Search results for "Nox"

showing 10 items of 727 documents

Structural and Dynamic Properties of the Homodimeric Hemoglobin from Scapharca inaequivalvis Thr-72→Ile Mutant: Molecular Dynamics Simulation, Low Te…

1998

AbstractMolecular dynamics simulations, low temperature visible absorption spectroscopy, and resonance Raman spectroscopy have been performed on a mutant of the Scapharca inaequivalvis homodimeric hemoglobin, where residue threonine 72, at the subunit interface, has been substituted by isoleucine. Molecular dynamics simulation indicates that in the Thr-72→Ile mutant several residues that have been shown to play a role in ligand binding fluctuate around orientations and distances similar to those observed in the x-ray structure of the CO derivative of the native hemoglobin, although the overall structure remains in the T state. Visible absorption spectroscopy data indicate that in the deoxy …

Absorption spectroscopyProtein subunitDimerResonance Raman spectroscopyMutantBiophysicsHemeSpectrum Analysis Ramanchemistry.chemical_compoundHemoglobinsMutant proteinAnimalsHemeHistidineCarbon MonoxideChemistrySettore BIO/11TemperatureWaterCrystallographyMolluscaSpectrophotometryMutationDimerizationProtein BindingResearch ArticleBiophysical Journal
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Multi-experimental study of micro-structural and mechanical consequences of thermal cycles applied to a martensitic stainless steel « APX4 »

2010

The Direction des Applications Militaires at the Commissariat à l’Énergie Atomique, a French government-funded technological research organisation, selected a low carbon chromium rich martensitic stainless steel (APX4) to manufacture components with high yield strength and ultimate tensile strength. As such, this thesis is developed around three main axes. Firstly, the thesis summarizes the existing bibliography on this steel as well as its neighboring nuances. Secondly, it engages in a precise characterization of the material that is currently used for industrial manufacturing. Finally, this highly experimental work undertakes to observe and interpret the micro-structural and mechanical co…

Acier inoxydable martensitiqueTrempeX4CrNiMo16.5Austénisation[PHYS.COND.CM-GEN] Physics [physics]/Condensed Matter [cond-mat]/Other [cond-mat.other]APX4[PHYS.COND.CM-GEN]Physics [physics]/Condensed Matter [cond-mat]/Other [cond-mat.other]Propriétés mécaniquesNo english keywordsRevenuMétallurgie[ PHYS.COND.CM-GEN ] Physics [physics]/Condensed Matter [cond-mat]/Other [cond-mat.other]
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Modified arabinoxylan-based films

2004

Abstract Oxygen plasma and electron beam irradiation were used to graft hydrophobic substances and by this way, to reduce water vapor permeability (WVP) of arabinoxylan-based (AX-based) films. Stearyl acrylate (SA) and stearyl methacrylate (SM) were used as reactive monomers. The homogeneous AX-based films, which were pre-activated by oxygen plasma and impregnated with a solution of SA before being exposed to an electron beam (EB), had contact angles that increased from 71° (untreated films) to 122° (treated films). A decrease of about 24% in the WVP was obtained and new chemical groupings were observed on the FTIR spectra of these films. Acrylate monomers were also dispersed into the arabi…

AcrylateMaterials scienceFiltration and SeparationMethacrylateBiochemistryHydrophobeContact anglechemistry.chemical_compoundMonomerchemistryChemical engineeringPolymer chemistryArabinoxylanCopolymerGeneral Materials ScienceIrradiationPhysical and Theoretical ChemistryJournal of Membrane Science
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Sul regime classico dell'indefensio nelle azioni nossali

2019

The paper aims to review the prevailing opinion according to which the sanctions of the indefensio in the classical noxal actions for the delicta servorum were the ductio or the missio in bona. For the author this opinion has no foundation in the texts while he thinks that the sanction in this matter was an action sine noxae deditione.

