Search results for "Hox"

showing 10 items of 1357 documents

(Trifluoromethoxy)Phenylboronic Acids: Structures, Properties, and Antibacterial Activity.

2021

Three isomers of (trifluoromethoxy)phenylboronic acids were studied in the context of their physicochemical, structural, antimicrobial and spectroscopic properties. They were characterized by 1H, 13C, 11B and 19F NMR spectroscopy. The acidity of all the isomers was evaluated by both spectrophotometric and potentiometric titrations. The introduction of the -OCF3 group influences the acidity, depending, however, on the position of a substituent, with the ortho isomer being the least acidic. Molecular and crystal structures of ortho and para isomers were determined by the single crystal XRD method. Hydrogen bonded dimers are the basic structural motives of the investigated molecules in the sol…

Models MolecularMagnetic Resonance SpectroscopyPotentiometric titrationSubstituentMolecular ConformationPharmaceutical ScienceContext (language use)Crystal structureMicrobial Sensitivity TestsDFTMedicinal chemistryArticleOCF<sub>3</sub>Analytical Chemistrylcsh:QD241-441chemistry.chemical_compoundlcsh:Organic chemistryDrug StabilityIsomerismtrifluoromethoxyDrug DiscoveryMoleculePhysical and Theoretical ChemistryMolecular StructureHydrogen bondOrganic ChemistryBoronic AcidsNMRAnti-Bacterial AgentsantibacterialchemistryChemistry (miscellaneous)Intramolecular forceX-RayMolecular MedicineisomersOCF3Derivative (chemistry)Molecules (Basel, Switzerland)
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Selection on Coding Regions Determined Hox7 Genes Evolution

2003

The important role of Hox genes in determining the regionalization of the body plan of the vertebrates makes them invaluable candidates for evolutionary analyses regarding functional and morphological innovation. Gene duplication and gene loss led to a variable number of Hox genes in different vertebrate lineages. The evolutionary forces determining the conservation or loss of Hox genes are poorly understood. In this study, we show that variable selective pressures acted on Hox7 genes in different evolutionary lineages, with episodes of positive selection occurring after gene duplications. Tests for functional divergence in paralogs detected significant differentiation in a region known to …

Molecular Sequence DataBiologyEvolution MolecularOpen Reading FramesNegative selectionGene DuplicationGene duplicationGene clusterGeneticsAnimalsHumansCoding regionAmino Acid SequenceHox geneMolecular BiologyGenePhylogenyEcology Evolution Behavior and SystematicsGeneticsLikelihood FunctionsGenes HomeoboxGenetic VariationSequence Analysis DNABody planEvolutionary biologyMultigene FamilyVertebratesFunctional divergenceMolecular Biology and Evolution
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Determination of ketosteroid hormones in meat by liquid chromatography tandem mass spectrometry and derivatization chemistry.

2015

A method for the determination and quantification of ketosteroid hormones in meat by mass spectrometry, based on the derivatization of the carbonyl moiety of steroids by O-methylhydroxylamine, is presented. The quantitative assay is performed by means of multiple-reaction-monitoring (MRM) scan mode and using the corresponding labelled species, obtained by reaction with d 3-methoxylamine, as internal standard. The accuracy of the method was established by evaluating artificially spiked samples, obtaining values in the range 90-110%. Recovery tests were performed on blank matrix samples spiked with non-natural steroids including trenbolone and melengestrol acetate. The latter experiment revea…

Multiple reaction monitoringChromatographyMeatMass spectrometrySelected reaction monitoringKetosteroidMass spectrometrySolid-phase microextractionKetosteroidsBiochemistryAnalytical ChemistryMatrix (chemical analysis)chemistry.chemical_compoundTrenbolonechemistryLiquid chromatography–mass spectrometryTandem Mass SpectrometryKetosteroidMethoxylamineUHPLCmedicineDerivatizationSolid Phase Microextractionmedicine.drugAnalytical and bioanalytical chemistry
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CCDC 883070: Experimental Crystal Structure Determination

