Search results for "Euphorbia"

showing 4 items of 34 documents

Ingenane and lathyrane diterpenes from the latex of Euphorbia canariensis

1997

The latex of Euphorbia canariensis yielded, in addition to five known ingenol esters, the ingenane derivatives ingenol 3-angelate 5,20-diacetate and 5-deoxyingenol 3-angelate 20-acetate, and the lathyrane derivatives 2,3-diepiingol 7,12-diacetate 8-benzoate, 2,3-diepiingol 7,12-diacetate 8-isobutyrate and 2-epiingol 3,7,12-triacetate 8-benzoate. The structures were established with the aid of spectroscopic methods, mainly NMR, and molecular mechanics calculations. They were also supported by the results of some chemical transformations.

chemistry.chemical_classificationbiologyStereochemistryEuphorbiaceaePlant ScienceGeneral MedicineHorticulturebiology.organism_classificationBiochemistryEuphorbia canariensisTerpenechemistry.chemical_compoundchemistryTriterpeneOrganic chemistryDiterpeneMolecular BiologyPhytochemistry
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Jatrophane and tigliane diterpenes from the latex of Euphorbia obtusifolia

1999

The latex of Euphorbia obtusifolia var. obtusifolia yielded twelve new diterpene polyesters. Seven of them displayed the jatrophane framework and five were 4-deoxyphorbol esters. A further isolated tigliane diterpene, a derivative of 4-epi-4-deoxyphorbol, was most likely an artifact of the isolation procedure. All structures were established with the aid of spectroscopic methods.

chemistry.chemical_compoundEuphorbiabiologyChemistryStereochemistryEuphorbiaceaePlant ScienceGeneral MedicineHorticultureDiterpenebiology.organism_classificationMolecular BiologyBiochemistry
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Jatrophane derivatives and a rearranged jatrophane from Euphorbia terracina

1998

Abstract The aerial parts of Euphorbia terracina yielded 11 new jatrophane derivatives as well as a further diterpene displaying the novel 1(15 → 14) abeo -jatrophane framework.

chemistry.chemical_compoundbiologychemistryStereochemistryEuphorbiaceaeEuphorbia terracinaPlant ScienceGeneral MedicineHorticultureDiterpenebiology.organism_classificationMolecular BiologyBiochemistryPhytochemistry
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Analysis of Rabbit Vascular Responses to DBI, an Ingol Derivative Isolated from Euphorbia canariensis

1997

Abstract We have analysed the effects of 7,12-O-diacetyl-8-O-benzoil-2,3-diepiingol (DBI), an ingol derivative isolated from E. canariensis, on isometric tension developed by isolated rabbit basilar and carotid arteries. Concentration-response curves to DBI (10−8 - 3 × 10−5 m) were obtained cumulatively in both arteries at resting tension and active tone (KC1, 50 mm). At resting tension, DBI induced a concentration-dependent contraction, which was not inhibited in Ca2+-free medium. H7 (1-(5-isoquinoline sulphonyl)-2-methylpiperazine dichloride) (10−4 m) inhibited the DBI-induced contraction both in basilar and in carotid arteries. Calmidazolium (10−4 m) inhibited the maximum contraction of …

medicine.medical_specialtyContraction (grammar)LatexCarotid Artery CommonMuscle RelaxationPharmaceutical ScienceProstacyclinNitric OxideNitroarginineMuscle Smooth VascularEuphorbia canariensisCalmodulin1-(5-Isoquinolinesulfonyl)-2-MethylpiperazineInternal medicinemedicine.arterymedicineBasilar arteryAnimalsEnzyme InhibitorsProtein Kinase CPharmacologyPlants MedicinalLagomorphabiologyPlant Extractsbiology.organism_classificationEpoprostenolEndocrinologymedicine.anatomical_structureBasilar ArteryCirculatory systemcardiovascular systemCalciumRabbitsDiterpenesMuscle Contractionmedicine.drugBlood vesselArteryJournal of Pharmacy and Pharmacology
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