Search results for "ODR"

showing 10 items of 434 documents

Intestinal transport of cefuroxime axetil in rats: absorption and hydrolysis processes.

2002

Studies were performed using three cefuroxime axetil solutions (11.8, 118 and 200 microM) in three selected intestinal segments and one cefuroxime axetil solution (118 microM) in colon of anaesthetized rats. First-order absorption rate pseudoconstants, k(ap) and effective permeability coefficients, P(eff), were calculated in each set. Absorption of cefuroxime axetil can apparently be described as a carrier-mediated transport, which obeys Michaelis-Menten and first order kinetics in the proximal segment of the small intestine and a passive diffusion mechanism in the mean and distal segments. The absorption kinetic parameters for cefuroxime axetil were obtained: Vm=0.613 (0.440) microM min-1;…

MaleStereochemistryPharmaceutical ScienceModels BiologicalIntestinal absorptionPharmacokineticsmedicineAnimalsProdrugsIntestinal MucosaRats WistarBiotransformationAntibacterial agentCefuroximeIntestinal permeabilityChromatographyChemistryHydrolysisBiological TransportProdrugmedicine.diseaseSmall intestineCephalosporinsRatsPerfusionmedicine.anatomical_structureIntestinal AbsorptionCefadroxilCefuroximeAlgorithmsmedicine.drugInternational journal of pharmaceutics
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Prenatal exposure to residential air pollution and infant mental development: modulation by antioxidants and detoxification factors.

2011

Background: Air pollution effects on children’s neurodevelopment have recently been suggested to occur most likely through the oxidative stress pathway. Objective: We aimed to assess whether prenatal exposure to residential air pollution is associated with impaired infant mental development, and whether antioxidant/detoxification factors modulate this association. Methods: In the Spanish INfancia y Medio Ambiente (INMA; Environment and Childhood) Project, 2,644 pregnant women were recruited during their first trimester. Nitrogen dioxide (NO2) and benzene were measured with passive samplers covering the study areas. Land use regression models were developed for each pollutant to predict aver…

Malecognitionvegetablesnitrogen dioxideHealth Toxicology and Mutagenesisaromatic hydrocarbonsEnvironmental pollutionvitamin DPrenatal Nutritional Physiological PhenomenaInfants -- CreixementBayley Scales of Infant DevelopmentAntioxidantsPregnancyEnvironmental healthVitamin D and neurologyMedicineHumansPrenatal Nutritional Physiological Phenomenachild developmentPregnancyAir Pollutantsbusiness.industryResearchPublic Health Environmental and Occupational HealthInfantfruitintelligencemedicine.diseaseChild developmentInfants -- AlimentacióConfidence intervalMaternal ExposureEnvironmental chemistrybreast-feedingVitamines en nutrició humanaNodrissons -- AlimentacióFemaleenvironmental pollutionbusinessBreast feedingEnvironmental health perspectives
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Amino Acid Derivatives as Palmitoylethanolamide Prodrugs: Synthesis, In Vitro Metabolism and In Vivo Plasma Profile in Rats

2015

Palmitoylethanolamide (PEA) has antinflammatory and antinociceptive properties widely exploited in veterinary and human medicine, despite its poor pharmacokinetics. Looking for prodrugs that could progressively release PEA to maintain effective plasma concentrations, we prepared carbonates, esters and carbamates at the hydroxyl group of PEA. Chemical stability (pH 7.4) and stability in rat plasma and liver homogenate were evaluated by in vitro assays. Carbonates and carbamates resulted too labile and too resistant in plasma, respectively. Ester derivatives, prepared by conjugating PEA with various amino acids, allowed to modulate the kinetics of PEA release in plasma and stability in liver …

Malelcsh:MedicinePalmitic AcidsChemical synthesisAmidohydrolasesPalmitic acidchemistry.chemical_compoundHydrolysisPharmacokineticsIn vivoAnimalsProdrugsAmino AcidsEnzyme InhibitorsRats Wistarlcsh:Sciencechemistry.chemical_classificationPalmitoylethanolamideMultidisciplinarylcsh:Rfood and beveragesEstersProdrugAmidesAmino acidchemistryBiochemistryEthanolamineslcsh:QResearch ArticlePLOS ONE
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CERAD neuropsychological battery total score in multinational mild cognitive impairment and control populations: the AddNeuroMed study.

2010

An important focus in Alzheimer's disease (AD) research is the development of methods for early diagnosis. Despite progress with some other biomarkers, sensitive and specific neuropsychological measures for identifying subjects in the prodromal phase of AD remain the most promising early diagnostic tool. We evaluated the value of the composite score for the Consortium to Establish a Registry for Alzheimer's disease Neuropsychological Battery (CERAD-NB) in Europeans with mild cognitive impairment (MCI) and in control populations. Baseline clinical data were analyzed from 223 healthy elderly and 224 subjects with MCI from the prospective AddNeuroMed study carried out in Finland, France, Greec…