2018

Related Article: Arri Priimagi, Marco Saccone, Gabriella Cavallo, Atsushi Shishido, Tullio Pilati, Pierangelo Metrangolo and Giuseppe Resnati|2012|Adv.Mater.|24|OP345|doi:10.1002/adma.201204060

NN-dimethyl-4-((2356-tetrafluoro-4-iodophenyl)diazenyl)aniline 4-(2-(4-methoxyphenyl)vinyl)pyridineSpace GroupCrystallographyCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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CCDC 1008820: Experimental Crystal Structure Determination

2015

Related Article: Bernd Elsler, Anton Wiebe, Dieter Schollmeyer, Katrin M. Dyballa, Robert Franke, Siegfried R. Waldvogel|2015|Chem.-Eur.J.|21|12321|doi:10.1002/chem.201501604

N-(3'-t-butyl-2'-hydroxy-45-dimethoxy-5'-methylbiphenyl-2-yl)acetamide methanol solvateSpace GroupCrystallographyCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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Melatonin and phytomelatonin: Chemistry, biosynthesis, metabolism, distribution and bioactivity in plants and animals—an overview

2021

Melatonin is a ubiquitous indolamine, largely investigated for its key role in the regulation of several physiological processes in both animals and plants. In the last century, it was reported that this molecule may be produced in high concentrations by several species belonging to the plant kingdom and stored in specialized tissues. In this review, the main information related to the chemistry of melatonin and its metabolism has been summarized. Furthermore, the biosynthetic pathway characteristics of animal and plant cells have been compared, and the main differences between the two systems highlighted. Additionally, in order to investigate the distribution of this indolamine in the plan…

N-acetyl-5-methoxytrip-tamineIndolesQH301-705.5Exogenous melatoninReviewN-acetyl-5-methoxytriptamineCatalysisInorganic ChemistryMelatoninchemistry.chemical_compoundCluster analysisIndolamineBiosynthesisSettore BIO/10 - BiochimicamedicineDistribution (pharmacology)AnimalsBiology (General)Physical and Theoretical ChemistryQD1-999Molecular BiologySpectroscopyMelatoninOrganic ChemistryGeneral MedicineMetabolismPlantsPlant cellComputer Science ApplicationsBiostimulantChemistryBiochemistrychemistryDietary Supplementsmedicine.drugBiostimulant; Cluster analysis; Dietary supplements; Indolamine; N-acetyl-5-methoxytrip-tamine
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CCDC 705757: Experimental Crystal Structure Determination

2010

Related Article: K.Salorinne, D.P.Weimann, C.A.Schalley, M.Nissinen|2009|Eur.J.Org.Chem.|2009|6151|doi:10.1002/ejoc.200900814

N^1^N^1^'N^1^''N^1^'''-((281420-tetraethyl-6121824-tetramethoxypentacyclo[19.3.1.1^37^.1^913^.1^1519^]octacosa-1(25)3(28)469(27)101215(26)16182123-dodecaene-4101622-tetrayl)tetrakis(oxyethane-21-diyl))tetrabenzene-12-diamine acetonitrile ethanol clathrateSpace GroupCrystallographyCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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Kelfiprim, a new sulpha-trimethoprim combination, versus cotrimoxazole, in the treatment of urinary tract infections: a multicentre, double-blind tri…

1982

A new combination of trimethoprim with a sulphonamide, named Kelfiprim, differs from cotrimoxazole in that: a) the sulpha drug is sulphamethopyrazine instead of sulphamethoxazole; b) the trimethoprim to sulpha ratio is 5:4 instead of 1:5;c) the presence of a long-acting sulphonamide allows the administration of a daily dose of one capsule, following an initial loading dose of two capsules; d) a reduced amount of trimethoprim is given, as compared to cotrimoxazole, without any decrease of efficacy. Kelfiprim [KP] was compared to contrimoxazole [Co] in a multicentre double blind trial. Sixty four patients suffering from acute and chronic infections of the upper and lower urinary tract entered…

