Search results for "PHOSPHATE"

showing 10 items of 1874 documents

Coordination and Integration of Metabolism in Insect Flight*

1997

Abstract Insect flight is the most energy-demanding activity of animals. It requires the coordination and cooperation of many tissues, with the nervous system and neurohormones controlling the performance and energy metabolism of muscles, and of the fat body, ensuring that the muscles and nerves are supplied with essential fuels throughout flight. Muscle metabolism can be based on several different fuels, the proportions of which vary according to the insect species and the stage in flight activity. Octopamine, which acts as neurotransmitter, neuromodulator or neurohormone in insects, has a central role in flight. It is present in brain, ventral ganglia and nerves, supplying peripheral tiss…

Nervous systemPhysiologyOctopamine (drug)BiologyBiochemistryInsect flightchemistry.chemical_compoundmedicine.anatomical_structureFructose 26-bisphosphatechemistryBiochemistryHemolymphmedicinemedicine.symptomNeurohormonesMolecular BiologyMuscle contractionPhosphofructokinaseComparative Biochemistry and Physiology Part B: Biochemistry and Molecular Biology
researchProduct

The Measurement of Enzyme Activities in the Resting Human Polymorphonuclear Leukocyte — Critical Estimate of a Method

1993

As a system for study, the isolated human polymorphonuclear leukocyte combines the advantages of a quasi-non-invasive preparation with a nearly complete complement of enzymes of carbohydrate and energy metabolism. However, small sample volumes and, in some cases, very low enzyme activities make high demands on sample processing, storage, and performance of continuous measurements, if the enzyme activities are to be measured with acceptable reproducibility. In the presented study several aspects of homogenization, storage, and continuous measurement were scrutinized, to identify critical steps and consider ways of optimizing the method. Polymorphonuclear leukocytes were separated from the bl…

NeutrophilsCitric Acid CycleeducationClinical BiochemistryTransketolaseGranulocytePhotometrychemistry.chemical_compoundCentrifugation Density GradientmedicineHumansCitrate synthaseHexosephosphatesDifferential centrifugationchemistry.chemical_classificationStaining and LabelingbiologyBiochemistry (medical)Deoxycholic acidReproducibility of ResultsGeneral MedicineEnzyme assayEnzymesmedicine.anatomical_structureEnzymeBiochemistrychemistrybiology.proteinGlycolysisGlycogenHomogenization (biology)Clinical Chemistry and Laboratory Medicine
researchProduct

Metabolic profiling reveals distinct variations linked to nicotine consumption in humans--first results from the KORA study.

2008

Exposure to nicotine during smoking causes a multitude of metabolic changes that are poorly understood. We quantified and analyzed 198 metabolites in 283 serum samples from the human cohort KORA (Cooperative Health Research in the Region of Augsburg). Multivariate analysis of metabolic profiles revealed that the group of smokers could be clearly differentiated from the groups of former smokers and non-smokers. Moreover, 23 lipid metabolites were identified as nicotine-dependent biomarkers. The levels of these biomarkers are all up-regulated in smokers compared to those in former and non-smokers, except for three acyl-alkyl-phosphatidylcholines (e.g. plasmalogens). Consistently significant r…

Nicotinemedicine.medical_specialtyPublic Health and Epidemiology/Environmental HealthMetabolitelcsh:MedicineBiologyPharmacologyCohort StudiesNicotinechemistry.chemical_compoundInternal medicineDiabetes and Endocrinology/EndocrinologyGene expressionmedicineMetabolomeCluster AnalysisHumansAlkylglycerone-phosphate synthaselcsh:Sciencechemistry.chemical_classificationAlkyl and Aryl TransferasesMultidisciplinarySmokinglcsh:RLipid metabolismPublic Health and Epidemiology/Global HealthChemical Biology/Small Molecule ChemistryEnzymeEndocrinologychemistryBiochemistry/Small Molecule ChemistryGlycerophospholipidMetabolomePhosphatidylcholineslcsh:Qbiology.geneMental Health/Personality DisordersBiomarkersResearch Articlemedicine.drugPLoS ONE
researchProduct

