Search results for "Tegmen"

showing 10 items of 76 documents

Glutamate and opioid antagonists modulate dopamine levels evoked by innately attractive male chemosignals in the nucleus accumbens of female rats

2017

Sexual chemosignals detected by vomeronasal and olfactory systems mediate intersexual attraction in rodents, and act as a natural reinforcer to them. The mesolimbic pathway processes natural rewards, and the nucleus accumbens receives olfactory information via glutamatergic projections from the amygdala. Thus, the aim of this study was to investigate the involvement of the mesolimbic pathway in the attraction toward sexual chemosignals. Our data show that female rats with no previous experience with males or their chemosignals display an innate preference for male-soiled bedding. Focal administration of the opioid antagonist b-funaltrexamine into the posterior ventral tegmental area does no…

0301 basic medicinemedicine.medical_specialtySexual attractionmedicine.drug_classSistema nerviós central MalaltiesNeuroscience (miscellaneous)olfactory systemMesolimbic pathwayNucleus accumbensAmygdalaNaltrexonePheromones03 medical and health sciencesCellular and Molecular NeuroscienceFeromones0302 clinical medicineNeurochemicalRewardDopamineInternal medicinemedicinerewardOriginal ResearchMesolimbic systemsexual attractionOlfactory systemVentral tegmental areaNeuroanatomy030104 developmental biologymedicine.anatomical_structureEndocrinologymesolimbic systemAnatomypheromonesPsychologyNeuroscience030217 neurology & neurosurgeryOpioid antagonistTecnologia farmacèuticamedicine.drug
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The neurobiological bases for the pharmacotherapy of nicotine addiction.

2007

Nicotine, the major psychoactive agent present in tobacco, acts as a potent addictive drug both in humans and laboratory animals, whose locomotor activity is also stimulated. A large body of evidence indicates that the locomotor activation and the reinforcing effects of nicotine may be related to its stimulatory effects on the mesolimbic dopaminergic function. Thus, it is now well established that nicotine can increase in vivo DA outflow in the nucleus accumbens and the corpus striatum. The stimulatory effect of nicotine on DA release most probably results from its ability to excite the neuronal firing rate and to increase the bursting activity of DA neurons in the substantia nigra pars com…

RAT STRIATAL SYNAPTOSOMESNicotineINDUCED BEHAVIORAL SENSITIZATIONmedia_common.quotation_subjectSubstantia nigraStriatumNicotinic AntagonistsBiologyNucleus accumbensPharmacologyReceptors NicotinicNicotineDrug DiscoverySUSTAINED-RELEASE BUPROPIONmedicineLOCOMOTOR STIMULANT ACTIONAnimalsHumansNicotinic Agonistsmedia_commonPharmacologyMIDBRAIN DOPAMINE NEURONSPars compactaAddictionNIGRA PARS COMPACTAFACILITATES SMOKING CESSATIONTobacco Use DisorderSUBUNIT MESSENGER-RNAAntidepressive AgentsVentral tegmental areaVENTRAL TEGMENTAL AREANicotinic agonistmedicine.anatomical_structurenervous systemmedicine.drugSEROTONIN(2C) RECEPTORS BLOCKSCurrent pharmaceutical design
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Lateral Habenula 5-HT2C Receptor Function Is Altered by Acute and Chronic Nicotine Exposures

2021

Serotonin (5-HT) is important in some nicotine actions in the CNS. Among all the 5-HT receptors (5-HTRs), the 5-HT2CR has emerged as a promising drug target for smoking cessation. The 5-HT2CRs within the lateral habenula (LHb) may be crucial for nicotine addiction. Here we showed that after acute nicotine tartrate (2 mg/kg, i.p.) exposure, the 5-HT2CR agonist Ro 60-0175 (5–640 µg/kg, i.v.) increased the electrical activity of 42% of the LHb recorded neurons in vivo in rats. Conversely, after chronic nicotine treatment (6 mg/kg/day, i.p., for 14 days), Ro 60-0175 was incapable of affecting the LHb neuronal discharge. Moreover, acute nicotine exposure increased the 5-HT2CR-immunoreactive (IR)…

0301 basic medicinenucleus accumbensdorsal raphe nucleusmedicine.medical_treatmentstriatumStriatumSmoking cessationSettore BIO/09 - FisiologiaSerotonin -- ReceptorsNicotineNicotine addiction -- Treatment0302 clinical medicinesingle cell-extracellular recordingMedicinesubstantia nigra pars compactadentate gyrusBiology (General)SpectroscopyGeneral MedicineDorsal raphe nucleuComputer Science ApplicationsVentral tegmental area5-HT2C receptorChemistrymedicine.anatomical_structuredepressionaddictionmedicine.drugAgonistmedicine.medical_specialtyendocrine systemQH301-705.5medicine.drug_classRo 60-0175ventral tegmental areaNucleus accumbensDentate gyruCatalysisInorganic Chemistry03 medical and health sciencesInternal medicineNucleus accumbenPhysical and Theoretical ChemistryQD1-999Molecular BiologyHabenulabusiness.industryOrganic Chemistry030104 developmental biologyEndocrinologySmoking cessationSerotoninbusinessSerotonin -- Agonists030217 neurology & neurosurgerymedial prefrontal cortexInternational Journal of Molecular Sciences
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Central Serotonin2C Receptor: From Physiology to Pathology

