Search results for "SELE"

showing 10 items of 4721 documents

Development of predictive retention-activity relationship models of tricyclic antidepressants by micellar liquid chromatography.

1999

The distribution of tricyclic antidepressants from plasma to brain, where these drugs exert their main clinical action, and other organs is related to transport events across the cell membranes of the different tissues. It could be expected that all the molecular features that condition the transport processes (mainly hydrophobicity and molar total charge) also control the pharmacokinetic and biochemical behavior. Micellar liquid chromatography (MLC) has been proposed to emulate in vitro the partitioning process in the biomembranes. The use of micellar solutions of Brij35 as mobile phases in reversed-phase liquid chromatography has proven to be valid to predict the biological activities of …

SerotoninAntidepressive Agents TricyclicModels BiologicalMicellar electrokinetic chromatographyNorepinephrineStructure-Activity RelationshipPharmacokineticsReceptors Adrenergic alpha-1Drug DiscoveryDistribution (pharmacology)AnimalsEnzyme InhibitorsAdrenergic alpha-AntagonistsMicelleschemistry.chemical_classificationChromatographyChemistryCapacity factorRatsMembraneMicellar liquid chromatographyMicellar solutionsAdenylyl Cyclase InhibitorsHistamine H1 AntagonistsMolecular MedicineSelective Serotonin Reuptake InhibitorsTricyclicChromatography LiquidJournal of medicinal chemistry
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Central Serotonin2C Receptor: From Physiology to Pathology

2006

Since the 1950s, when serotonin (5-HT) was discovered in the mammalian central nervous system (CNS), an enormous amount of experimental evidence has revealed the pivotal role of this biogenic amine in a number of cognitive and behavioural functions. Although 5-HT is synthesized by a small group of neurons within the raphe nuclei of the brain stem, almost all parts of the CNS receive serotonergic projections. Furthermore, the importance of 5-HT modulation and the fine-tuning of its action is underlined by the large number of 5-HT binding sites found in the CNS. Hitherto, up to 15 different 5-HT receptors subtypes have been identified. This review was undertaken to summarize the work that has…

SerotoninDORSAL RAPHE NUCLEUSPathologymedicine.medical_specialtyProtein ConformationCentral nervous systemPhysiologyRAT NUCLEUS-ACCUMBENSBiologySerotonergicDorsal raphe nucleusPLEXUS EPITHELIAL-CELLSAGONIST-DIRECTED TRAFFICKINGDrug DiscoveryReceptor Serotonin 5-HT2CmedicineAnimalsHumansserotonergic receptorselective 5-HT2C drugs Key Words Plus: VENTRAL TEGMENTAL AREAReceptor5-HT receptorReceptor Serotonin 5-HTCENTRAL-NERVOUS-SYSTEMGeneral MedicineEXTRACELLULAR DOPAMINE LEVELSmedicine.diseaseschizophreniamedicine.anatomical_structureGene Expression RegulationDepression Mentaldrug of abuse5-HT2 ANTAGONIST RITANSERINSchizophreniadepressionSchizophreniaATYPICAL ANTIPSYCHOTIC-DRUGSSerotoninRaphe nucleiPRIMATE CEREBRAL-CORTEXSignal TransductionCurrent Topics in Medicinal Chemistry
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Gaining Competitive Advantage through Standardization and Differentiation of Services

2015

The goal of the paper is to study the question of whether or not differences between cultural groups influence the decision of a consumer wishing to avail himself of a particular service. Therefore we have developed a semiotic extension of the means-end approach as the theoretical basis for elaborating a solution to this problem. The conjoint analysis specifies the results of the meansend analysis.

Service (business)Knowledge managementStandardizationbusiness.industryCultural group selectionSemioticsBusinessRepertory gridMarketingCompetitive advantageConjoint analysis
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Design and optimisation of an innovative two-hub-and-spoke network for the Mediterranean short-sea-shipping market

2020

Abstract Short Sea Shipping (SSS) is generally considered as a privileged transport mode in terms of reducing road congestion and related external costs. In the last two decades, SSS has attracted a lot of attention in the European Union, where it is also regarded as a key factor for economic and social cohesion between countries. In this regard, the present study proposes a new network design that aims at improving and increasing freight traffic between the north-western and the south-eastern shores of the Mediterranean Basin. The proposed model, designed for Ro-Ro (Roll-on Roll-off) freight transport, tries to overcome the limits of the existing multi-port-calling services through an inno…

