Search results for "Terpene"

showing 10 items of 816 documents

Crystal structure and Hirshfeld surface analysis of 3-oxours-12-ene-27a,28-dioic acid (quafrinoic acid)

2017

The title compound, known as quafrinoic acid, is a penta­cyclic triterpene isolated from Nauclea Pobeguinii. The compound is composed of five fused six-membered rings and the mol­ecular conformation is stabilized by intra­molecular C—H⋯O inter­action, forming S6 and S8 rings.

Surface (mathematics)crystal structurepentacyclic triterpene010405 organic chemistryHydrogen bondStereochemistryChemistryCyclohexane conformationGeneral ChemistryCrystal structure010403 inorganic & nuclear chemistryCondensed Matter Physics01 natural sciences0104 chemical sciencesResearch CommunicationsCrystalNauclea pobeguiniialcsh:Chemistrylcsh:QD1-999Hirshfeld surface analysisGeneral Materials Sciencequafrinoic acidEne reactionpenta­cyclic triterpeneActa Crystallographica Section E: Crystallographic Communications
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Development of antimigraine transdermal delivery systems of pizotifen malate.

2015

Abstract The aim of this study was to develop and evaluate a transdermal delivery system of pizotifen malate. Pizotifen is frequently used in the preventive treatment of migraine, but is also indicated in eating disorders. In the course of the project, the effects of chemical enhancers such as ethanol, 1,8-cineole, limonene, azone and different fatty acids (decanoic, decenoic, dodecanoic, linoleic and oleic acids) were determined, first using a pizotifen solution. Steady state flux, diffusion and partition parameters were estimated by fitting the Scheuplein equation to the data obtained. Among the chemical enhancers studied, decenoic acid showed the highest enhancement activity, which seeme…

SwineMigraine DisordersSkin AbsorptionPharmaceutical ScienceAbsorption (skin)PizotifenIn Vitro TechniquesAdministration Cutaneouschemistry.chemical_compoundDrug Delivery SystemsCyclohexenesmedicineOrganic chemistryAnimalsTransdermalDegree of unsaturationPizotylineEucalyptolIontophoresisEthanolTerpenesFatty AcidsAzepinesAnalgesics Non-NarcoticIontophoresisCyclohexanolsOleic acidchemistryMonoterpenesDecenoic AcidAzoneLimonenemedicine.drugInternational journal of pharmaceutics
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Induction of apoptosis in a leukemia cell line by triterpene saponins from Albizia adianthifolia

2004

Abstract Triterpenoid saponins, which are present in plants and some marine animals, exert various important pharmacological effects. The present study examines the effects of adianthifoliosides A, B, and D (AdA, AdB, and AdD) together with two prosapogenins (Pro1 and Pro2) obtained from Albizia adianthifolia (Mimosaceae) on human leukemia T-cells (Jurkat cells) and on splenocytes. AdA, AdB, and AdD were found to exhibit a cytotoxic effect on Jurkat cells, whereas the prosapogenins were found to exert a lymphoproliferative effect on this cell type. Furthermore, all tested compounds were found to exert a synergistic lymphoproliferative activity with concanavalin A (ConA) on splenocytes. The …

T-LymphocytesClinical BiochemistryPharmaceutical ScienceAlbizziaApoptosisHemolysisBiochemistryJurkat cellsCell LineJurkat Cellschemistry.chemical_compoundDrug DiscoveryTumor Cells CulturedHumansCytotoxic T cellPropidium iodideOleanolic AcidCytotoxicityMolecular BiologyPlants MedicinalDose-Response Relationship DrugbiologyChemistryOrganic ChemistryBiological activitySaponinsbiology.organism_classificationAntineoplastic Agents PhytogenicTriterpenesBiochemistryConcanavalin ACell culturebiology.proteinMolecular MedicineAlbizia adianthifoliaBioorganic & Medicinal Chemistry
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Relevant essential oil components: a minireview on increasing applications and potential toxicity.

2021

[EN] Phenolic compounds carvacrol, thymol, eugenol, and vanillin are four of the most thoroughly investigated essential oil components given their relevant biological properties. These compounds are generally considered safe for consumption and have been used in a wide range of food and non-food applications. Significant biological properties, including antimicrobial, antioxidant, analgesic, anti-inflammatory, anti-mutagenic, or anti-carcinogenic activity, have been described for these components. They are versatile molecules with wide-ranging potential applications whose use may substantially increase in forthcoming years. However, some in vitro and in vivo studies, and several case report…

