Search results for "RIMI"

showing 10 items of 3981 documents

Rational design of covalently bridged [FeIII2MIIO] clusters

2010

We are reporting the first supramolecular dimeric units of basic carboxylates. The neutral [FeIII 2MIIO] motif for different 3d M metals is covalently bound through 2,2′-bipyrimidine. We have structurally characterized the hexanuclear clusters and the related trinuclear building blocks. Their magnetic properties have been fully analyzed and DFT calculations have been performed as a supplementary tool. All results evidence a weak antiferromagnetic interaction through the bpym bridge between isolated spin ground states (in some examples) arising from intra-Fe 2MO core exchange couplings. Fil: Alborés, Pablo. Johannes Gutenberg Universitat Mainz; Alemania. Consejo Nacional de Investigaciones C…

ChemistryOtras Ciencias Químicasbasic carboxylateCiencias QuímicasRational designSupramolecular chemistrybipyrimidineInorganic Chemistrycovalently linkComputational chemistryCovalent bondAntiferromagnetismmagnetic propertiesSpin (physics)CIENCIAS NATURALES Y EXACTASDalton Transactions
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In silico, spectroscopic, and biological insights on annelated pyrrolo[3,2-e]pyrimidines with antiproliferative activity

2013

The in silico COMPARE analysis was performed on 8-[3-(piperidino)propyl]-4,10-dimethyl-9-phenyl-6-(methylsulfanyl)-3,4-dihydropyrimido[1,2-c]pyrrolo[3,2-e]pyrimidin-2(8H)-one, a compound with promising antiproliferative activity, previously synthetized and screened against a panel of 60 human tumor cell lines. The results evidenced that this compound matches the biological properties of Chromomycin A3 and Actinomycin D, known drugs with high DNA binding affinity. Prompted by such results, a thorough spectroscopic investigation of its DNA aqueous solutions was performed, with the aim to verify its DNA-binding properties. DNA groove-binding interaction was assigned by UV-vis spectrophotometri…

ChemistryStereochemistrySettore CHIM/03 - Chimica Generale E InorganicaIn silicoSettore BIO/10 - BiochimicaDrug DiscoveryPharmaceutical ScienceMolecular MedicineAnticancer drugs DNA interactive drugs COMPARE analysis Annelated pyrrolo-pyrimidines UV-vis DNA titrations Circular Dichroism Ethidium bromide displacement assay Cell CycleSettore CHIM/08 - Chimica Farmaceutica
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Preclinical and clinical evidence of activity of pazopanib in solitary fibrous tumour

2014

Abstract Background To explore the activity of pazopanib in solitary fibrous tumour (SFT). Patients and methods In a preclinical study, we compared the activity of pazopanib, sorafenib, sunitinib, regorafenib, axitinib and bevacizumab in a dedifferentiated-SFT (DSFT) xenotransplanted into Severe Combined Immunodeficiency (SCID) mice. Antiangiogenics were administered at their reported optimal doses when mean tumour volume (TV) was 80 mm3. Drug activity was assessed as TV inhibition percentage (TVI%). From May 2012, six consecutive patients with advanced SFT received pazopanib, on a national name-based programme. In one case sunitinib was administered after pazopanib failure. Results In the …