2006

Since the 1950s, when serotonin (5-HT) was discovered in the mammalian central nervous system (CNS), an enormous amount of experimental evidence has revealed the pivotal role of this biogenic amine in a number of cognitive and behavioural functions. Although 5-HT is synthesized by a small group of neurons within the raphe nuclei of the brain stem, almost all parts of the CNS receive serotonergic projections. Furthermore, the importance of 5-HT modulation and the fine-tuning of its action is underlined by the large number of 5-HT binding sites found in the CNS. Hitherto, up to 15 different 5-HT receptors subtypes have been identified. This review was undertaken to summarize the work that has…

SerotoninDORSAL RAPHE NUCLEUSPathologymedicine.medical_specialtyProtein ConformationCentral nervous systemPhysiologyRAT NUCLEUS-ACCUMBENSBiologySerotonergicDorsal raphe nucleusPLEXUS EPITHELIAL-CELLSAGONIST-DIRECTED TRAFFICKINGDrug DiscoveryReceptor Serotonin 5-HT2CmedicineAnimalsHumansserotonergic receptorselective 5-HT2C drugs Key Words Plus: VENTRAL TEGMENTAL AREAReceptor5-HT receptorReceptor Serotonin 5-HTCENTRAL-NERVOUS-SYSTEMGeneral MedicineEXTRACELLULAR DOPAMINE LEVELSmedicine.diseaseschizophreniamedicine.anatomical_structureGene Expression RegulationDepression Mentaldrug of abuse5-HT2 ANTAGONIST RITANSERINSchizophreniadepressionSchizophreniaATYPICAL ANTIPSYCHOTIC-DRUGSSerotoninRaphe nucleiPRIMATE CEREBRAL-CORTEXSignal TransductionCurrent Topics in Medicinal Chemistry
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Salsolinol and ethanol-derived excitation of dopamine mesolimbic neurons: new insights

2013

Evidence supporting the essential role of brain-derived ethanol metabolites in the excitation of dopamine (DA) midbrain neurons has multiplied in the last 10–15 years. The pioneer and influential behavioral studies by CM Aragon and colleagues (see Correa et al., 2012 for a complete review) and more recent data (Sanchez-Catalan et al., 2009; Marti-Prats et al., 2010, 2013) have repeatedly demonstrated the crucial role displayed by acetaldehyde (ACD) in the locomotor and other behavioral responses elicited by ethanol. Although these experiments mainly used an indirect measure (exploratory locomotion) as an index of the excitation of DA neurons in the ventral tegmental area (VTA), results stro…

Cognitive NeuroscienceAcetaldehydeStriatumInhibitory postsynaptic potentiallcsh:RC321-571Behavioral NeuroscienceGlutamatergicDopaminemedicinePremovement neuronal activitylcsh:Neurosciences. Biological psychiatry. NeuropsychiatryGeneral Commentary ArticleSalsolinolElectrophysiologyVentral tegmental areaµ-Opioid ReceptorsElectrophysiologyNeuropsychology and Physiological Psychologymedicine.anatomical_structurenervous systemHypothalamusDopamine Midbrain NeuronsPsychologyNeuroscienceNeurosciencemedicine.drugFrontiers in Behavioral Neuroscience
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Influence of ventral tegmental area (A10 region) on flight behaviour elicited by hypothalamic stimulation in the cat.

1993

The influence of the ventral tegmental area (VTA) (dopaminergic A10 group neurons) on flight behaviour, induced by hypothalamic stimulation, was studied in the cat. Co-stimulation of hypothalamus and VTA (ipsi- or contralateral) induced an increase of the flight latency. Slow-motion analysis of flight behaviour showed that this increase was due to the augmentation of the fixation latency (FL) whereas the upright latency (UL) was not modified. Sulpiride injection (50 mg/kg i.p.) provoked the disappearance of VTA effect without affecting the basal behavioural sequence. The results show that DA A10 group neurons increase the attentive component of the flight reaction, suggesting a possible inf…

