Search results for "MDMA"

showing 10 items of 51 documents

Behavioural and neurotoxic long-lasting effects of MDMA plus cocaine in adolescent mice

2008

The poly-drug pattern is the most common among MDMA users, with cocaine being a frequently associated drug. The aim of the present work was to evaluate the behavioural and neurotoxic long-term effects of exposure during adolescence to MDMA alone or plus cocaine. Mice of 28 to 30 days of age received a treatment of two daily injections of an identical dose of MDMA (5, 10 or 20 mg/kg), alone or plus cocaine (25 mg/kg), for 3 days (6 administrations). Three weeks after receiving MDMA, an increase in the time dedicated by the animals to social contacts with their conspecifics was observed, whilst their behaviour in the elevated plus maze showed no differences from that of non-treated mice. Afte…

MaleSerotoninElevated plus mazemedicine.drug_classDopamineN-Methyl-34-methylenedioxyamphetamineMotor ActivityPharmacologyAnxiolyticBody TemperatureMicechemistry.chemical_compoundCocaineDopaminemental disordersmedicineAnimalsMaze LearningSocial BehaviorNeurotransmitterPharmacologyBehavior AnimalLocal anestheticDopaminergicBrainMDMACorpus StriatumchemistrySerotoninPsychologypsychological phenomena and processesmedicine.drugEuropean Journal of Pharmacology
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Neurochemical Substrates of MDMA Reward: Effects of the Inhibition of Serotonin Reuptake on the Acquisition and Reinstatement of MDMA-induced CPP

2013

Different neurotransmitter brain systems have been implicated in the rewarding effects of 3,4-methylenedioxymetamphetamine (MDMA), including dopamine or serotonin. Serotonin selective reuptake inhibitors (SSRI) are a commonly prescribed therapy for psychiatric disorders, and the SSRI fluoxetine is recommended for MDMA users due to its neuroprotective effect against MDMAinduced neurotoxicity. In the present work, we employed the conditioned place preference (CPP) paradigm to study how the inhibition of serotonin reuptake with fluoxetine affected the rewarding and reinstating effects of MDMA in adolescent male mice. Firstly, we evaluated the motivational effects of fluoxetine (1 and 10 mg/kg)…

MaleSerotoninN-Methyl-34-methylenedioxyamphetaminePharmacologyMicechemistry.chemical_compoundNeurochemicalRewardDopamineFluoxetineConditioning Psychologicalmental disordersDrug DiscoveryAnimalsMedicineNeurotransmitterPharmacologyFluoxetineDose-Response Relationship Drugbusiness.industryMDMAConditioned place preferencechemistryHallucinogensSerotoninbusinessReuptake inhibitorSelective Serotonin Reuptake Inhibitorspsychological phenomena and processesmedicine.drugCurrent Pharmaceutical Design
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Adolescent pre-exposure to ethanol or MDMA prolongs the conditioned rewarding effects of MDMA

2011

Adolescents often take ethanol (EtOH) in combination with MDMA (3,4-methylenedioxymethylamphetamine). In the present work we studied the effect of repeated intermittent adolescent pre-exposure to both drugs on the behavioral and neurochemical effects of MDMA in mice. Sixteen days after pre-treatment, the rewarding and reinstating effects of MDMA in the conditioned place preference (CPP) paradigm were evaluated, along with the levels of biogenic amines, basal motor activity and corticosterone response to different challenges. Pre-exposure to EtOH, MDMA or EtOH+MDMA did not affect the CPP induced by 10mg/kg of MDMA. However, adolescent exposure to EtOH or MDMA increased the duration of the co…

MaleSerotoninmedicine.medical_specialtyDopamineN-Methyl-34-methylenedioxyamphetaminePoison controlExperimental and Cognitive PsychologyStriatumMotor ActivityChoice BehaviorHippocampusDrug Administration ScheduleExtinction PsychologicalMiceBehavioral Neurosciencechemistry.chemical_compoundNeurochemicalRewardCorticosteroneInternal medicineConditioning Psychologicalmental disordersAnimals Outbred StrainsmedicineAnimalsDrug InteractionsCerebral CortexEthanolIllicit DrugsMDMAExtinction (psychology)Hydroxyindoleacetic AcidCorpus StriatumConditioned place preferenceMonoamine neurotransmitterEndocrinologychemistryAnesthesia34-Dihydroxyphenylacetic AcidCorticosteronePsychologypsychological phenomena and processesmedicine.drugPhysiology & Behavior
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Effect of intermittent exposure to ethanol and MDMA during adolescence on learning and memory in adult mice