Chemotherapy; Pazopanib; Sarcoma; Solitary fibrous tumour; Sunitinib; Tyrosine kinase; Administration Oral; Adult; Aged; Angiogenesis Inhibitors; Animals; Antibodies Monoclonal Humanized; Antineoplastic Agents; Bevacizumab; Humans; Imidazoles; Indazoles; Indoles; MAP Kinase Signaling System; Male; Mice SCID; Middle Aged; Neoplasm Transplantation; Niacinamide; Phenylurea Compounds; Pyridines; Pyrimidines; Pyrroles; Receptor Platelet-Derived Growth Factor beta; Solitary Fibrous Tumors; Sulfonamides; Transplantation Heterologous; Vascular Endothelial Growth Factor Receptor-2; Cancer Research; Oncology; Medicine (all)OncologyMaleCancer ResearchIndolesAxitinibPyridinesPyridinemedicine.medical_treatmentSolitary fibrous tumourAdministration OralAngiogenesis InhibitorsMice SCIDPharmacologyPyrroleAntineoplastic Agentchemistry.chemical_compoundMiceSolitary Fibrous TumorChemotherapy; Pazopanib; Sarcoma; Solitary fibrous tumour; Sunitinib; Tyrosine kinase; Cancer Research; Oncology; Medicine (all)Transplantation HeterologouMonoclonalSunitinibHumanizedSulfonamidesHeterologousSunitinibMedicine (all)ImidazolesSarcomaMiddle AgedSorafenibPlatelet-Derived Growth Factor betaAxitinibBevacizumabOncologySolitary Fibrous TumorsAdministrationAngiogenesis InhibitorHumanmedicine.drugReceptorPhenylurea CompoundSorafenibOralAdultNiacinamidemedicine.medical_specialtyIndazolesBevacizumabMAP Kinase Signaling SystemTransplantation HeterologousAntineoplastic AgentsSulfonamideAntibodies Monoclonal HumanizedSCIDAntibodiesReceptor Platelet-Derived Growth Factor betaPazopanibInternal medicineRegorafenibmedicineAnimalsHumansChemotherapyPyrrolesImidazoleTyrosine kinaseAgedChemotherapyTransplantationAnimalbusiness.industryPhenylurea CompoundsPazopanibmedicine.diseaseChemotherapy; Pazopanib; Sarcoma; Solitary fibrous tumour; Sunitinib; Tyrosine kinase; Administration Oral; Adult; Aged; Angiogenesis Inhibitors; Animals; Antibodies Monoclonal Humanized; Antineoplastic Agents; Axitinib; Bevacizumab; Humans; Imidazoles; Indazoles; Indoles; MAP Kinase Signaling System; Male; Mice SCID; Middle Aged; Neoplasm Transplantation; Niacinamide; Phenylurea Compounds; Pyridines; Pyrimidines; Pyrroles; Receptor Platelet-Derived Growth Factor beta; Solitary Fibrous Tumors; Sorafenib; Sulfonamides; Sunitinib; Transplantation Heterologous; Vascular Endothelial Growth Factor Receptor-2Vascular Endothelial Growth Factor Receptor-2IndazolePyrimidinesPyrimidinechemistryIndolebusinessProgressive diseaseNeoplasm Transplantation
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L’analyse de la criminalité à Chicago : de nouvelles perspectives offertes par l’économétrie spatiale à une question ancienne

2015

International audience

ChicagoEconométrieCriminalité[ SHS.ECO ] Humanities and Social Sciences/Economies and finances[SHS.ECO] Humanities and Social Sciences/Economics and Finance[SHS.ECO]Humanities and Social Sciences/Economics and FinanceComputingMilieux_MISCELLANEOUS
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The Relevance of Sexual Biographies in Individuals Convicted of Child Sexual Abuse Offenses for the Development of Pedosexual Interests and Sexual Re…

2020

In the literature concerning the etiology of pedosexual interests, the potential role of early sexual experiences in childhood and adolescence has been discussed. Several studies demonstrated a link between own sexually abusive experiences in childhood and sexual offending later in life which tends to be even stronger for pedosexual offenders. Furthermore, some findings indicate associations between other developmental factors and deviant sexual interests in adulthood. For the present study, sexual biographical data of N = 223 imprisoned men convicted of sexual offenses against children from Austria was analyzed to retrospectively examine whether own sexually abusive experiences and non-abu…

Child abuse050103 clinical psychologyrecidivismRecidivismchild abuse05 social sciencesrisk assessmentsexual offenderBF1-990PedophiliapedophiliaChild sexual abuse050501 criminologyRelevance (law)Psychology0501 psychology and cognitive scienceschild molesterPsychologysexual reoffending0505 lawClinical psychologySexual Offending
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Does Childhood Psychological Abuse Contribute to Intimate Partner Violence Victimization? An Investigation Using the Childhood Experience of Care and…

