Search results for "Isomer"

showing 10 items of 1308 documents

Induction of apoptosis in human retinoblastoma cells by topoisomerase inhibitors

1998

PURPOSE:To examine the apoptotic effect induced in human retinoblastoma Y79 cells by camptothecin, etoposide, and amsacrine, to examine the effect of these drugs on the expression of many apoptosis-related modulators, and to test the antiapoptotic effect exerted by insulin-like growth factor-I (IGF-I). METHODS:Morphologic features of apoptosis were demonstrated using acridine orange- ethidium bromide staining and electron microscopy. DNA fragmentation was determined by means of an in situ cell detection procedure (TdT-dUTP terminal nick-end labeling [TUNEL]) or by electrophoresis on agarose gels and was quantified by enzyme-linked immunosorbent assay. The expression of apoptosis-related mod…

AmsacrineCyclin-Dependent Kinase Inhibitor p21topoisomeraseCell SurvivalRetinal NeoplasmsRetinoblastomaApoptosisDNA NeoplasmInsulin-Like Growth Factor Binding Protein 3DNA Topoisomerases Type IProto-Oncogene Proteins c-bcl-2CyclinsProto-Oncogene ProteinsDactinomycinTumor Cells CulturedHumansCamptothecinCycloheximideEnzyme InhibitorsTopoisomerase I InhibitorsTumor Suppressor Protein p53DNA DamageEtoposidebcl-2-Associated X Protein
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Application of solid-phase microextraction combined with derivatization to the enantiomeric determination of amphetamines.

2005

Abstract The utility of combining chiral derivatization and solid-phase microextraction (SPME) for the enantiomeric analysis of primary amphetamines by liquid chromatography has been investigated. Different derivatization/extraction strategies have been evaluated and compared using the chiral reagent o -phthaldialdehyde (OPA)– N -acetyl- l -cysteine (NAC) and fibres with a Carbowax-templated resin coating. Amphetamine, norephedrine and 3,4-methylenedioxyamphetamine (MDA) were used as model compounds. On the basis of the results obtained, a new method is presented based on the derivatization of the analytes in solution followed by SPME of the OPA–NAC derivatives formed. The proposed conditio…

AnalyteClinical BiochemistryPhenylpropanolaminePharmaceutical ScienceSolid-phase microextractionAnalytical Chemistrychemistry.chemical_compoundDrug DiscoveryHumansDerivatizationSpectroscopyChromatography High Pressure LiquidAqueous solutionChromatographyExtraction (chemistry)AmphetaminesReproducibility of ResultsStereoisomerismSolutionsSpectrometry FluorescencechemistryReagentCentral Nervous System StimulantsIndicators and ReagentsEnantiomerQuantitative analysis (chemistry)Journal of pharmaceutical and biomedical analysis
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Off-line coupling of multidimensional immunoaffinity chromatography and ion mobility spectrometry: A promising partnership.

2015

The extreme specificity of immunoaffinity chromatography (IAC) columns coupled to the high sensitivity of ion mobility spectrometry (IMS) measurements makes this combination really useful for rapid, selective, and sensitive determination of a high variety of analytes in different samples. The capabilities of the IAC-IMS coupling have been highlighted under three different scenarios: (i) multiclass residue analysis using a single IAC column, (ii) multiclass residue analysis using stacked IAC columns, and (iii) isomer analysis. In the first case, the determination of three strobilurin fungicides - azoxystrobin, picoxystrobin, and pyraclostrobin - in water and strawberry juice was considered, …

AnalyteIon-mobility spectrometryPyridinesAnalytical chemistryWineBiochemistryFragariaSensitivity and SpecificityChromatography AffinityAnalytical Chemistrychemistry.chemical_compoundWineResidue (complex analysis)ChromatographyElutionOrganic ChemistryWaterStereoisomerismGeneral MedicineStrobilurinsFungicides IndustrialFruit and Vegetable JuicesPyrimidineschemistryAcrylatesAzoxystrobinStrobilurinMethacrylatesPyrazolesPyrimethanilCarbamatesJournal of chromatography. A
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Multivariate optimization approach for chiral resolution of drugs using human serum albumin in affinity electrokinetic chromatography-partial filling…

