Search results for "Zolpidem"

showing 3 items of 13 documents

Intrinsic activation of GABAA receptors suppresses epileptiform activity in the cerebral cortex of immature mice

2010

SUMMARY Purpose: Activation of ionotropic c-aminobutyric acid type A (GABAA) receptors induces in immature neocortical neurons a membrane depolarization that may contribute to the higher epilepsy susceptibility in newborns. To elucidate whether depolarizing GABAergic responses enhance or attenuate epileptiform activity in the immature neocortex, we investigated the effect of agonists, antagonists, and positive modulators of GABAA receptors on epileptiform activity. Methods: We performed in vitro field potential recordings on isolated whole neocortex preparations and whole cell recordings of identified pyramidal neurons in 400-lm slices of immature (postnatal day 1–7) mice. Epileptiform acti…

medicine.medical_specialtyZolpidemNeocortexbiologyGABAA receptormusculoskeletal neural and ocular physiologynervous system diseaseschemistry.chemical_compoundEndocrinologymedicine.anatomical_structurenervous systemNeurologychemistryInternal medicinemedicinebiology.proteinGabazineGABA transporterGABAergicNeurology (clinical)PicrotoxinIonotropic effectmedicine.drugEpilepsia
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Behavioural responsiveness to picrotoxin and desipramine in adult rats prenatally exposed to different benzodiazepine receptor agonists

1995

The behavioural responsiveness to picrotoxin and desipramine was investigated in adult rats prenatally exposed to different benzodiazepine receptor agonists such as diazepam, alprazolam and zolpidem. Prenatal exposure to diazepam and alprazolam similarly potentiated the anti-immobility effect on the forced swimming test and the inhibitory effect on spontaneous motor activity of picrotoxin and desipramine and increased the seizure sensitivity to picrotoxin. Prenatal zolpidem seems to be ineffective. These data suggest that, despite the differences in their pharmacodynamic profile, prenatal exposure to diazepam and alprazolam, but not zolpidem, may have similar permanent consequences on the b…

medicine.medical_specialtyZolpidemmedicine.drug_classPharmacologychemistry.chemical_compoundInternal medicineDesipraminemedicinePharmacology (medical)Biological PsychiatryPharmacologyBenzodiazepineGABAA receptorbusiness.industrymusculoskeletal neural and ocular physiologyPsychiatry and Mental healthEndocrinologynervous systemNeurologychemistryAlprazolamNeurology (clinical)businessDiazepamPicrotoxinBehavioural despair testmedicine.drugEuropean Neuropsychopharmacology
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Prenatal exposure to diazepam and alprazolam, but not to zolpidem, affects behavioural stress reactivity in handling-naïve and handling-habituated ad…

2002

A gentle long-lasting handling produces persistent neurochemical and behavioural changes and attenuates the impairment in the behavioural reactivity to novelty induced by the prenatal exposure to diazepam (DZ) in adult male rat progeny. This study investigated the consequences of a late prenatal treatment with three GABA/BDZ R agonists (DZ) alprazolam (ALP) and zolpidem (ZOLP)), on different stress-related behavioural patterns, in non-handled (NH), short-lasting handled (SLH) and long-lasting handled (LLH) adult male rats exposed to forced swim test (FST), acoustic startle reflex (ASR) and Vogel test (VT). The effects on motor activity were evaluated in the open field and in the Skinner box…

prenatal treatment; BDZ R agonist; handling; stress-related behaviorMaleReflex StartlePyridinesprenatal exposureConvulsantsOpen fieldchemistry.chemical_compoundPregnancyPicrotoxinstress-related behaviorHabituationBenzodiazepineBehavior AnimalGeneral Neurosciencestress behaviourAge FactorsAlprazolamPrenatal Exposure Delayed EffectsFemalePsychologyhandlingmedicine.drugmedicine.medical_specialtyZolpidemmedicine.drug_classprenatal treatmentHandling PsychologicalBDZ R agonistStress PhysiologicalInternal medicineReflexmedicineAnimalsRats WistarHabituation PsychophysiologicMolecular BiologyGABA AgonistsSwimmingBenzodiazepineDiazepamAlprazolamRatsZolpidemEndocrinologychemistryAnti-Anxiety AgentsSettore BIO/14 - FarmacologiaExploratory BehaviorRatNeurology (clinical)DiazepamDevelopmental BiologyBehavioural despair testPicrotoxinBrain research
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