Malemedicine.medical_specialtyComposite scoreNeuropsychological TestsStatistics NonparametricDevelopmental psychologyProdromal phaseAlzheimer DiseaseInternal medicinemental disordersmedicineHumansRegistriesCognitive impairmentAgedAged 80 and overAnalysis of VarianceGeneral NeuroscienceNeuropsychologyGeneral MedicineHealthy elderlyNeuropsychological batteryEuropePsychiatry and Mental healthClinical PsychologyStatus examinationEarly DiagnosisROC CurveFemaleGeriatrics and GerontologyPsychologyCognition DisordersJournal of Alzheimer's disease : JAD
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Starpdisciplinārie pētījumi medicīnas koledžās : tēžu krājums

2021

Latvijas Universitātes 79. starptautiskās zinātniskās konferences “Starpdisciplinārie pētījumi medicīnas koledžās” tēzes raksturo medicīnas koledžās veikto pētījumu daudzpusību, pētniecības kvalitāti un arī lietišķumu, kas šogad izceļas ar raksturvārdiem “drošība” un “atbildība”. Konferencē prezentēto un diskutēto jautājumu loks ievērojami pārsniedz veselības aprūpē apskatīto jautājumu loku un veicinās studentus, pētniekus un sociālos partnerus aktīvāk sadarboties ne tikai studiju kvalitātes uzlabošanā, bet arī pētniecībā.

Malnutrīcijapacientu apkope:MEDICINE [Research Subject Categories]urīna nesaturēšanaVecmāšu darbība - vēstureDarba vides risks - sociālā aprūpeErgonomika masu praksēmasāžaKlausīšanās prasme (rehabitaloģija)Marfāna sindroms - aprūpes problēmasTiesu medicīnaKlasiskā kāju masāžaStudiju process- medicīnas koledžaDezinfekcijas līdzekļu efektivitāterehabilitācijaHallux valgusvides riskiAutonomija māsu praksēādas un nagu izmaiņasLipidogrammas rādītājiEelpceļu nodrošināšanaMedikamentozā aprūpe pēcoperācijas periodāHospitālās infekcijasOsteoartrīta pacienta dzīves kvalitātes pašnovērtējumsAntibakteriālo līdzekļu ietošanavīrusu izplatībaMotivācija darbam Neatliekamās medicīniskās palīdzības dienestāRoku mikrofloraRecepšu zāļu izsniegšanaKognitīvie traucējumiAtbalsta un izglītošanas programma nedzirdīgām grūtniecēm
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Supuestos metodológicos y epistemológicos del análisis de género en cinco estudios de casos latinoamericanos

2019

MarcelaJuan Antonio estudios de génerogender perspectivemetodologíaestudios de casoperspectiva de género1696-1676 2341 Quaderns de ciències socials 538523 2019 42 7268707 Supuestos metodológicos y epistemológicos del análisis de género en cinco estudios de casos latinoamericanos Jabbaztécnicas de investigaciónresearch techniques 6 21case studiesgender studiesNavajas-PertegásmethodNina MaríaRodríguez del Pino
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Dibujando una nueva cartografía de la colonialidad Sur-Norte en época de crisis: la reproducción de la episteme y el estilo de vida europeo en las mi…

2018

El artículo analiza la migración de cualificados españoles a los espacios de Educación Superior ecuatoriana desde 2010 a 2016, con el objetivo de entender la experiencia de movilidad cualificada española hacia Ecuador. Para ello se ha utilizado una metodología cualitativa a través de entrevistas semiestructuradas a españoles y ecuatorianos que trabajan en los espacios de la Educación Superior. Además, se ha complementado con encuestas online autoadministradas y con observación participante. Se concluye que entre España y Ecuador se han creado espacios de circularidad promovidos por un contexto de crisis económica en España y por una gran inversión en la Educación Superior ecuatoriana. Sin e…

María El artículo analiza la migración de cualificados españoles a los espacios de Educación Superior ecuatoriana desde 2010 a 2016circularidadse ha complementado con encuestas online autoadministradas y con observación participante. Se concluye que entre España y Ecuador se han creado espacios de circularidad promovidos por un contexto de crisis económica en España y por una gran inversión en la Educación Superior ecuatoriana. Sin embargocircularityEspañaJara Rodríguez FariñaEducación SuperiorHigher Education. 81 94:SOCIOLOGÍA [UNESCO]1137-7038 8537 Arxius de sociologia 514142 2018 39 6874488 Dibujando una nueva cartografía de la colonialidad Sur-Norte en época de crisis: la reproducción de la episteme y el estilo de vida europeo en las migraciones cualificadas Norte-Sur hacia Ecuador Pérez Gañáncualificaciónexistiendo un entramado de distintas estrategias y diferentes realidades. EcuadorSpainUNESCO::SOCIOLOGÍAcon el objetivo de entender la experiencia de movilidad cualificada española hacia Ecuador. Para ello se ha utilizado una metodología cualitativa a través de entrevistas semiestructuradas a españoles y ecuatorianos que trabajan en los espacios de la Educación Superior. AdemásRocíoEcuadorqualificationla reproducción de la episteme y el estilo de vida europeo en las migraciones cualificadas Norte-Sur hacia Ecuador Pérez Gañán [1137-7038 8537 Arxius de sociologia 514142 2018 39 6874488 Dibujando una nueva cartografía de la colonialidad Sur-Norte en época de crisis]la movilidad e inserción de las y los españoles en estos espacios no se conforman de manera lineal y homogénea
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Zvaigžņotā Debess: 2010, Rudens (209)

