Search results for "Kynuramine"

showing 2 items of 2 documents

Oxidation of melatonin by oxoferryl hemoglobin: A mechanistic study

2002

Reaction of melatonin with the hypervalent iron centre of oxoferryl hemoglobin, produced in aqueous solution from methemoglobin and H2O2, has been investigated at 37 degrees C and pH 7.4, by absorption spectroscopy. The reaction results in reduction of the oxoferryl moiety with formation of a heme-ferric containing hemoprotein. Stopped-flow spectrophotometric measurements provide evidence that the reduction of oxoferryl-Hb by melatonin is first-order in oxoferryl-Hb and first-order in melatonin. The bimolecular reaction constant at pH 7.4 and 37 degrees C is 112 +/- 1.0 M(-1) s(-1). Two major oxidation products from melatonin have been found by gas chromatography-mass spectroscopy: the cycl…

HemeproteinMagnetic Resonance SpectroscopyTime FactorsKynuraminePhotochemistryBiochemistryMethemoglobinGas Chromatography-Mass SpectrometryMelatoninHemoglobinsReaction rate constantmedicineAnimalsMethemoglobinMelatoninIndole testCyclic compoundChemistryOxidesGeneral MedicineHydrogen PeroxideKineticsYield (chemistry)CattleSpectrophotometry UltravioletHemoglobinChlorineOxidation-Reductionmedicine.drug
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Increase by 5-hydroxykynuramine of spontaneous acetylcholine release from myenteric neurons: mediated by serotonin M receptors

1987

The effects of 5-hydroxykynuramine (5-OH-K) and of 3-(2-amino-5-hydroxyphenyl)-propaneamine (AHPP) on spontaneous and electrically evoked release of [3H]acetylcholine were studied in the guinea-pig myenteric plexus longitudinal muscle preparation preincubated with [3H]choline. 5-OH-K caused a concentration-dependent increase in spontaneous [3H]acetylcholine release (EC50 5.3 microM). This effect was diminished in the presence of a desensitizing concentration of 5-hydroxytryptamine (5-HT). AHPP (1-100 microM) did not affect the spontaneous outflow of [3H]acetylcholine. The electrically evoked release of [3H]acetylcholine was significantly reduced in the presence of 100 microM of either 5-OH-…

MaleAgonistSerotoninmedicine.medical_specialtymedicine.drug_classKynuramineMethiothepinGuinea PigsMyenteric PlexusIn Vitro TechniquesBiologychemistry.chemical_compoundInternal medicinemedicineAnimalsCholineReceptorNeurotransmitterMyenteric plexusPharmacologyPropiophenonesPropylaminesAcetylcholineElectric StimulationEndocrinologychemistryReceptors SerotoninMetitepineFemaleSerotoninAcetylcholinemedicine.drugEuropean Journal of Pharmacology
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