAD"

showing 10 items of 5911 documents

Pharmacophore-Based Design of New Chemical Scaffolds as Translational Readthrough-Inducing Drugs (TRIDs)

2020

[Image: see text] Translational readthrough-inducing drugs (TRIDs) rescue the functional full-length protein expression in genetic diseases, such as cystic fibrosis, caused by premature termination codons (PTCs). Small molecules have been developed as TRIDs to trick the ribosomal machinery during recognition of the PTC. Herein we report a computational study to identify new TRID scaffolds. A pharmacophore approach was carried out on compounds that showed readthrough activity. The pharmacophore model applied to screen different libraries containing more than 87000 compounds identified four hit-compounds presenting scaffolds with diversity from the oxadiazole lead. These compounds have been s…

010405 organic chemistryChemistryOrganic ChemistryTranslational readthroughNonsense mutationHTVSnonsense mutationOxadiazoleBenzoxazoleRibosomal RNA01 natural sciencesBiochemistrySmall molecule0104 chemical sciencescystic fibrosis010404 medicinal & biomolecular chemistrychemistry.chemical_compoundBiochemistryDrug Discoverypremature termination codonsPharmacophoreDerivative (chemistry)Pharmacophore modeling
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Modelling and Analysis of Flow Rate and Pressure Head in Pipelines

2019

Currently, various approaches with several utilities are proposed to identify damage in the pipeline. The pipeline system is modeled in the form of a distributed parameter system, such that the state space related to the distributed parameter system contains infinite dimension. In this paper, a novel technique is proposed to analyze and model the flow in the pipeline. Important theorems are proposed for testing the observability as well as controllability of the proposed model.

010504 meteorology & atmospheric sciencesComputer sciencePipeline (computing)05 social sciences01 natural sciencesControllabilityPipeline transportPressure headFlow (mathematics)Distributed parameter systemControl theory0502 economics and businessState spaceObservability050207 economics0105 earth and related environmental sciences2019 16th International Conference on Electrical Engineering, Computing Science and Automatic Control (CCE)
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Apparent boudinage in dykes

2004

Intrusive rocks may be arranged in the form of strings of lenses or beads, as found on the Cap de Creus Peninsula, NE Spain, and in the South Finland Migmatite-Granite Belt. These structures first appear to be the result of stretching and boudinage of intrusive sheets or dykes. However, closer examination reveals that they are not boudins, but are instead primary intrusive structures. A detailed study was performed on a swarm of pegmatite intrusions at Cap de Creus. Layering is often continuous between beads, and, in some cases, individual beads exhibit a very irregular shape. These observations are shown to be incompatible with an origin by boudinage. Analogue experiments were used to test…

010504 meteorology & atmospheric sciencesDeformation (mechanics)Irregular shapeMineralogyGeologyBead010502 geochemistry & geophysics01 natural sciences/dk/atira/pure/sustainabledevelopmentgoals/life_below_watervisual_artBoudinageMagmavisual_art.visual_art_mediumSDG 14 - Life Below WaterLayeringPetrologyGeologyPegmatite0105 earth and related environmental sciencesWall rockJournal of Structural Geology
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A record of seafloor methane seepage across the last 150 million years

2020

<p>Methane seepage at the seafloor is a source of carbon in the marine environment and has long been recognized as an important window into the deep geo-, hydro-, and bio-spheres. However, the processes and temporal patterns of natural methane emission over multi-million-year time scales are still poorly understood. The microbially-mediated methane oxidation leads to the precipitation of authigenic carbonate minerals within subseafloor sediments, thus providing a potentially extensive record of past methane emission. In this study, we used data on methane-derived authigenic carbonates to build a proxy time series of seafloor methane emission over the last 150 My. We quantitat…

010504 meteorology & atmospheric sciencesEarth scienceCarbonate mineralslcsh:Medicine010502 geochemistry & geophysics01 natural sciencesMethaneArticlechemistry.chemical_compoundlcsh:ScienceSea level0105 earth and related environmental sciencesTotal organic carbonMultidisciplinarylcsh:RBiogeochemistryCretaceousSeafloor spreadingOceanographyOcean scienceschemistryEnvironmental scienceSeawaterlcsh:QArctic methane releaseGeologyScientific Reports
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Diving into exoplanets: Are water seas the most common?