Effects of ouabain on human bronchial muscle in vitro

2003

The effects of ouabain, an inhibitor of the plasmalemmal Na(+)/K(+)-ATPase activity, were examined in human isolated bronchus. Ouabain produced concentration-dependent contraction with -logEC(50)=7.16+/-0.11 and maximal effect of 67+/-4% of the response to acetylcholine (1 mM). Ouabain (10 microM)-induced contraction was epithelium-independent and was not depressed by inhibitors of cyclooxygenase and lipoxygenase, antagonists of muscarinic, histamine H(1)-receptors and alpha-adrenoceptors, or neuronal Na(+) channel blockade. The inhibition of ouabain contraction in tissues bathed in K(+)-free medium, and the inhibition by ouabain of the K(+)-induced relaxation confirm that the contractile a…

NitroprussideCromakalimmedicine.medical_specialtySodium-Hydrogen ExchangersTime FactorsInositol PhosphatesMuscle RelaxationVasodilator AgentsBronchiIn Vitro TechniquesOuabainMembrane Potentialschemistry.chemical_compoundSodium Potassium Chloride Symporter InhibitorsInternal medicineMuscarinic acetylcholine receptormedicineHumansVasoconstrictor AgentsNa+/K+-ATPaseOuabainInositol phosphateProtein Kinase CPharmacologychemistry.chemical_classificationForskolinColforsinIsoproterenolMuscle SmoothGeneral MedicineCalcium Channel BlockersAcetylcholineAmilorideEndocrinologychemistryCalciumSodium-Potassium-Exchanging ATPaseHistamineAcetylcholineHistaminemedicine.drugNaunyn-Schmiedeberg's Archives of Pharmacology
researchProduct

NANC inhibitory neurotransmission in mouse isolated stomach: Involvement of nitric oxide, ATP and vasoactive intestinal polypeptide

2003

1. The neurotransmitters involved in NANC relaxation and their possible interactions were investigated in mouse isolated stomach, recording the motor responses as changes of endoluminal pressure from whole organ. 2. Field stimulation produced tetrodotoxin-sensitive, frequency-dependent, biphasic responses: rapid transient relaxation followed by a delayed inhibitory component. 3. The inhibitor of the synthesis of nitric oxide (NO), L-NAME, abolished the rapid relaxation and significantly reduced the slow relaxation. Apamin, blocker of Ca 2+-dependent K + channels, or ADPβS, which desensitises P 2y purinoceptors, reduced the slow relaxation to 2-8 Hz, without affecting that to 16-32 Hz or the…

NitroprussideMuscle RelaxationNANC inhibitory neurotransmitterNitric OxideSynaptic TransmissionSettore BIO/09 - FisiologiaGastric relaxationMiceAdenosine TriphosphateAdrenergic FiberChymotrypsinEnzyme InhibitorThionucleotideCholinergic FiberPharmacologyDose-Response Relationship DrugAnimalIn Vitro TechniqueMouse stomachStomachNitric Oxide DonorElectric StimulationATPVIPAdenosine DiphosphateMice Inbred C57BLNG-Nitroarginine Methyl EsterApaminReceptors Vasoactive Intestinal PeptideNitric Oxide SynthaseVasoactive Intestinal Peptide
researchProduct

BANΔIT: B’‐factor Analysis for Drug Design and Structural Biology

2020

The analysis of B‐factor profiles from X‐ray protein structures can be utilized for structure‐based drug design since protein mobility changes have been associated with the quality of protein‐ligand interactions. With the BANΔIT (B’‐factor analysis and ΔB’ interpretation toolkit), we have developed a JavaScript‐based browser application that provides a graphical user interface for the normalization and analysis of B’‐factor profiles. To emphasize the usability for rational drug design applications, we have analyzed a selection of crystallographic protein‐ligand complexes and have given exemplary conclusions for further drug optimization including the development of a B’‐factor‐supported pha…