NephrologyMalemedicine.medical_specialtySulfamethoxazoleUrologyUrinary systemUrineGastroenterologyLoading doseTrimethoprimDouble blindDouble-Blind MethodInternal medicineSulfanilamidesTrimethoprim Sulfamethoxazole Drug CombinationmedicineHumansClinical Trials as Topicbusiness.industrySulfaleneTrimethoprimSurgeryDrug CombinationsUrinary Tract InfectionsFemalebusinessmedicine.drugUrological research
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Antagonistic roles for Ultrabithorax and Antennapedia in regulating segment-specific apoptosis of differentiated motoneurons in the Drosophila embryo…

2008

The generation of morphological diversity among segmental units of the nervous system is crucial for correct matching of neurons with their targets and for formation of functional neuromuscular networks. However, the mechanisms leading to segment diversity remain largely unknown. We report here that the Hox genes Ultrabithorax (Ubx) and Antennapedia (Antp) regulate segment-specific survival of differentiated motoneurons in the ventral nerve cord of Drosophilaembryos. We show that Ubx is required to activate segment-specific apoptosis in these cells, and that their survival depends on Antp. Expression of the Ubx protein is strongly upregulated in the motoneurons shortly before they undergo a…

Nervous systemCentral Nervous SystemProgrammed cell deathanimal structuresEmbryo NonmammalianApoptosisBiologyAntennapediaDownregulation and upregulationmedicineAnimalsDrosophila ProteinsHox geneMolecular BiologyUltrabithoraxGeneticsHomeodomain ProteinsGene Expression Regulation DevelopmentalCell DifferentiationEmbryonic stem cellCell biologymedicine.anatomical_structureVentral nerve cordembryonic structuresAntennapedia Homeodomain ProteinDrosophilaDevelopmental BiologyTranscription FactorsDevelopment (Cambridge, England)
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The columnar gene vnd is required for tritocerebral neuromere formation during embryonic brain development of Drosophila.

2006

International audience; In Drosophila, evolutionarily conserved transcription factors are required for the specification of neural lineages along the anteroposterior and dorsoventral axes, such as Hox genes for anteroposterior and columnar genes for dorsoventral patterning. In this report, we analyse the role of the columnar patterning gene ventral nervous system defective (vnd) in embryonic brain development. Expression of vnd is observed in specific subsets of cells in all brain neuromeres. Loss-of-function analysis focussed on the tritocerebrum shows that inactivation of vnd results in regionalized axonal patterning defects, which are comparable with the brain phenotype caused by mutatio…

Nervous systemMutantApoptosis0302 clinical medicineMESH: Gene Expression Regulation DevelopmentalDrosophila ProteinsMESH: AnimalsAxonHox geneMESH: MelatoninGenetics0303 health sciencesMESH: Pineal GlandBrainGene Expression Regulation DevelopmentalMESH: Transcription FactorsNeuromerePhenotypeBiological EvolutionCell biologymedicine.anatomical_structureDrosophila melanogasterPhenotypeMESH: Photic StimulationMESH: Body PatterningMESH: MutationMESH: Drosophila ProteinsBiologyMESH: PhenotypeMESH: Drosophila melanogaster03 medical and health sciencesMESH: BrainNeuroblastMESH: EvolutionMESH: Homeodomain ProteinsmedicineAnimalsMESH: Circadian RhythmMolecular Biology030304 developmental biologyBody PatterningHomeodomain ProteinsMESH: HumansMESH: ApoptosisEmbryogenesis[SDV.BBM.BM]Life Sciences [q-bio]/Biochemistry Molecular Biology/Molecular biologyMESH: LightMutationMESH: SerotoninMESH: Seasons030217 neurology & neurosurgeryDevelopmental BiologyTranscription Factors
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