2012

Abstract Background Heavy binge drinking is increasingly frequent among adolescents, and consumption of 3,4-methylenedioxymethamphetamine (MDMA) is often combined with ethanol (EtOH). The long-lasting effects of intermittent exposure to EtOH and MDMA during adolescence on learning and memory were evaluated in adult mice using the Hebb-Williams maze. Methods Adolescent OF1 mice were exposed to EtOH (1.25 g/kg) on two consecutive days at 48-h intervals over a 14-day period (from PD 29 to 42). MDMA (10 or 20 mg/kg) was injected twice daily at 4-h intervals over two consecutive days, and this schedule was repeated six days later (PD 33, 34, 41 and 42), resulting in a total of eight injections. …

MaleSerotoninmedicine.medical_specialtyMDMA34-Dihydroxyphenylacetic acidDopamineN-Methyl-34-methylenedioxyamphetamineCognitive NeuroscienceBinge drinkingStriatumHippocampuslcsh:RC346-429MiceBehavioral Neurosciencechemistry.chemical_compoundSerotonin AgentsMemoryDopamineSerotonin AgentsInternal medicinemental disordersmedicineAnimalsLearningHippocampus (mythology)Maze Learninglcsh:Neurology. Diseases of the nervous systemBiological PsychiatryBehavior AnimalEthanolResearchMDMAGeneral MedicineHydroxyindoleacetic AcidCorpus StriatumEndocrinologychemistryAnesthesia34-Dihydroxyphenylacetic AcidHebb Williams mazeSerotoninPsychologypsychological phenomena and processesmedicine.drugBehavioral and Brain Functions
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Role of NMDA and AMPA glutamatergic receptors in the effects of social defeat on the rewarding properties of MDMA in mice

2019

Exposure to social stress alters the response to drugs of abuse of experimental animals. Changes in the glutamatergic system seem to play a role in the effects of social defeat stress on the rewarding properties of cocaine and amphetamine. The aim of the present study was to evaluate the involvement of N-methyl-D-aspartate (NMDA) and alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) glutamate receptors in the effects of social defeat on the conditioned place preference induced by 3,4-methylenedioxymethamphetamine (MDMA). Our hypothesis was that changes in these receptors could mediate the effects of social defeat on MDMA reward. Young adult male mice were exposed to an episode…

Maledrug addictionglutamate receptorN-Methyl-34-methylenedioxyamphetamineAMPA receptorPharmacologyReceptors N-Methyl-D-AspartateSocial defeatMice03 medical and health scienceschemistry.chemical_compoundstress0302 clinical medicineRewardConditioning PsychologicalmedicineAnimalsReceptors AMPASocial BehaviorAmphetamine030304 developmental biologySocial stress0303 health sciencesAdrenergic Uptake Inhibitorsbusiness.industryGeneral NeuroscienceMemantineMDMAconditioned place preferenceConditioned place preferencechemistrynervous systemCNQXbusinessExcitatory Amino Acid AntagonistsStress Psychological030217 neurology & neurosurgerymedicine.drug
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The novelty-seeking phenotype modulates the long-lasting effects of adolescent MDMA exposure.

2015

Exposure to drugs such as ethanol or cocaine during adolescence induces alterations in the central nervous system that are modulated by the novelty-seeking trait. Our aim was to evaluate the influence of this trait on the long-term effects of MDMA administration during adolescence on spontaneous behavior and conditioned rewarding effects in adulthood. Adolescent mice were classified as high or low novelty seekers (HNS or LNS) according to the hole-board test and received either MDMA (0, 10 or 20mg/kg PND 33-42) or saline. Three weeks later, having entered adulthood (PND>68), one set of mice performed the elevated plus maze and social interaction tests, while another set performed the condit…

Malemedicine.medical_specialtyElevated plus mazemedicine.drug_classN-Methyl-34-methylenedioxyamphetamineCentral nervous systemPoison controlExperimental and Cognitive PsychologyStriatumMotor ActivityAnxiolyticBehavioral NeuroscienceMiceInternal medicinemental disordersmedicineAnimalsSocial BehaviorAdrenergic Uptake InhibitorsBehavior AnimalNovelty seekingAssociation LearningMDMAEndocrinologymedicine.anatomical_structurePhenotypeAnesthesiaExploratory BehaviorConditioning OperantSerotoninPsychologypsychological phenomena and processesmedicine.drugPhysiologybehavior
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Long-term effects of repeated social stress on the conditioned place preference induced by MDMA in mice.