Service (systems architecture)021103 operations researchMotorways of the SeaGeneral Computer ScienceOperations researchComputer scienceMotorways of the SeaNetwork Design OptimisationShort Sea ShippingService Frequency Selection0211 other engineering and technologiesGeneral EngineeringMode (statistics)Cohesion (computer science)02 engineering and technologyRo-Ro MarketSupply and demandNetwork planning and designMediterranean Corridors0202 electrical engineering electronic engineering information engineeringShort sea shippingmedia_common.cataloged_instance020201 artificial intelligence & image processingEuropean unionmedia_common
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Automating the Parameter Selection in VRP: An Off-line Parameter Tuning Tool Comparison

2014

Vehicle route optimization is an important application of combinatorial optimization. Therefore, a variety of methods has been proposed to solve different challenging vehicle routing problems. An important step in adopting these methods to solve real-life problems is to find appropriate parameters for the routing algorithms. In this chapter, we show how this task can be automated using parameter tuning by presenting a set of comparative experiments on seven state-of-the-art tuning methods. We analyze the suitability of these methods in configuring routing algorithms, and give the first critical comparison of automated parameter tuners in vehicle routing. Our experimental results show that t…

Set (abstract data type)Computer scienceVehicle routing problemCombinatorial optimizationTunerControl engineeringRouting (electronic design automation)AlgorithmTravelling salesman problemSelection (genetic algorithm)Task (project management)
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The DrosDel Collection

2004

Abstract We describe a collection of P-element insertions that have considerable utility for generating custom chromosomal aberrations in Drosophila melanogaster. We have mobilized a pair of engineered P elements, p{RS3} and p{RS5}, to collect 3243 lines unambiguously mapped to the Drosophila genome sequence. The collection contains, on average, an element every 35 kb. We demonstrate the utility of the collection for generating custom chromosomal deletions that have their end points mapped, with base-pair resolution, to the genome sequence. The collection was generated in an isogenic strain, thus affording a uniform background for screens where sensitivity to genetic background is high. The…

Set (abstract data type)Whole genome sequencingGeneticsP elementbiologyMolecular screeningStrain (biology)GeneticsDrosophila melanogasterbiology.organism_classificationSelection (genetic algorithm)Sequence (medicine)Genetics
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INTRA-CULTIVAR DIVERSITY IN SOUTHERN ITALY OLIVE CULTIVARS DEPICTED BY MORPHOLOGICAL TRAITS AND SSR MARKERS

2014

In this study, SSR analysis was performed on a large number of putative clones of the main olive cultivars from two Italian regions, Sicily and Calabria, in order to study the genetic relatedness, and to detect any degree of genetic diversity, which can be used to unambiguously identify possible superior clones. These putative clones have been collected and observed in the last ten years, following an extensive investigation carried out in traditional olive growing areas, thanks to the reports of farmers, millers, technician, growers and nurseries. The set of microsatellite (SSR) markers used allowed the detection of the genetic diversity, resulting from somatic mutation, indicating the pre…

Settore AGR/03 - Arboricoltura Generale E Coltivazioni ArboreeHorticultureGeographymedia_common.quotation_subjectCultivarHorticultureOlea europaea clonal selection SSR fingerprinting germplasmDiversity (politics)media_common
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Intra-cultivar Diversity in sicilian and calabrian olive (olea europaea L.) Cultivars Depicted by Morphological Traits and SSR Markers

2012

In this study, SSR analysis was performed on a large number of putative clones of the main olive cultivars from two Italian regions, Sicily and Calabria, in order to study the genetic relatedness, and to detect any degree of genetic diversity, which can be used to unambiguously identify possible superior clones. These putative clones have been collected and observed in the last ten years, following an extensive investigation carried out in traditional olive growing areas, thanks to the reports of farmers, millers, technician, growers and nurseries. The set of microsatellite (SSR) markers used allowed the detection of the genetic diversity, resulting from somatic mutation, indicating the pre…

Settore AGR/03 - Arboricoltura Generale E Coltivazioni ArboreeOlea europaea clonal selection SSR Fingerprinting Germplasm
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ADATTAMENTO ALLA GESTIONE BIOLOGICA DI CULTIVAR DI PESCO ( PRUNUS PERSICA L. BATSCH ) SICILIANE OTTENUTE ATTRAVERSO SELEZIONE MASSALE E INCROCIO.

2011

Settore AGR/03 - Arboricoltura Generale E Coltivazioni ArboreeSELEZIONE MASSALE E INCROCIO.CULTIVAR DI PESCO ( PRUNUS PERSICA L. BATSCH)SICILIANEADATTAMENTO ALLA GESTIONE BIOLOGICA
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Ottenere cloni moderni

2008

Settore AGR/03 - Arboricoltura Generale E Coltivazioni ArboreeSelezione clonale vitis vinifera
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