Search results for "Trichlorfon"

showing 2 items of 2 documents

Galantamine is an allosterically potentiating ligand of neuronal nicotinic but not of muscarinic acetylcholine receptors.

2003

Galantamine (Reminyl), an approved treatment for Alzheimer's disease (AD), is a potent allosteric potentiating ligand (APL) of human alpha 3 beta 4, alpha 4 beta 2, and alpha 6 beta 4 nicotinic receptors (nAChRs), and of the chicken/mouse chimeric alpha 7/5-hydroxytryptamine3 receptor, as was shown by whole-cell patch-clamp studies of human embryonic kidney-293 cells stably expressing a single nAChR subtype. Galantamine potentiates agonist responses of the four nAChR subtypes studied in the same window of concentrations (i.e., 0.1-1 microM), which correlates with the cerebrospinal fluid concentration of the drug at the recommended daily dosage of 16 to 24 mg. At concentrations10 microM, gal…

Agonistmedicine.medical_specialtymedicine.drug_classRecombinant Fusion ProteinsAllosteric regulationPhenylcarbamatesRivastigminePharmacologyReceptors NicotinicMiceAllosteric RegulationPiperidinesInternal medicineMuscarinic acetylcholine receptormedicineGalantamineAnimalsHumansDonepezilReceptorTrichlorfonCells CulturedPharmacologyNeuronsChemistryGalantamineLigand (biochemistry)Receptors MuscarinicEndocrinologyNicotinic agonistIndansTacrineMolecular MedicineCholinergicCarbamatesCholinesterase Inhibitorsmedicine.drugThe Journal of pharmacology and experimental therapeutics
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Acute lethal toxicity of some pesticides toBrachionus calyciflorus andBrachionus plicatilis

1991

Due to their widespread distribution and toxic nattwe pesticides may have a serious impact on the aquatic environment and exert adverse effects on the associated organisms. Acute bioassay tests have been used to determine the actual impact of various pesticides on aquatic life. Static acute toxicity tests provide rapid and reproductible concentration-response curves for estimating toxic effects of chemicals on aquatic organisms. These tests provide a data base for determining relative toxicity to a variety of species.

Health Toxicology and MutagenesisRotiferaFresh WaterBiologyToxicologyLethal Dose 50ToxicologySpecies SpecificityBrachionus calyciflorusAnimalsEcotoxicologyBioassaySeawaterPesticidesTrichlorfonAniline CompoundsEcologyAquatic ecosystemFenitrothionGeneral MedicinePesticideBrachionusbiology.organism_classificationPollutionAcute toxicityToxicityChlorpyrifosHexachlorocyclohexaneBulletin of Environmental Contamination and Toxicology
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