Search results for "RAPTA"

showing 4 items of 4 documents

Frontiers of metal-coordinating drug design

2020

INTRODUCTION: The occurrence of metal ions in biomolecules is required to exert vital cellular functions. Metal-containing biomolecules can be modulated by small-molecule inhibitors targeting their metal-moiety. As well, the discovery of cisplatin ushered the rational discovery of metal-containing-drugs. The use of both drug types exploiting metal–ligand interactions is well established to treat distinct pathologies. Therefore, characterizing and leveraging metal-coordinating drugs is a pivotal, yet challenging, part of medicinal chemistry. AREA COVERED: Atomic-level simulations are increasingly employed to overcome the challenges met by traditional drug-discovery approaches and to compleme…

DrugaromataseComputer sciencemedia_common.quotation_subject1.1 Normal biological development and functioningChemistry PharmaceuticalCellular functionsCYP450Antineoplastic AgentsComputational biologyLigandsQM/MMArticleruthenium drug03 medical and health sciences0302 clinical medicinebreast cancerUnderpinning researchCoordination ComplexesRAPTADrug Discoverymetal-binding inhibitorsHumansComputer SimulationPharmacology & Pharmacy030304 developmental biologymedia_commonQM0303 health sciencesMetallodrugPharmacology and Pharmaceutical Sciencesmetallo-beta-lacatamasesMMprostate cancermolecular dynamicsChemistry5.1 PharmaceuticalsMetals030220 oncology & carcinogenesisDrug DesignPharmaceuticalGeneric health relevanceDevelopment of treatments and therapeutic interventions
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Data from: Phylogenomics of Lophotrochozoa with consideration of systematic error

2021

Phylogenomic studies have improved understanding of deep metazoan phylogeny and show promise for resolving incongruences among analyses based on limited numbers of loci. One region of the animal tree that has been especially difficult to resolve, even with phylogenomic approaches, is relationships within Lophotrochozoa (the animal clade that includes molluscs, annelids, and flatworms among others). Lack of resolution in phylogenomic analyses could be due to insufficient phylogenetic signal, limitations in taxon and/or gene sampling, or systematic error. Here, we investigated why lophotrochozoan phylogeny has been such a difficult question to answer by identifying and reducing sources of sys…

Helobdella robustaGlycera dibranchiataMytilus edulisAnnelidaEntalina tetragonaLeptochiton asellusCerebratulus marginatusLoxosomella cf. viviparaGraptacme eboreaLineus longissimusmedicine and health careClymenella torquataRuditapes philippinarumNucella lapillusHaliotis rufescenslong branch attractionPlatyzoaBarentsia gracilisPriapulus caudatusLineus ruberAlitta virenssaturationProchaetoderma californicumLife SciencesPinctada fucataSchistosoma mansoniPolyzoaCephalothrix hongkongensisRhyssoplax olivaceusLoxosoma pectinaricolaPhascolosoma agassiziiAdineta vagaDrosophila melanogasterEntoproctaBugula neritinaPhoronis vancouverensisMedicineNovocrania anomalaVillosa lienosaDaphnia pulexSagitta sp.Pectinaria gouldiiSymbion americanusNuculana pernulaSepia esculentaEnucula tenuisSolemya velumLineus lacteusTubulanus polymorphus-StruckGnathostomula paradoxaBoccardia proboscideaMacellomenia schanderiLaevipilina hyalinaTubulanus polymorphus-HalanychBryozoaPomatoceros lamarckiiSepioteuthis lessonianaParanemertes peregrinaMalacobdella grossaHemithiris psittaceaLeptochiton rugatusTrochozoaBrachionus plicatilisSpathoderma clenchiLaqueus californicusPatella vulgataLottia giganteaCrepidula fornicataPhoronidaAplysia californicaGlottidia pyramidataPhoronis psammophilaSchmidtea mediterraneaAlexandromenia crassaBrachiopodaMegadasys sp.Octopus vulgarisCapitella teletaNeomenia carinatacompositional heterogeneityNemerteaPhenacolepas pulchellaGadila tolmieiMolluscaMacrodasys sp.Crassostrea gigasPedicellina cernuaTaenia pisiformisDosidicus gigasCephalothrix linearisSpiralia
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Data from: Phylogenomics of Lophotrochozoa with consideration of systematic error