2015

Previous studies have demonstrated that social defeat stress increases the rewarding effects of psychostimulant drugs such as cocaine and amphetamine. In the present study we evaluated the long-term effects of repeated social defeat (RSD) on the rewarding effects of ±3,4-methylenedioxymethamphetamine (MDMA) hydrochloride in the conditioned place preference (CPP) paradigm. Adolescent and young adult mice were exposed to four episodes of social defeat (on PND 29-40 and PND 47-56, respectively) and were conditioned three weeks later with 1.25 or 10mg/kg i.p. of MDMA (experiment 1). The long-term effects of RSD on anxiety, social behavior and cognitive processes were also evaluated in adult mic…

Malemedicine.medical_specialtyN-Methyl-34-methylenedioxyamphetamineDevelopmental psychologyExtinction PsychologicalSocial defeatMiceAdrenal Cortex HormonesInternal medicinemental disordersmedicineAvoidance LearningAnimalsInterpersonal RelationsYoung adultAmphetamineMaze LearningBiological PsychiatryPharmacologySocial stressAnalysis of VarianceDose-Response Relationship DrugAge FactorsMDMAConditioned place preferenceSocial relationEndocrinologyHallucinogensAnxietyConditioning Operantmedicine.symptomPsychologyReinforcement Psychologypsychological phenomena and processesStress Psychologicalmedicine.drugProgress in neuro-psychopharmacologybiological psychiatry
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MDMA Administration and Heat Shock Proteins Response: Foreseeing a Molecular Link

2010

Molecular and cellular mechanisms of MDMA-induced toxicity have been extensively studied in a number of experimental models. Nevertheless, only few studies investigated the involvement of HSPs ("molecular chaperones") in MDMA organs toxicity. In the present minireview we highlight this subject analysing the results of these studies conducted especially on brain tissue. Despite of it seems obvious that HSPs overexpression is a protective reaction against MDMA treatment, the molecular mechanisms for exerting their action are far to be undiscovered. At the same time, we need of comprehensive studies concerning the whole range of Hsps/chaperones expressions in all organs after acute and chronic…

N-Methyl-34-methylenedioxyamphetamineModels NeurologicalBrainPharmaceutical ScienceMDMABrain tissuePharmacologyBiologyHeat shock proteinmental disordersToxicityHallucinogensmedicineAnimalsHumans34-Methylenedioxy-N-methylamphetamine brain toxicity Hsp27 Hsp32 Hsp60 Hsp70.Heat-Shock ProteinsHeat-Shock Responsepsychological phenomena and processesBiotechnologymedicine.drugCurrent Pharmaceutical Biotechnology
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Involvement of 5-hydroxytryptamine 5-HT3 serotonergic receptors in the acquisition and reinstatement of the conditioned place preference induced by M…

2013

Some MDMA (3,4-methylenedioxymethamphetamine) users develop dependence as a result of chronic consumption. The present study evaluated the role of 5-hydroxytryptamine 5-HT₃ receptors in the acquisition, expression and reinstatement of the conditioned place preference (CPP) induced by MDMA. Adolescent male mice were conditioned with 10 mg/kg of MDMA and then treated with 1 or 3mg/kg of the 5-hydroxytryptamine 5-HT₃ antagonist MDL72222 during acquisition of conditioning (experiment 1), before expression of CPP in a post-conditioning test (experiment 2) or before a reinstatement test (experiment 3). MDL72222 was devoid of motivational effects but blocked acquisition of the MDMA-induced CPP. Mo…

PharmacologyAntagonistMDMAExtinction (psychology)StriatumPharmacologySerotonergicConditioned place preferencenervous systemDopaminemental disordersmedicineSerotoninPsychologypsychological phenomena and processesmedicine.drugEuropean Journal of Pharmacology
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Adolescent pre-exposure to ethanol and 3,4-methylenedioxymethylamphetamine (MDMA) increases conditioned rewarding effects of MDMA and drug-induced re…

2011

Many adolescents often take ethanol (EtOH) in combination with 3,4-methylenedioxymethylamphetamine (MDMA). In the present work, we used a mouse model to study the effect of repeated pre-exposure during adolescence to EtOH (2 g/kg), MDMA (10 or 20 mg/kg) or EtOH + MDMA on the rewarding and reinstating effects of MDMA in the conditioned place preference (CPP) paradigm. Pre-exposure to EtOH, MDMA or both increased the rewarding effects of a low dose of MDMA (1.25 mg/kg). These pre-treatments did not affect the acquisition of the CPP induced by 5 mg/kg of MDMA. However, the CPP was more persistent in mice pre-exposed to both doses of MDMA or to EtOH + MDMA20. After extinction of the CPP induced…

PharmacologyEthanolHomovanillic acidMedicine (miscellaneous)MDMAExtinction (psychology)StriatumPharmacologyConditioned place preferencePsychiatry and Mental healthchemistry.chemical_compoundchemistryDopaminemental disordersmedicineSerotoninpsychological phenomena and processesmedicine.drugAddiction Biology
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