2005

The enantiomeric resolution of chiral compounds using HSA by means of affinity EKC (AEKC)-partial filling technique is the result of a delicate balance between different experimental variables such as protein concentration, running pH (background electrophoretic buffer, protein and compound solutions) and protein solution plug length. In this paper multivariate optimization approaches for chiral separation of four basic drugs (alprenolol, oxprenolol, promethazine and propranolol) using HSA as chiral selector in AEKC-partial filling technique are studied. The experimental conditions to achieve maximum resolution are optimized using the Box-Behnken experimental design. Partial least squares a…

AnalyteResolution (mass spectrometry)Clinical BiochemistryAnalytical chemistryBiochemistryPromethazineChromatography AffinityAnalytical ChemistryElectrokinetic phenomenaPartial least squares regressionmedicineHumansAminesAlprenololSerum AlbuminChromatographyChemistryElectrophoresis CapillaryOxprenololStereoisomerismHuman serum albuminPropranololChiral resolutionElectrophoresisPharmaceutical PreparationsMultivariate AnalysisEnantiomerHydrophobic and Hydrophilic Interactionsmedicine.drugElectrophoresis
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Strategies for the enantiomeric determination of amphetamine and related compounds by liquid chromatography.

2002

This paper summarizes recent research on the stereospecific analysis of amphetamine, its analogs and metabolites, by liquid chromatography. The different methods proposed have been evaluated and compared in terms of resolution power, time of analysis, sensitivity, or potential for automation. Chiral derivatization, followed by separation of the diastereomers formed in achiral chromatographic systems, is still the method preferred for the analysis of amphetamines at trace levels, as derivatization also improves analyte detectability. This is the method of choice for the enantiomeric analysis of amphetamines at the low concentrations typically encountered in biological samples. In recent year…

AnalyteResolution (mass spectrometry)medicine.drug_classBiophysicsBiochemistrySensitivity and Specificitychemistry.chemical_compoundIsomerismmedicineHumansEphedrineDerivatizationAmphetamineChromatography High Pressure LiquidChromatographyStaining and LabelingIllicit DrugsAmphetaminesDiastereomerReproducibility of ResultsDesigner drugSubstance Abuse DetectionchemistryModels ChemicalEnantiomermedicine.drugChromatography LiquidJournal of biochemical and biophysical methods
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Headspace–mass spectrometry determination of benzene, toluene and the mixture of ethylbenzene and xylene isomers in soil samples using chemometrics

2007

A simple and fast method has been developed for the determination of benzene, toluene and the mixture of ethylbenzene and xylene isomers (BTEX) in soils. Samples were introduced in 10 mL standard glass vials of a headspace (HS) autosampler together with 150 microL of 2,6,10,14-tetramethylpentadecane, heated at 90 degrees C for 10 min and introduced in the mass spectrometer by using a transfer line heated at 250 degrees C as interface. The volatile fraction of samples was directly introduced into the source of the mass spectrometer which was scanned from m/z 75 to 110. A partial least squares (PLS) multivariate calibration approach based on a classical 3(3) calibration model was build with m…

Analytical chemistryBTEXXylenesMass spectrometryBiochemistryEthylbenzeneGas Chromatography-Mass SpectrometryMass SpectrometryAnalytical ChemistryChemometricsSoilchemistry.chemical_compoundIsomerismBenzene DerivativesEnvironmental ChemistryBenzeneSpectroscopyChromatographyChromatographyXyleneTemperatureBenzeneTolueneHydrocarbonsBiodegradation EnvironmentalModels ChemicalchemistryCalibrationGas chromatographyTolueneAnalytica Chimica Acta
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Pressure-induced magnetic switching and linkage isomerism in K0.4Fe4[Cr(CN)6]2.8 x 16 H2O: X-ray absorption and magnetic circular dichroism studies.

2008

The effect of applied pressure on the magnetic properties of the Prussian blue analogue K0.4Fe4[Cr(CN)6]2.8 x 16 H2O (1) has been analyzed by dc and ac magnetic susceptibility measurements. Under ambient conditions, 1 orders ferromagnetically at a critical temperature (T(C)) of 18.5 K. Under application of pressure in the 0-1200 MPa range, the magnetization of the material decreases and its critical temperature shifts to lower temperatures, reaching T(C) = 7.5 K at 1200 MPa. Pressure-dependent Raman and Mossbauer spectroscopy measurements show that this striking behavior is due to the isomerization of some Cr(III)-C[triple bond]N-Fe(II) linkages to the Cr(III)-N[triple bond]C-Fe(II) form. A…