2018

International audience; Although psychological abuse is recognized as a particularly insidious form of child abuse, research on the impact of this type of abuse related to intimate partner violence (IPV) is scant. This study examined the contribution of childhood psychological abuse to IPV in female victims and non-victims. Furthermore, it investigated the role of cumulative abuse in predicting IPV. The study included 38 women victims of IPV and 40 non-IPV women. All participants were investigated using the Childhood Experience of Care and Abuse Interview (CECA); the Revised Conflict Tactics Scale (CTS2) and the IPV History Interview were used to assess IPV in the last year and lifetime, re…

Child abuseCECA intervieweducation[SHS.PSY]Humanities and Social Sciences/PsychologyIntimate Partner Violencebehavioral disciplines and activities[SHS]Humanities and Social SciencesChildhood maltreatment5. Gender equalitySettore M-PSI/08 - Psicologia Clinicamental disordersSettore M-PSI/07 - Psicologia DinamicaHumans0501 psychology and cognitive scienceschildhood maltreatment family violence intimate partner violence psychological abuse CECA interview.Child AbusePsychological abuseChildApplied PsychologyCrime VictimsConflict tactics scale050901 criminology05 social sciencesBullyingsocial sciences16. Peace & justiceIntervention planningFamily violenceEmotional Abuse3. Good healthClinical PracticePsychological abuseClinical PsychologyDomestic violencepopulation characteristicsFemale0509 other social sciencesPsychology050104 developmental & child psychologyClinical psychology
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Poly-Victimization in Polish Adolescents: Risk Factors and the Moderating Role of Coping.

2018

This study aimed to investigate the prevalence of poly-victimization in Polish adolescents and assess factors associated with poly-victimization risk across different ecological levels. This study further examined whether coping styles could moderate the impact of poly-victimization on emotional well-being. Participants were 454 adolescents, aged between 13 and 19 years, from an urban region of Poland. Adolescents completed self-report measures assessing community, school, and family risks, along with a peer nomination task measuring social preference. Teachers also completed a measure assessing adolescent problem behaviors. Findings revealed that the majority of the sample (70%) experience…

Child abuseFamily managementMaleCoping (psychology)anything related to child abuseAdolescentchild abuseetiologyeducationSocial preferencesDevelopmental psychologyYoung AdultRisk FactorsDistractionAdaptation PsychologicalPrevalenceHumans0501 psychology and cognitive scienceshealth care economics and organizationsApplied PsychologyCrime VictimsProblem Solvingcultural contextsHigh rateProblem Behavior050901 criminology05 social sciencesLife satisfactionSocial Supportsocial sciencesModerationhumanitiesClinical PsychologyAdolescent BehaviorbullyingFemalePoland0509 other social sciencesPsychology050104 developmental & child psychologyClinical psychologyJournal of interpersonal violence
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Childhood adversities and distress - The role of resilience in a representative sample.

2016

While adverse childhood experiences have been shown to contribute to adverse health outcomes in adulthood, specifically distress and somatic symptoms, few studies have examined their joint effects with resilient coping style on adult adjustment. Hence, we aim to determine the association between resilient coping and distress in participants with and without reported childhood adversities. A representative German community sample (N = 2508) between 14-92 years (1334 women; 1174 men) was examined by the short form of the Childhood Trauma Questionnaire, the Brief Resilience Coping Scale, standardized scales of distress and somatoform symptoms. Childhood adversity was associated with reduced ad…

Child abuseMaleCoping (psychology)Emotionslcsh:MedicinePoison controlSocial SciencesCriminologyAnxietySuicide preventionPediatrics0302 clinical medicineSociologyChild and adolescent psychiatryMedicine and Health SciencesPsychologyPublic and Occupational HealthChild Abuselcsh:ScienceChildAged 80 and overChild PsychiatryMultidisciplinaryDepressionTraumatic Injury Risk FactorsPost-Traumatic Stress DisorderChild HealthMiddle AgedResilience PsychologicalAnxiety DisordersDistressFemaleCrimePsychologyResearch ArticleAdultmedicine.medical_specialtyAdolescentNeuropsychiatric DisordersNeuroses03 medical and health sciencesSocial supportInjury preventionMental Health and PsychiatrymedicineHumansAdultsPsychiatryAgedMood Disorderslcsh:RBiology and Life Sciences030227 psychiatryAge GroupsPeople and Placeslcsh:QPopulation Groupings030217 neurology & neurosurgeryPloS one
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Neighborhood characteristics and violence behind closed doors: The spatial overlap of child maltreatment and intimate partner violence