Actiones noxaleindefensioductiomissio in bonaiudicium sine noxae deditione
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Synthesis of novel organic-based fluorophores – Implementation to the design of fluorogenic enzyme substrates based on the principle of in situ synth…

2020

Detection and fluorescence imaging of biologic systems requires the implementation of efficient, robust and easy-to-use tools. Conventional fluorogenic probes currently used in microbiology lack efficiency since they are based on the single chemical modification of a fluorophore bearing an optically tunable reactive group, which often leads to incomplete fluorescence quenching. The main goal of my Ph.D thesis was to develop novel fluorogenic enzymatic substrates based on the "covalent assembly" principle. This approach also named "in situ synthesis" is based on the use of domino reactions to form a fluorescent moiety starting from a "caged" non-fluorescent molecule. In our case, the bioanal…

Activation enzymatique[CHIM.ORGA]Chemical Sciences/Organic chemistryHétéro-XanthènesSynthèse in situHetero-Xanthene dyesQuinoxalinonesIn situ synthesis[CHIM.ORGA] Chemical Sciences/Organic chemistryEnzymatic activationFluorogenic probesSonde fluorogéniquesFluorescence
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Efficacy and safety of glecaprevir/pibrentasvir in renally impaired patients with chronic HCV infection

2019

Background and aims Chronic hepatitis C virus (HCV) infection increases the risk of incident chronic kidney disease (CKD) and progression to end-stage renal disease (ESRD). Previously available direct-acting antiviral regimens are not approved for patients with advanced CKD across all HCV genotypes. Methods EXPEDITION-5 is a phase 3 study to evaluate efficacy and safety of the fixed-dose combination of glecaprevir and pibrentasvir (G/P) for chronic HCV infection (genotype 1 through 6) in adults without cirrhosis or with compensated cirrhosis and with stage 3b, 4 or 5 CKD. Patients received approved duration of G/P according to HCV genotype, cirrhosis status and prior HCV treatment experienc…

AdultCyclopropaneshepatitis C virusmedicine.medical_specialtyAminoisobutyric AcidsPyrrolidinesCirrhosisProlineLactams Macrocyclicmedicine.medical_treatmentAntiviral Agents03 medical and health sciences0302 clinical medicineLeucineQuinoxalinesInternal medicineGenotypeHumansMedicineAdverse effectDialysisSulfonamidesdirect-acting antiviralpangenotypicHepatologychronic kidney disease; cirrhosis; direct-acting antiviral; hepatitis C virus; pangenotypicbusiness.industrycirrhosisGlecaprevirHepatitis C Chronicmedicine.diseasePibrentasvirDrug Combinations030220 oncology & carcinogenesisBronchitisBenzimidazoles030211 gastroenterology & hepatologybusinesschronic kidney diseaseKidney disease
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Multicenter Phase I Study of Erdafitinib (JNJ-42756493), Oral Pan-Fibroblast Growth Factor Receptor Inhibitor, in Patients with Advanced or Refractor…

2018

AbstractPurpose:Here, we report results of the first phase I study of erdafitinib, a potent, oral pan-FGFR inhibitor.Patients and Methods:Patients age ≥18 years with advanced solid tumors for which standard antineoplastic therapy was no longer effective were enrolled (NCT01703481). Parts 2 to 4 employed molecular screening for activating FGFR genomic alterations. In patients with such alterations, two selected doses/schedules identified during part 1 dose-escalation [9 mg once daily and 10 mg intermittently (7 days on/7 days off), as previously published (Tabernero JCO 2015;33:3401-8)] were tested.Results:The study included 187 patients. The most common treatment-related adverse events were…

AdultMale0301 basic medicineCancer Researchmedicine.medical_specialtyAdministration OralAntineoplastic AgentsDrug resistanceGastroenterologyYoung Adult03 medical and health sciencesHyperphosphatemia0302 clinical medicineRefractoryErdafitinibNeoplasmsQuinoxalinesInternal medicinemedicineHumansNeoplasmDosingAdverse effectProtein Kinase InhibitorsAgedNeoplasm StagingAged 80 and overbusiness.industryGenetic VariationMiddle AgedPrognosismedicine.diseaseReceptors Fibroblast Growth FactorTreatment Outcome030104 developmental biologyOncologyTolerabilityDrug Resistance Neoplasm030220 oncology & carcinogenesisRetreatmentPyrazolesFemalebusinessClinical Cancer Research
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Lipid Peroxidation, Nitric Oxide Metabolites, and Their Ratio in a Group of Subjects with Metabolic Syndrome

