Search results for "arthritis"

showing 10 items of 1029 documents

Biowaiver Monographs for Immediate Release Solid Oral Dosage Forms: Piroxicam

2014

ABSTRACT Literature and experimental data relevant to the decision to allow a waiver of in vivo bioequivalence (BE) testing for the approval of immediate release (IR) solid oral dosage forms containing piroxicam in the free acid form are reviewed. Piroxicam solubility and permeability, its therapeutic use and therapeutic index, pharmacokinetic properties, data related to the possibility of excipient interactions and reported BE/bioavailability (BA), and corresponding dissolution data are taken into consideration. The available data suggest that according to the current biopharmaceutics classification system (BCS) and all current guidances, piroxicam would be assigned to BCS Class II. The ex…

DrugChemistry Pharmaceuticalmedia_common.quotation_subjectBiological AvailabilityPharmaceutical ScienceExcipientBioequivalencePharmacologyPiroxicamDosage formBiopharmaceuticsArthritis RheumatoidExcipientsFood-Drug InteractionsPiroxicamPharmacokineticsmedicineAnimalsHumansTissue Distributionmedia_commonChemistryAnti-Inflammatory Agents Non-SteroidalStereoisomerismBiopharmaceutics Classification SystemRatsBioavailabilityIntestinal AbsorptionSolubilityTherapeutic EquivalencyCaco-2 CellsHalf-Lifemedicine.drugJournal of Pharmaceutical Sciences
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Immunomodulatory drugs: Oral and systemic adverse effects

2013

Objectives: The main objectives are to present the different adverses effects of the immunomodulatory drugs that can impair the quality of life of the immunosupressed patients and study the impact of immunomodualtion on oral diseases. Immunomodulatory drugs have changed the treatment protocols of many diseases where immune functions play a central role, such as rheumatic diseases. Their effect on oral health has not been systematically investigated, however. Study Design: We review current data on the new immunomodulatory drugs from the oral health perspective based on open literature search of the topic. Results: These target specific drugs appear to have less drug interactions than earlie…

DrugPathologymedicine.medical_specialtymedia_common.quotation_subjectPlacebo-controlled studyOdontologíaReviewBioinformaticsInflammatory bowel diseaselaw.inventionImmune systemRandomized controlled triallawmedicineHumansImmunologic FactorsAdverse effectGeneral Dentistrymedia_commonOral Medicine and PathologyLupus erythematosusbusiness.industry:CIENCIAS MÉDICAS [UNESCO]medicine.diseaseCiencias de la saludstomatognathic diseasesOtorhinolaryngologyRheumatoid arthritisUNESCO::CIENCIAS MÉDICASSurgeryMouth DiseasesbusinessMedicina Oral Patología Oral y Cirugia Bucal
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Dose adjustments and discontinuation in TNF inhibitors treated patients: when and how. A systematic review of literature.

2018

Objectives To review the available evidence concerning the possibility of discontinuing and/or tapering the dosage of TNF inhibitors (TNFi) in RA patients experiencing clinical remission or low disease activity. Methods A systematic review of the literature concerning the low dosage and discontinuation of TNFi in disease-controlled RA patients was performed by evaluation of reports published in indexed international journals (Medline via PubMed, EMBASE), in the time frame from 8 April 2013 to 15 January 2016. Results We analysed the literature evaluating the efficacy and the safety of two different strategies using TNFi, decreasing dosage or discontinuation, in patients experiencing clinica…

Drugmedicine.medical_specialtymedia_common.quotation_subjectMEDLINEArthritisEtanerceptDose-Response RelationshipArthritis Rheumatoid03 medical and health sciences0302 clinical medicineRheumatologyRheumatoidInternal medicinemedicineAdalimumabHumansPharmacology (medical)030212 general & internal medicinemedia_common030203 arthritis & rheumatologyDose-Response Relationship Drugbusiness.industryTumor Necrosis Factor-alphaArthritisRemission Inductionmedicine.diseaseRheumatologyAntirheumatic Agents; Arthritis Rheumatoid; Dose-Response Relationship Drug; Humans; Remission Induction; Tumor Necrosis Factor-alpha; Rheumatology; Pharmacology (medical)DiscontinuationRheumatoid arthritisAntirheumatic AgentsDrugbusinessmedicine.drugRheumatology (Oxford, England)
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OP0023 Targeted Polymeric Nanoparticles as Diagnostic and Therapeutic Tool for Rheumatoid Arthritis