2018

In this study, we analyze first whether there is a common spatial distribution of child maltreatment (CM) and intimate partner violence (IPV), and second, whether the risks of CM and IPV are influenced by the same neighborhood characteristics, and if these risks spatially overlap. To this end we used geocoded data of CM referrals (N = 588) and IPV incidents (N = 1450) in the city of Valencia (Spain). As neighborhood proxies, we used 552 census block groups. Neighborhood characteristics analyzed at the aggregated level (census block groups) were: Neighborhood concentrated disadvantage (neighborhood economic status, neighborhood education level, and policing activity), immigrant concentration…

Child abuseMaleEconomicsEconomics of Training and Educationlcsh:MedicinePoison controlIntimate Partner ViolenceSocial SciencesCriminology0302 clinical medicineSociologyResidence CharacteristicsRisk FactorsMedicine and Health SciencesEconomic StatusPublic and Occupational Health030212 general & internal medicineChild Abuselcsh:ScienceChildPolicingHuman CapitalMultidisciplinarySocial ResearchGeography05 social sciencesTraumatic Injury Risk FactorsHuman factors and ergonomicsPoliceSocial researchProfessionsGeographyResearch Designpopulation characteristicsNeighborhoodsEducational StatusFemaleCrime050104 developmental & child psychologyResearch ArticleCensusAdolescentEmigrants and ImmigrantsHuman GeographyResearch and Analysis MethodsEducation03 medical and health sciencesInjury preventionHumans0501 psychology and cognitive sciencesSocioeconomic statusViolent CrimeEducational AttainmentSurvey Researchlcsh:Rsocial sciencesEducational attainmentSpainPeople and PlacesSpouse AbuseEarth SciencesDomestic violencelcsh:QPopulation GroupingsDemographyPLoS ONE
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Childhood Adversities and Adult Headache in Poland and Germany.

2015

Objective Various childhood adversities have been found to be associated with chronic pain in adulthood. However, associations were moderate in most studies, i.e. odds ratios (OR) were between one and two. Method An internet survey was performed in 508 Polish and 500 German subjects. A total of 19 childhood adversities were selected and their associations with headaches explored. Age, gender and country were included as potential confounders, as well as their two-way interaction with the risk factors. Results Two strong risk factors were identified. (1) A combined score for physical and emotional neglect showed an odds ratio (OR) of 2.78 (p < .002) to the frequency of headache in adulthood …

Child abuseMalePhysiologyEconomicsSensory PhysiologySocial Scienceslcsh:MedicineCriminologyPathology and Laboratory MedicinePediatrics0302 clinical medicineSociology030202 anesthesiologyRisk FactorsGermanyOdds RatioMedicine and Health SciencesMicroeconomicsMedicineChild AbuseComputer NetworksChildlcsh:ScienceEmotional neglectmedia_commonMultidisciplinaryHeadachesOrganic CompoundsConfoundingChronic painHeadacheSensory SystemsChemistryAdult Survivors of Child Adverse EventsSomatosensory SystemChild PreschoolPhysical SciencesFemaleCrimeHeadachesmedicine.symptomResearch ArticleAdultmedicine.medical_specialtyComputer and Information Sciencesmedia_common.quotation_subjectNeglect03 medical and health sciencesSigns and SymptomsHumansAdultsPsychiatryMigraineInternetbusiness.industryOrganic Chemistrylcsh:RInfant NewbornChemical CompoundsInfantBiology and Life SciencesPain SensationOdds ratiomedicine.diseaseHealth SurveysHousehold EconomicsMigraineAge GroupsAlcoholsPeople and PlacesPopulation Groupingslcsh:QPolandbusiness030217 neurology & neurosurgeryDemographyNeurosciencePLoS ONE
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