2019

One of the basic tenets of exobiology is the need for a liquid substratum in which life can arise, evolve, and develop. The most common version of this idea involves the necessity of water to act as such a substratum, both because that is the case on Earth and because it seems to be the most viable liquid for chemical reactions that lead to life. Other liquid media that could harbor life, however, have occasionally been put forth. In this work, we investigate the relative probability of finding superficial seas on rocky worlds that could be composed of nine different, potentially abundant, liquids, including water. We study the phase space size of habitable zones defined for those substance…

010504 meteorology & atmospheric sciencesExtraterrestrial EnvironmentMilky WayOrigin of LifePlanets01 natural sciencesAstrobiologyAbundance (ecology)Planet0103 physical sciencesExobiology010303 astronomy & astrophysicsEcosystem0105 earth and related environmental sciencesProbabilityExoseasModels StatisticalHabitable zoneExoplanetsLead (sea ice)WaterAgricultural and Biological Sciences (miscellaneous)ExoplanetTidal lockingSpace and Planetary ScienceSolventsAstrophysics::Earth and Planetary AstrophysicsRelative probabilityCircumstellar habitable zoneGeology
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Remote sensing of solar-induced chlorophyll fluorescence (SIF) in vegetation: 50 years of progress

2019

Remote sensing of solar-induced chlorophyll fluorescence (SIF) is a rapidly advancing front in terrestrial vegetation science, with emerging capability in space-based methodologies and diverse application prospects. Although remote sensing of SIF – especially from space – is seen as a contemporary new specialty for terrestrial plants, it is founded upon a multi-decadal history of research, applications, and sensor developments in active and passive sensing of chlorophyll fluorescence. Current technical capabilities allow SIF to be measured across a range of biological, spatial, and temporal scales. As an optical signal, SIF may be assessed remotely using high-resolution spectral sensors in …

010504 meteorology & atmospheric sciencesFIS/06 - FISICA PER IL SISTEMA TERRA E PER IL MEZZO CIRCUMTERRESTRE0208 environmental biotechnologySoil ScienceReview02 engineering and technologyPhotochemical Reflectance Index01 natural sciencesArticleGEO/11 - GEOFISICA APPLICATASIF retrieval methodsRadiative transfer modellingRadiative transfer910 Geography & travelComputers in Earth SciencesChlorophyll fluorescence1111 Soil Science1907 GeologyAirborne instruments0105 earth and related environmental sciencesRemote sensingStress detectionGEO/12 - OCEANOGRAFIA E FISICA DELL'ATMOSFERA1903 Computers in Earth SciencesPrimary productionGeologyVegetationPassive optical techniquesField (geography)020801 environmental engineeringGEO/10 - GEOFISICA DELLA TERRA SOLIDA10122 Institute of GeographySun-induced fluorescenceRemote sensing (archaeology)Sun-induced fluorescence Steady-state photosynthesis Stress detection Radiative transfer modelling SIF retrieval methods. Satellite sensors Airborne instruments Applications Terrestrial vegetation Passive optical techniques. ReviewApplicationsTerrestrial vegetationEnvironmental scienceSatelliteSteady-state photosynthesisSatellite sensors
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Enhanced detection of terrestrial gamma-ray flashes by AGILE

2015

At the end of March 2015 the onboard software configuration of the Astrorivelatore Gamma a Immagini Leggero (AGILE) satellite was modified in order to disable the veto signal of the anticoincidence shield for the minicalorimeter instrument. The motivation for such a change was the understanding that the dead time induced by the anticoincidence prevented the detection of a large fraction of Terrestrial Gamma-Ray Flashes (TGFs). The configuration change was highly successful resulting in an increase of one order of magnitude in TGF detection rate. As expected, the largest fraction of the new events has short duration (<100 μs), and part of them has simultaneous association with lightning sfer…

010504 meteorology & atmospheric sciencesGamma rayRadio atmosphericDead time01 natural sciencesLightningWorld wideGeophysics13. Climate action0103 physical sciencesGeneral Earth and Planetary SciencesEnvironmental scienceSatelliteAtmospheric electricity010303 astronomy & astrophysicsShort duration0105 earth and related environmental sciencesRemote sensingGeophysical Research Letters
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Two decades of monitoring in marine debris ingestion in loggerhead sea turtle, Caretta caretta, from the western Mediterranean