2016

Phylogenomic studies have improved understanding of deep metazoan phylogeny and show promise for resolving incongruences among analyses based on limited numbers of loci. One region of the animal tree that has been especially difficult to resolve, even with phylogenomic approaches, is relationships within Lophotrochozoa (the animal clade that includes molluscs, annelids, and flatworms among others). Lack of resolution in phylogenomic analyses could be due to insufficient phylogenetic signal, limitations in taxon and/or gene sampling, or systematic error. Here, we investigated why lophotrochozoan phylogeny has been such a difficult question to answer by identifying and reducing sources of sys…

Helobdella robustaGlycera dibranchiataMytilus edulisAnnelidaEntalina tetragonaLeptochiton asellusCerebratulus marginatusLoxosomella cf. viviparaGraptacme eboreaLineus longissimusmedicine and health careClymenella torquataRuditapes philippinarumNucella lapillusHaliotis rufescenslong branch attractionPlatyzoaBarentsia gracilisPriapulus caudatusLineus ruberAlitta virenssaturationProchaetoderma californicumPinctada fucataSchistosoma mansoniLife sciencesPolyzoaCephalothrix hongkongensisRhyssoplax olivaceusLoxosoma pectinaricolaPhascolosoma agassiziiAdineta vagaDrosophila melanogasterEntoproctaBugula neritinaPhoronis vancouverensisMedicineNovocrania anomalaVillosa lienosaDaphnia pulexSagitta sp.Pectinaria gouldiiSymbion americanusNuculana pernulaSepia esculentaEnucula tenuisSolemya velumLineus lacteusTubulanus polymorphus-StruckGnathostomula paradoxaBoccardia proboscideaMacellomenia schanderiLaevipilina hyalinaTubulanus polymorphus-HalanychBryozoaPomatoceros lamarckiiSepioteuthis lessonianaParanemertes peregrinaMalacobdella grossaHemithiris psittaceaLeptochiton rugatusTrochozoaBrachionus plicatilisSpathoderma clenchiLaqueus californicusPatella vulgataLottia giganteaCrepidula fornicataPhoronidaAplysia californicaGlottidia pyramidataPhoronis psammophilaSchmidtea mediterraneaAlexandromenia crassaBrachiopodaMegadasys sp.Octopus vulgarisCapitella teletaNeomenia carinatacompositional heterogeneityNemerteaPhenacolepas pulchellaGadila tolmieiMolluscaMacrodasys sp.Crassostrea gigasPedicellina cernuaTaenia pisiformisDosidicus gigasCephalothrix linearisSpiralia
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Ķīnas politiskā un ekonomiskā interese Baltijas jūras reģionā

2020

Bakalaura darba tēma ir “Ķīnas politiskā un ekonomiskā interese Baltijas jūras reģionā”. Darba mērķis ir izpētīt Ķīnas politiskās un ekonomiskās intereses Baltijas jūras reģionā, kā arī aplūkot kādi iekšēji un ārēji faktori varētu būt vadījuši līdzšinējo Ķīnas pieeju šajā reģionā. Par darba teorētisko bāzi tiks izmantota sinerģija starp defensīvā neoreālisma un konstruktīvisma teorijām, autoram tā cenšoties parādīt gan materiālos, gan ideoloģiskos apsvērumus Ķīnas rīcībai un interesēm.

neoreālismsĶīnaBRIBaltijas jūras reģionsstraptautiskās attiecībasPolitikas zinātne
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