TECNOLOGIA DE ALIMENTOSHealth Toxicology and Mutagenesis010501 environmental sciencesToxicology01 natural scienceslaw.invention03 medical and health scienceschemistry.chemical_compoundMicelawCarvacrolBiological propertyEugenolOils VolatileAnimalsCarvacrolFood scienceThymolEssential oil0105 earth and related environmental sciences0303 health sciencesToxicityChemistryVanillin030302 biochemistry & molecular biologyThymolAnti-Bacterial AgentsRatsEugenolToxicityVanillinMonoterpenesRabbitsPotential toxicityToxicology mechanisms and methods
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Addition of pasture plant essential oil in milk: Influence on chemical and sensory properties of milk and cheese

2007

The aim of this experiment was to study the effect of the addition, to milk, of an essential oil (EO) obtained from the hydrodistillation of plants collected from a mountain natural pasture on the milk and cheese sensory properties. The EO was mainly composed of terpenoid compounds (67 of the 95 compounds identified) as well as ketones, aldehydes, alcohols, esters, alkanes, and benzenic compounds. In milk, the addition of this EO at the concentration of 0.1 microL/L did not influence its sensory properties, whereas at 1.0 microL/L, sensory properties were modified. In cheeses, the effect of adding EO into milk was studied in an experimental dairy plant allowing the production of small Canta…

TERPENE[SDV.SA]Life Sciences [q-bio]/Agricultural sciencesGas Chromatography-Mass SpectrometryVOLATILE COMPOUNDlaw.inventionSENSORY PROPERTYTerpene0404 agricultural biotechnologyCheeselawGeneticsAnimalsHumansPlant OilsFood scienceEssential oilAromaComputingMilieux_MISCELLANEOUS2. Zero hungerbiologyTerpenesChemistry0402 animal and dairy scienceRipening04 agricultural and veterinary sciencesRaw milkbiology.organism_classification040401 food science040201 dairy & animal scienceTerpenoidESSENTIAL OILMilkOdorTasteOdorantsFood TechnologyCattleAnimal Science and ZoologyComposition (visual arts)Food Science
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Changes in terpene content in milk from pasture-fed cows

2006

International audience

TERPENE[SDV.SA]Life Sciences [q-bio]/Agricultural sciencesPASTURE DEVELOPMENT GRAZING MANAGMENT MILK TERPENE UPLAND PASTURE[SDV.SA] Life Sciences [q-bio]/Agricultural sciencesGRAZING MANAGEMENTUPLAND PASTUREPASTURE DEVELOPMENTMILK TERPENEComputingMilieux_MISCELLANEOUS
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Essential Oil in Milk: Its Influence on Milk and Cheese Chemical and Sensory Properties.

2007

TERPENES SENSORY PROPERTY ESSENTIAL OIL VOLATILE COMPOUND
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ChemInform Abstract: Synthesis of (+)-Pechueloic Acid and (+)-Aciphyllene. Revision of the Structure of (+)-Aciphyllene.

2008

Abstract 1α H ,7α H ,10α H -Guaia-4,11-dien-3-one and its 1β H ,10β H diastereomer, easily obtained from (+)-dihydrocarvone, are good starting materials for the synthesis of natural guaiane derivatives. Allylic oxidation of the 1α H ,10α H isomer gave as main product its 13-hydroxy derivative and a small amount of (+)-7β-hydroxy-1α H ,10α H -guaia-4,11-dien-3-one, whereas the 1β H ,10β H diastereomer afforded selectively the (−)-7α-hydroxy-1β H ,10β H enantiomer in excellent yield. From the 13-hydroxy derivative (+)-pechueloic acid and (+)-methyl pechueloate were synthesized. Deoxygenation at C 3 of the 1β H ,10β H guaiadienone afforded a guaiadiene with the reported structure for aciphylle…

TerpeneAllylic rearrangementchemistry.chemical_compoundDienechemistryYield (chemistry)DiastereomerGeneral MedicineEnantiomerSpectral dataMedicinal chemistryDeoxygenationChemInform
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ChemInform Abstract: Sterelactones: New Isolactarane Type Sesquiterpenoids with Antifungal Activity from Stereum sp. IBWF 01060.

2009

Four members of a new family of tetracyclic sesquiterenoids possessing the isolactarane skeleton have been isolated from mycelial cultures of Stereum sp. IBWF 01060. Their structure elucidation and their antifungal activity against several plant pathogens as well as other microorganisms are reported.

TerpeneAntifungalStereum sp.Stereochemistrymedicine.drug_classChemistrymedicineGeneral MedicineMyceliumChemInform
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ChemInform Abstract: Stereoselective Construction of the Tetracyclic Scalarane Skeleton from Carvone.

2010

The tetracyclic scalarane skeleton 22 has been constructed from (S)-(+)-carvone using two intramolecular Diels–Alder reactions as key synthetic steps.

TerpeneCarvonechemistry.chemical_compoundChemistryStereochemistryIntramolecular forceStereoselectivityGeneral MedicineSkeleton (category theory)ChemInform
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