2014

Our aim was to evaluate lipid peroxidation, expressed as thiobarbituric acid-reactive substances (TBARS), nitric oxide metabolites (nitrite + nitrate) expressed asNOx, and TBARS/NOxratio in a group of subjects with metabolic syndrome (MS). In this regard we enrolled 106 subjects with MS defined according to the IDF criteria, subsequently subdivided into diabetic (DMS) and nondiabetic (NDMS) and also into subjects with a low triglycerides/HDL-cholesterol (TG/HDL-C) index or with a high TG/HDL-C index. In the entire group and in the four subgroups of MS subjects we found an increase in TBARS andNOxlevels and a decrease in TBARS/NOxratio in comparison with normal controls. Regarding all these …

AdultMaleAgingmedicine.medical_specialtySettore MED/09 - Medicina InternaArticle SubjectInflammationNitric OxideThiobarbituric Acid Reactive SubstancesBiochemistryNitric oxideLipid peroxidationchemistry.chemical_compoundInsulin resistanceInternal medicinemedicineTBARSHumanslcsh:QH573-671NitriteNitritesTriglyceridesNOxMetabolic SyndromeNitrateslcsh:CytologyCell BiologyGeneral MedicineMiddle Agedmedicine.diseaseEndocrinologyBiochemistrychemistryLipid Peroxidation Nitric Oxide Metabolites Metabolic SyndromeFemaleLipid Peroxidationmedicine.symptomMetabolic syndromeLipoproteins HDLResearch ArticleOxidative Medicine and Cellular Longevity
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Characterization of blink reflex interneurons by activation of diffuse noxious inhibitory controls in man.

1998

The blink reflex consists of an early, pontine R1-component and a late, medullary R2-component. R1 and R2 can be evoked by innocuous stimuli, but only the R2 also by painful heat, suggesting that the R2 is mediated by wide dynamic range neurons (WDR) of the spinal trigeminal nucleus. Remote noxious stimuli suppress the activity in WDR neurons via activation of diffuse noxious inhibitory controls (DNIC), whereas low-threshold mechanoreceptive neurons (LTM) are unaffected. In order to characterize the trigeminal interneurons of R1 and R2 we investigated the modulation of the blink reflex by remote painful heat. The blink reflex was elicited in 11 healthy subjects by innocuous electrical pulse…

AdultMaleHot TemperatureInterneuronPainInhibitory postsynaptic potentialInterneuronsPhysical StimulationPonsmedicineNoxious stimulusHumansCorneal reflexMolecular BiologyMedulla OblongataBlinkingbusiness.industryFootGeneral NeuroscienceDiffuse noxious inhibitory controlSpinal trigeminal nucleusNeural InhibitionSupraorbital nerveElectric StimulationForearmmedicine.anatomical_structureAnesthesiaSensory ThresholdsFemaleNeurology (clinical)BrainstemTrigeminal Nucleus SpinalbusinessNeuroscienceDevelopmental BiologyBrain research
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C- and Aδ-fiber components of heat-evoked cerebral potentials in healthy human subjects

1999

Feedback-controlled laser heat was used to stimulate the hairy skin of the hand dorsum and forearm, and heat-evoked cerebral potentials were recorded at midline (Fz, Cz, Pz) and temporal (T3, T4) scalp positions. Based on data from primary afferent electrophysiology a stimulus level (40 degrees C) was chosen, which is above C-fiber heat threshold, but clearly below A delta-nociceptor heat threshold in order to excite selectively C-fibers without concomitant excitation of A delta-fibers. Feedback-controlled stepped heat stimuli to 40 degrees C elicited ultralate laser evoked potentials (LEPs) at the vertex in a high proportion of experiments (90%). Estimates of conduction velocity calculated…

AdultMaleHot TemperatureLaser-Evoked PotentialsStimulus (physiology)Nerve conduction velocityFeedbackNerve FibersReference ValuesReaction TimeNoxious stimulusHumansEvoked potentialEvoked PotentialsSkinChemistryLasersBrainMiddle AgedElectrophysiologyAnesthesiology and Pain MedicineNociceptionNeurologyNociceptorFemaleNeurology (clinical)NeurosciencePain
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