Search results for "Farm"

showing 10 items of 3554 documents

SOLID LIPID NANOPARTICLES CONTAINING AN ANTIOXIDANT COMPOUND IN ALZHEIMER’S DISEASE

2008

solid lipid nanoparticles drug delivery alzheimer's diseaseSettore CHIM/09 - Farmaceutico Tecnologico Applicativo
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SOLID LIPID NANOPARTICLES (SLNs) CONTAINING FERULIC ACID AGAINST OXIDATIVE STRESS IN NEURODEGENERATIVE DISEASES

2008

solid lipid nanoparticles ferulic acid neurodegenerative diseases.Settore CHIM/09 - Farmaceutico Tecnologico Applicativo
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Somatoforma veģetatīva disfunkcija farmaceita praksē

2020

Ar terminu “somatoforma veģetatīva disfunkcija” (SVD) tiek apzīmēti ķermeņa funkciju un sajūtu traucējumi, gadījumos, kad objektīvs un medicīniski izskaidrojams šo traucējumu iemesls netiek atrasts. Cilvēki ar SVD izjūt dažādus simptomus, piemēram, trauksmi, nemieru, paaugstinātu uzbudināmību, sāpes, kuņģa-zarnu trakta darbības traucējumus, sirds un asinsvadu sistēmas traucējumus, kas izraisa pastāvīgu uztraukumu un diskomfortu. Šie pacienti pārmērīgi meklē medicīnisko palīdzību un mierinājumu, bet viņiem ir grūti pieņemt ne patoloģiskus rezultātus medicīniskajā izmeklēšanā. SVD ir grūti diagnosticējama un prasa vairāku speciālistu palīdzību, ka arī paša cilvēka izturību un līdzestību. SVD …

somatoforma veģetatīva disfunkcijasomatoformie traucējumiFarmācijasomatoform disordersnomierinošie līdzekļisomatoform autonomic dysfunction
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Discovery of a new class of sortase a transpeptidase inhibitors to tackle gram-positive pathogens: 2-(2-phenylhydrazinylidene)alkanoic acids and rela…

2016

A FRET-based random screening assay was used to generate hit compounds as sortase A inhibitors that allowed us to identify ethyl 3-oxo-2-(2-phenylhydrazinylidene)butanoate as an example of a new class of sortase A inhibitors. Other analogues were generated by changing the ethoxycarbonyl function for a carboxy, cyano or amide group, or introducing substituents in the phenyl ring of the ester and acid derivatives. The most active derivative found was 3-oxo-2-(2-(3,4dichlorophenyl)hydrazinylidene)butanoic acid (2b), showing an IC50 value of 50 µM. For a preliminary assessment of their antivirulence properties the new derivatives were tested for their antibiofilm activity. The most active compo…

sortase A; biofilms; 2-(2-phenylhydrazinylidene)alkanoic acid derivatives; FRET0301 basic medicineStaphylococcus aureusStereochemistryPharmaceutical ScienceRelated derivativesmedicine.disease_causeSettore BIO/19 - Microbiologia Generale01 natural sciencesArticleAnalytical Chemistrylcsh:QD241-441Inhibitory Concentration 5003 medical and health scienceschemistry.chemical_compound2-(2-phenylhydrazinylidene)alkanoic acid derivativeAnti-Infective AgentsBacterial Proteinslcsh:Organic chemistryStaphylococcus epidermidisAmideDrug DiscoveryStaphylococcus epidermidismedicineEnzyme InhibitorsPhysical and Theoretical ChemistryIC50Grambiology010405 organic chemistryChemistryBiofilmSortase AOrganic ChemistryBiofilmAminoacyltransferasesbiology.organism_classificationSettore CHIM/08 - Chimica Farmaceutica2-(2-phenylhydrazinylidene)alkanoic acid derivativesPhenylhydrazines0104 chemical sciencesCysteine Endopeptidases030104 developmental biologyChemistry (miscellaneous)Staphylococcus aureusSortase AFRETMolecular Medicinebiofilms
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Valutazione del profilo di rilascio e dell'attività biologica di sostanze attive veicolate mediante sistemi particellari a matrice lipidica

sostanze naturali.MADSettore CHIM/09 - Farmaceutico Tecnologico ApplicativoSLNNLCnanoparticelle lipidiche
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Un ritratto tra ideale e reale: lo speziale siciliano dal XIV al XVI secolo

2008

Lo studio inquadra le tappe della formazione dello speziale siciliano nel tardomedioevo, con un’attenzione a Capitoli e normativa in uso nell’isola. Viene esaminato nel dettaglio un testamento del 1455 che consente di tracciare lo spaccato familiare e sociale di una famiglia di speziali, ricostruendo beni, attività, qualità di vita.

speziale farmacia capitula testamento formazioneSettore M-STO/01 - Storia Medievale
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Profili di speziali siciliani tra XIV e XV secolo

2007

Lo studio, che inquadra il radicamento degli speziali nel tessuto urbano isolano, esamina e rivela il rapporto di scambio tra liquidità e privilegi che i sovrani, tra XIV e XV secolo, sono disposti a concedere: con la conseguenza di una vera e propria scalata sociale che apre agli speziali, in virtù di quella liquidità, nuove prospettive e uno spazio affaristico ampio e variegato che va ben al di là di preparazione e vendita di farmaci.

speziali Palermo farmacopeaSettore M-STO/01 - Storia Medievale
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Polymeric micelles containing squalenoyl chains for the delivery of drugs to the central nervous system

2011

squalenoyl micelles central nervous systemSettore CHIM/09 - Farmaceutico Tecnologico Applicativomicelles Drug delivery system squalenic
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Single intense prenatal stress can differently affect emotional behavior according to the nature of the task. Influence of metyrapone

2007

stremetyraponeSettore BIO/14 - Farmacologia
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Diazepāma ļoti mazu devu ietekme uz telpisko iemācīšanos un atmiņu alcheimera slimības streptozocīna modeļa žurkām

2018

Šī daba mērķis bija pētīt diazepāma (DZP) iespējamo pozitīvo ietekmi uz telpisko iemācīšanos un atmiņu Alcheimera slimības (AD) streptozocīna (STZ) modeļa žurkām, rezultātus iegūstot Morisa ūdens labirinta testā. Iegūtie rezultāti rāda, ka diazepāms gan ļoti mazā devā (0,05 mg/kg), gan vidējā devā (1 mg/kg) būtiski uzlaboja AD modeļa žurku telpisko iemācīšanos un atmiņu. STZ izraisītajā AD modelī iegūtie dati varētu norādīt, ka diazepāma mazu un vidējo devu īstermiņa terapeitiska lietošana varētu būt labvēlīga atmiņas traucējumu novēršanai agrīnajā AD fāzē. Tomēr ir nepieciešami tālāki, padziļināti pētījumi, lai izskaidrotu šajā pētījumā iegūtos efektus.

streptozocīnsAlcheimera slimībaFarmācijaGABAA receptoridiazepāmstelpiskā atmiņa
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