Search results for "Salonitenolide"

showing 2 items of 2 documents

Acid Rearrangment of Epoxy-germacranolides and Absolute Configuration of 1β,10α-Epoxy-salonitenolide

2010

The acid-catalyzed cyclization of mono epoxides of cnicin acetonide (3) was investigated. Several 6,12-eudesmanolides were obtained, and their stereochemistry established by extensive spectroscopic analyses. Chemical correlations also led to the assignment of the absolute configuration of 1β,10α-epoxy-salonitenolide (13), a previously isolated natural product. The cytotoxic activities of some compounds were determined against A549 and MCF-7 tumor cell lines. The esterified germacranolides 2–6 were selectively cytotoxic against the MCF-7 breast cancer cell line.

PharmacologyNatural productStereochemistryAbsolute configurationSalonitenolidePlant ScienceGeneral MedicineEpoxyAcetonideCnicinchemistry.chemical_compoundComplementary and alternative medicineBreast cancer cell linechemistryvisual_artDrug Discoveryvisual_art.visual_art_mediumOrganic chemistryCytotoxicityNatural Product Communications
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Sesquiterpene lactones from Centaurea alba and C. conifera

1995

Abstract The aerial parts of Centaurea alba yielded five know germacranolides: salonitenolide, 11β, 13-dihydrosalonitenolide, salonitenolide 8- O -(4′-acetoxy-5′-hydroxy)-angelate, cnicin 4′-O-acetate and cnicin. The aerial parts of C. conifera yielded loliolide, 1β,6α-dihydroxy-4(15)-eudesmene, chlorojanerin, chlorohyssopifolin A (centaurepensin) and its C-17 epimer. The latter compound is described for the first time.

StereochemistryChlorojanerinSalonitenolidePlant ScienceGeneral MedicineHorticultureSesquiterpeneBiochemistryCnicinCentaurea albachemistry.chemical_compoundchemistryBotanyEpimerMolecular BiologyPhytochemistry
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