2018

Abstract Anthropogenic marine debris is one of the major worldwide threats to marine ecosystems. The EU Marine Strategy Framework Directive (MSFD) has established a protocol for data collection on marine debris from the gut contents of the loggerhead sea turtle (Caretta caretta), and for determining assessment values of plastics for Good Environmental Status (GES). GES values are calculated as percent turtles having more than average plastic weight per turtle. In the present study, we quantify marine debris ingestion in 155 loggerhead sea turtles collected in the period 1995–2016 in waters of western Mediterranean (North-east Spain). The study aims (1) to update and standardize debris inges…

010504 meteorology & atmospheric sciencesGood Environmental StatusOceans and SeasHealth Toxicology and Mutagenesis010501 environmental sciencesToxicology01 natural sciencesLoggerhead sea turtlelaw.inventionEatingMediterranean sealawMarine debrisMediterranean SeaAnimalsWater PollutantsMarine ecosystemTurtle (robot)Ecosystem0105 earth and related environmental sciencesWaste ProductsMarine biologyEcologybiologyGeneral Medicinebiology.organism_classificationPollutionDebrisGastrointestinal ContentsTurtlesFisheryItalySpainEnvironmental sciencePlasticsEnvironmental Pollution
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What is in our seas? Assessing anthropogenic litter on the seafloor of the central Mediterranean Sea

2020

Abstract Abundance, composition, and distribution of macro-litter found on the seafloor of the Strait of Sicily between 10 and 800 m depth has been studied using data collected by bottom trawl surveys MEDITS from 2015 to 2019. Three waste categories based on the items use were considered: single-use, fishing-related and generic-use. Over 600 sampling sites, just 14% of these were litter-free. The five-years average density of seafloor litter was 79.6 items/km2 and ranged between 46.8 in 2019 and 118.1 items/km2 in 2015. The predominant waste type was plastic (58% of all items). Regardless of material type, single-use items were a dominant (60% of items) and widespread (79% of hauls) fractio…

010504 meteorology & atmospheric sciencesHealth Toxicology and MutagenesisFishing010501 environmental sciencesFishing-related litterPlasticToxicologySpatial distribution01 natural sciencesMediterranean seaBaselineMediterranean SeaAnimalsSicily0105 earth and related environmental sciencesSingle-use litterWaste ProductsMaterial typeGeneral MedicinePollutionSeafloor spreadingStrait of SicilyEnvironmental scienceBaseline Fishing-related litter Plastics Single-use litter Strait of SicilyPhysical geographyPlasticsEnvironmental Monitoring
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Anthropogenic lead distribution in soils under arable land and permanent grassland estimated by Pb isotopic compositions

2008

International audience; The role of land use on fate of metals in soils is poorly understood. In this work, we studied the incorporation of lead in two neighboring soils with comparable pedogenesis but under long-term different agricultural management. Distributions of anthropogenic Pb were assessed from concentrations and isotopic compositions determined on bulk horizon samples, systematical 5–10 cm increment samples, and on 24-h EDTA extracts. Minor amounts of anthropogenic lead were detected until 1-m depth under permanent grassland, linked to high earthworm activity. In arable land, exogenous Pb predominantly accumulated at depths <60 cm. Although the proximity between the two sites ens…

010504 meteorology & atmospheric sciencesHealth Toxicology and MutagenesisMETAL POLLUTIONLANTHANUM010501 environmental sciencesToxicology01 natural sciencesanalyse de solIsotopesSoil PollutantsLAND USEIsotope analysis2. Zero hungerbiologySolid Phase ExtractionprairiePb ISOTOPIC COMPOSITIONSAgricultureGeneral Medicineanalyse comparativePollutionSoil contaminationDeposition (aerosol physics)Environmental chemistryFranceArable landEnvironmental MonitoringMETAL POLLUTION;LAND USE;Pb ISOTOPIC COMPOSITIONS;ANTHROPOGENIC;LANTHANUMIndustrial WastePoaceaesol cultivéplombmétal lourdEdetic Acid0105 earth and related environmental sciencesHydrologyLand useEnvironmental and SocietyEarthworm15. Life on landbiology.organism_classificationANTHROPOGENICpollution du sol[SDE.ES]Environmental Sciences/Environmental and SocietyPedogenesisLead13. Climate actionSoil waterEnvironmental scienceEnvironnement et Société
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