2010

Contents: G.Carevsky, I.Daube. Comet Bennett ; E.Fogels. Srinivasa Ramanujan ; M.Krastiņš. Smallest Planet of the Solar System: a Riddle of Centuries (1st part) ; A.Alksnis, Z.Alksne. Hot Jupiters and Their Retrograde Motion ; V.Karitāns. James Webb Space Telescope. What will it Be? ; K.Salmiņš. GFZ CHAMP Laser Tracking Award to SLR Station Riga ; J.Jansons. Vladimir Afanasjev, Officer of the Baikonur Cosmodrom in the 1970s (concluded) ; J.Limansky. International Year of Astronomy 2009 in Philately. Series EUROPA (2nd sequel) ; J.Dambītis. Centenary of Prominent Latvian Mathematician Ernests Fogels (1910-1985) ; J.Klētnieks. Sketches of History of Astronomy (concluded) ; M.Gills. Public Sun…

Matemātiķim Ernestam Fogelam – 100Starptautiskais astronomijas gads 2009 filatēlijā – sērija EUROPA (2.turpin.)Pirmie cilvēki uz Mēness – pastmarkasAstronomijas profesoram Kārlim Kaufmanim – 100GFZ Atzinība LU AI par CHAMP lāzernovērojumiemKarstie jupiteriPubliskie saules pulksteņi LatvijāMerkurs – gadsimtu mīklaArvīdam Lūsim – 110Trešais debess vērotāju salidojumsZenta Kauliņa (16.02.1914.-18.03.2010.)Astronomijas vēsture – komētu aprakstiIlgonim Vilkam – 50Citplanēta HD 209458b ar komētas astiDžeimsa Veba kosmiskais teleskops JWSTKrišjānim Baronam – 175Astronomiskās parādības - 2010Baikonuras kosmodroma virsnieks Vladimirs AfanasjevsMarss – vēju erozijaSkaitļu 1234589 pieraksti senajās kultūrāsLeonora Roze (5.08.1928-2.07.2010.)Lielo Greizo Ratu spožāko zvaigžņu attālumiLatvijas atklātā skolēnu astronomijas olimpiādeAsteroīds Lutetia un ESA’s Rozeta
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Ruthenium-Containing Block Copolymer Assemblies: Red-Light-Responsive Metallopolymers with Tunable Nanostructures for Enhanced Cellular Uptake and An…

2015

The use of self-assembled nanostructures consisting of red-light-responsive Ru(II)-containing block copolymers (BCPs) for anticancer phototherapy is demonstrated. Three Ru-containing BCPs with different molecular weights are synthesized. Each BCP contains a hydrophilic poly(ethylene glycol) block and an Ru-containing block. In the Ru-containing block, more than half of the side chains are coordinated with [Ru(2,2':6',2''-terpyridine)(2,2'-biquinoline)](2+) , resulting in more than 40 wt% Ru complex in the BCPs. The Ru complex acts as both a red-light-cleavable moiety and a photoactivated prodrug. Depending on their molecular weights, the BCPs assemble into micelles, vesicles, and large comp…

Materials scienceLightStereochemistryCell SurvivalPolymersBiomedical EngineeringPharmaceutical Sciencechemistry.chemical_element02 engineering and technology010402 general chemistry01 natural sciencesMicelleRutheniumPolyethylene GlycolsBiomaterialschemistry.chemical_compoundNeoplasmsSide chainCopolymerMoietyHumansProdrugsMicellesPhototherapy021001 nanoscience & nanotechnologyCombinatorial chemistry0104 chemical sciencesRutheniumNanostructuresMolecular WeightchemistrySelf-assemblyTerpyridine0210 nano-technologyEthylene glycolHydrophobic and Hydrophilic InteractionsHeLa CellsAdvanced healthcare materials
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Near-infrared photochemistry assisted by upconverting nanoparticles

2019

Abstract Upconverting nanoparticles (UCNPs) combine unique optical and imaging properties with high chemical and biological stability. The capability of UCNPs to emit visible light upon near-infrared light excitation, in an anti-Stokes fashion, is extremely attractive for the design of light-responsive nanomaterials whose action can be controlled spatially and temporally. In this chapter, we analyze the most promising approaches developed so far to functionalize the surface of UCNPs with photoactivatable organic and inorganic molecular systems. In particular, we emphasize the key advances in the design of upconverting nanosystems that exploit bioactive transition metal complexes.

Materials sciencePhotochemistryNear infraredNear-infrared spectroscopyOrganic chemistryNanotechnologyMolecular systemsCoordination chemistryNanomaterialsPhotochemotherapySettore CHIM/03 - Chimica Generale E InorganicaUpconverting nanoparticlesLanthanidesProdrugsLight excitationUpconverting nanoparticlesVisible spectrum
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