Analytical chemistryBiochemistryCatalysisMagnetizationsymbols.namesakeMagneticsColloid and Surface ChemistryIsomerismX-Ray DiffractionChromium CompoundsMössbauer spectroscopyTavernePressureLinkage isomerismCyanidesMagnetic circular dichroismChemistrySpectrum AnalysisX-RaysTemperatureWaterGeneral ChemistryMagnetic susceptibilityX-ray magnetic circular dichroismsymbolsDiamagnetismRaman spectroscopyCrystallizationIron CompoundsJournal of the American Chemical Society
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Spectroscopic Detection and Structure of Hydroxidooxidosulfur (HOSO) Radical, An Important Intermediate in the Chemistry of Sulfur-Bearing Compounds

2013

The rotational spectrum of hydroxidooxidosulfur, HOSO, an intermediate of particular interest in the combustion of sulfur-rich fuels, has been determined to high accuracy from gas-phase measurements. Detection of specific isotopic species using isotopically enriched gases suggests that HOSO is formed in our discharge nozzle via the reaction H + SO2 (+M) → HOSO (+M). A precise experimental r0 geometry has also been derived from the isotopic analysis; HOSO has a cis configuration, but the subtle structural question of its planarity remains unresolved. From the derived spectroscopic constants, in situ and remote sensing for this fundamental radical can now be undertaken in a variety of environ…

Analytical chemistrychemistry.chemical_elementCombustionSulfurGalilean moonsJupitersymbols.namesakechemistrysymbolsMoleculeGeneral Materials ScienceRotational spectroscopyPhysics::Chemical PhysicsPhysical and Theoretical ChemistryCis–trans isomerismEarth (classical element)The Journal of Physical Chemistry Letters
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First isomeric yield ratio measurements by direct ion counting and implications for the angular momentum of the primary fission fragments

2018

We report the first experimental determination of independent isomeric yield ratios using direct ion counting with a Penning trap, which offered such a high resolution in mass that isomeric states could be separated. The measurements were performed at the Ion Guide Isotope Separator On-Line (IGISOL) facility at the University of Jyvaskyla. The isomer production ratios of Ge-81, Y-96,Y-97 Sn-128(,1)30, and Sb-129 in the 25-MeV proton-induced fission of U-na(t) and Th-232 were studied. Three isomeric pairs (Ge-81, Y-96, and Sb-129) were measured for the first time for the U-na(t)(p, f) reaction, while all the reported yield ratios for the Th-232(p, f) reaction were determined for the first ti…

Angular momentumResolution (mass spectrometry)Fission01 natural sciencesIonSubatomär fysikydinreaktiotPrimary (astronomy)0103 physical sciencesSubatomic PhysicsPhysics::Atomic and Molecular ClustersfissionYield ratioPhysics::Atomic PhysicsPhysics::Chemical PhysicsNuclear Experiment010306 general physicsnuclear reactionsPhysicsta114010308 nuclear & particles physicsPenning trapfissioYield (chemistry)Atomic physicsisomer decaysydinfysiikka
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Reactions of platinum(iv)-bound nitriles with isomeric nitroanilines: addition vs. substitution

2012

The platinum(IV) complex trans-[PtCl(4)(EtCN)(2)] reacts smoothly and under mild conditions with isomeric o-, m- and p-nitroanilines (NAs) yielding two different types of products depending on the NA isomer, viz. the nitroaniline complexes cis/trans-[PtCl(4)(NA)(2)] (cis/trans-1-3) and the amidine species trans-[PtCl(4){NH=C(Et)NHC(6)H(4)NO(2)-m}(EtCN)] (4), trans-[PtCl(4){NH=C(Et)NHC(6)H(4)NO(2)-m}(2)] (5) and trans-[PtCl(4){NH=C(Et)NHC(6)H(4)NO(2)-p}(EtCN)] (6). Complexes 4 and 5 undergo cyclometalation, furnishing mer-[PtCl(3){NH=C(Et)NHC(6)H(3)NO(2)-m}(EtCN)] (7) and mer-[PtCl(3){NH=C(Et)NHC(6)H(4)NO(2)-m}{NH=C(Et)NHC(6)H(3)NO(2)-m}] (8), respectively. Moreover, 8 both in the solid stat…

Aniline CompoundsNucleophilic additionOrganoplatinum CompoundsNitrileLigandStereochemistrySolid-statechemistry.chemical_elementMedicinal chemistryNitroanilineInorganic ChemistryAmidinechemistry.chemical_compoundIsomerismchemistryNitrilesMethanolPlatinumta116PlatinumDalton Transactions
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