Tegmentum MesencephaliDopamineCentral nervous systemHypothalamusEscape ReactionmedicineCarnivoraAnimalsAnesthesiaAttentionLatency (engineering)Molecular BiologyNeuronsbiologyChemistryGeneral NeuroscienceFissipediaDopaminergicbiology.organism_classificationElectric StimulationVentral tegmental areamedicine.anatomical_structurenervous systemHypothalamusCatsNeurology (clinical)SulpirideSulpirideNeuroscienceDevelopmental Biologymedicine.drugBrain research
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Opposite motor responses elicited by ethanol in the posterior VTA: The role of acetaldehyde and the non-metabolized fraction of ethanol

2013

Recent electrophysiological evidence suggests that ethanol simultaneously exerts opposite effects on the activity of dopamine (DA) neurons in the ventral tegmental area (VTA) through two parallel mechanisms, one promoting and the other reducing the GABA release onto VTA DA neurons. Here we explore the possible behavioural implications of these findings by investigating the role displayed by acetaldehyde (the main metabolite of ethanol) and the non-metabolized fraction of ethanol in motor activity of rats. We analyse the appearance of motor activation or depression after intra-VTA administration of ethanol in rats subjected to different pharmacological pre-treatments designed to preferential…

MaleMicroinjectionsMetaboliteGABA(A) receptorsAcetaldehydePharmacologyMotor ActivityNon-metabolized fraction of ethanolBicucullineCellular and Molecular Neurosciencechemistry.chemical_compoundDopaminemedicineAnimalsGABA-A Receptor AntagonistsEnzyme InhibitorsRats WistarPharmacologyEthanolDose-Response Relationship DrugEthanolChemistryGABAA receptorVentral Tegmental AreaAcetaldehydeCentral Nervous System DepressantsBicucullineRatsVentral tegmental areaElectrophysiologymedicine.anatomical_structureBiochemistrynervous systemCyanamideVTAmedicine.drug
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Effect Of Inflammatory Pain On Alcohol-Induced Dopamine Release In The Nucleus Accumbens: Behavioural Implications In Rat Models

2019

AbstractRecent studies have drawn the attention to the link between Alcohol Use Disorder (AUD) and the presence of pain. Indeed, the correct management of pain in patients with a previous history of AUD has been reported to decrease the risk of relapse in alcohol drinking, suggesting that in this prone population, pain may increase the vulnerability to relapse. Previous data in male rats revealed that inflammatory pain desensitizes mu opioid receptors (MORs) in the ventral tegmental area (VTA) and increases intake of high doses of heroine. Due to the relevant role of MORs in alcohol effects, we hypothesize that pain may also alter alcohol reinforcing properties and therefore affect alcohol …

Microdialysiseducation.field_of_studymedicine.medical_specialtybusiness.industryPopulationAlcohol use disorderNucleus accumbensmedicine.diseaseVentral tegmental areamedicine.anatomical_structureEndocrinologyNeurochemicalDopamineInternal medicineMedicineμ-opioid receptorbusinesseducationmedicine.drug
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EFFERENT CONNECTIONS OF THE CEREBELLUM OF THE WEAKLY ELECTRIC FISH EIGENMANNIA SP. (GYMNOTODEI)

1981

An efferent connection of lobus caudalis cells of the cerebellum of the electric fish Eigenmannia sp. has been verified by means of electrical stimulation and recording techniques. Stimulating in the lobus caudalis, an orthodromic activation has been found in the reticular formation of the midbrain tegmentum. Switching recording and stimulating electrodes led to an antidromic activation in cells of the lobus caudalis. The area identified in the midbrain corresponds to what, in higher vertebrates, is called the red nucleus.

LobusMidbrainbiologyChemistryRed nucleusEfferentMidbrain tegmentumAnatomybiology.organism_classificationReticular formationNeuroscienceElectric fishAntidromic
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Sexual pheromones and the evolution of the reward system of the brain: the chemosensory function of the amygdala.

2008

The amygdala of all tetrapod vertebrates receives direct projections from the main and accessory olfactory bulbs, and the strong similarities in the organization of these projections suggest that they have undergone a very conservative evolution. However, current ideas about the function of the amygdala do not pay sufficient attention to its chemosensory role, but only view it as the core of the emotional brain. In this study, we propose that both roles of the amygdala are intimately linked since the amygdala is actually involved in mediating emotional responses to chemical signals. The amygdala is the only structure in the brain receiving pheromonal information directly from the accessory …

Olfactory systemVomeronasal organolfactory tuberclevomeronasalAmygdalaModels BiologicalRewardNeural PathwaysmedicineAnimalsHumansOlfactory memorySex AttractantsGeneral NeuroscienceOlfactory tubercleAmygdalaolfactoryBiological EvolutionChemoreceptor CellsVentral tegmental areamedicine.anatomical_structureSex pheromoneIslands of CallejadopamineIslands of CallejaPsychologyNeuroscienceVentral tegmental areaBrain research bulletin
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