Normalization (statistics)Source codeComputer scienceBioinformaticsmedia_common.quotation_subjectDrug designB-factorMolecular modelingWeb BrowserJavaScriptcomputer.software_genre01 natural sciences03 medical and health sciencesStructural BiologyFactor (programming language)Drug DiscoveryApplication NoteHumansProtein flexibilityProtease Inhibitors030304 developmental biologycomputer.programming_languagemedia_commonGraphical user interface0303 health sciencesbusiness.industrySARS-CoV-2Organic ChemistryComputational BiologyUsabilityAdenosine Monophosphate0104 chemical sciencesComputer Science ApplicationsCOVID-19 Drug Treatment010404 medicinal & biomolecular chemistryDrug DesignMolecular MedicineData miningPharmacophorebusinesscomputerMolecular Informatics
researchProduct

Anodic layers formed on steel in phosphate buffer solution

1986

In-situ gamma scattering and ex-situ conversion electron Mossbauer, and Auger spectroscopy were applied to investigate anodic layers on steel. Samples treated in the active potential range in phosphate buffer solution show a Fe(II)-phosphate deposit on the surface. After treatment in the passive potential region, only Fe3+was found to exist in the oxide layer. The passive layer does not consist of stoichiometric oxidic phases.

Nuclear and High Energy PhysicsAuger electron spectroscopyMaterials scienceInorganic chemistryOxideCondensed Matter PhysicsPhosphateAtomic and Molecular Physics and Opticschemistry.chemical_compoundchemistryMössbauer spectroscopyPhysical and Theoretical ChemistryThin filmSpectroscopyLayer (electronics)StoichiometryHyperfine Interactions
researchProduct

A CEMS-study of the passive layer on iron and steel

1988

From AES, ICEMS, and DCEMS experiments it was concluded that the passive layer formed on steel in a phosphate buffer consists of γ-FeOOH. Its thickness increases from 0.5 to 3.5 nm throughout the passive region. It is covered by noncorrelated layers of a precipitate and an adsorbate.

Nuclear and High Energy PhysicsMaterials sciencePhosphate buffered salineMetallurgyPhysical and Theoretical ChemistryCondensed Matter PhysicsLayer (electronics)Atomic and Molecular Physics and OpticsHyperfine Interactions
researchProduct

Photoaffinity cross-linking of F1ATPase from spinach chloroplasts by 3'-arylazido-beta-alanyl-8-azido ATP.

1994

UV irradiation of the ATPase (CF1) from spinach chloroplasts in the presence of 3'-arylazido-beta-alanyl-8-azido ATP (8,3'-DiN3ATP) results in a nucleotide-dependent inactivation of the enzyme and in a nucleotide-dependent formation of alpha-beta cross-links. The results demonstrate an interfacial localization of the nucleotide binding sites on CF1.

Nucleotide binding siteAzidesChloroplastsStereochemistryPhotochemistryAffinity labelATPaseBiophysicsBiochemistryChloroplastF1ATPasechemistry.chemical_compoundAdenosine TriphosphateStructural BiologyVegetablesGeneticsBinding siteChenopodiaceaeInterfacial localizationMolecular BiologyPhotoaffinity cross-linkingchemistry.chemical_classificationbiologyfood and beveragesAffinity LabelsCell Biologybiology.organism_classificationChloroplastProton-Translocating ATPasesEnzymeCross-Linking Reagentschemistrybiology.proteinSpinach chloroplastAdenosine triphosphateFEBS letters
researchProduct

Stability of parenteral nutrition admixtures containing organic phosphates

1995

The use of organic phosphates to avoid calcium phosphate precipitation in parenteral nutrition mixtures has been proposed. The purpose of this study was to evaluate the stability of total parenteral nutrition admixtures containing glucose-1-phosphate or glycerol phosphate as the phosphate source over 3 days. Three parenteral nutrition admixtures, each containing glucose-1-phosphate (30.0 mmol), glycerol phosphate (31.4 mmol) or inorganic phosphate (30.0 mmol), and their corresponding aqueous phases were prepared in 3-L ethylene vinyl acetate plastic bags and infusion bottles, and stored at 5 +/- 1 degrees C or 22 +/- 3 degrees C without light protection. Physical stability analysis and samp…

Nutrition and DieteticsAqueous solutionChromatographybusiness.industryPrecipitation (chemistry)Ethylene-vinyl acetateCritical Care and Intensive Care MedicinePhosphatechemistry.chemical_compoundCreamingParenteral nutritionBiochemistrychemistryDynamic light scatteringEmulsionMedicinebusinessClinical Nutrition
researchProduct