2016

Background Rheumatoid arthritis (RA) is a chronic, systemic autoimmune disease affecting joints due to the persistent synovial tissue inflammation. RA treatment has dramatically evolved in the last 20 years due to the production of biological Disease Modifying Antirheumatic Drugs (bDMARDs). However, side effects and the high costs of biological drugs are holding back their widespread usage. Moreover, some patients fail to respond to bDMARDs, for all of these reasons, DMARDs remains the main desired strategy for the treatment of RA, and Methotrexate (MTX) is still the “anchor” drug to treat RA. A successful treatment depends also on the early diagnosis, treating patients as soon as possible …

Drugrheumatoid arthritisInflammatory arthritismedia_common.quotation_subjectImmunologyArthritisInflammationPharmacologyGeneral Biochemistry Genetics and Molecular BiologymethotrexateRheumatologyIn vivomedicineImmunology and Allergyrheumatoid arthritis; nanoparticles; collagen induced arthritis; methotrexatemedia_commonbusiness.industrynanoparticleTherapeutic effectrheumatoid arthritimedicine.diseasecollagen induced arthritiscollagen induced arthritiRheumatoid arthritisImmunologyMethotrexatenanoparticlesmedicine.symptombusinessmedicine.drug
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Therapeutic administration of 3,4,5-trimethoxy-4'-fluorochalcone, a selective inhibitor of iNOS expression, attenuates the development of adjuvant-in…

2003

We have previously investigated the effects of a series of dimethoxy- and trimethoxychalcone derivatives, with various patterns of fluorination, on nitric oxide production in LPS-stimulated murine RAW 264.7. The present study was designed to determine if 3,4,5-trimethoxy-4'-fluorochalcone (CH 17) could modulate the production of NO and/or prostaglandins in vivo. On the mouse macrophage cell line RAW 264.7 CH 17 inhibited dose-dependently NO production, with an IC(50) value in the nanomolar range, and reduced PGE(2) levels by a 58% at 10 microM. This compound had no direct inhibitory effect on iNOS and COX-2 activities. NO reduction was the consequence of inhibition of the expression of iNOS…

ElectrophoresisMaleBlotting WesternNitric Oxide Synthase Type IIArthritisPharmacologyNitric OxideMonocytesNitric oxideMicechemistry.chemical_compoundChalconeChalconesIn vivoOral administrationmedicineAnimalsHumansEnzyme InhibitorsProstaglandin E2IC50Cells CulturedPharmacologyDose-Response Relationship DrugNF-kappa BMembrane ProteinsGeneral Medicinemedicine.diseaseArthritis ExperimentalIn vitroRatsIsoenzymesDose–response relationshipBiochemistrychemistryCyclooxygenase 2Prostaglandin-Endoperoxide SynthasesRats Inbred LewCyclooxygenase 1Nitric Oxide Synthasemedicine.drugNaunyn-Schmiedeberg's Archives of Pharmacology
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Note: Critical Factors in Opening Pharmaceutical Packages: a Usability Study among Healthcare Workers, Women with Rheumatoid Arthritis and Elderly Wo…

2016

This cross-sectional study compared the usability of pharmaceutical packages to determine the critical factors involved in packages with different opening mechanisms. Four packaging types (a bottle with a screw cap, a box with a pill plate, disposable plastic droppers with a container and a jar with a hinge cap) were evaluated by 45 women (nurses, older women and women with rheumatoid arthritis). Usability was evaluated for subjective measures related to the ease of opening and for objective measures related to the time needed to open the packaging, electrical muscular activity (electromyography, EMG) and ranges of motion of the upper extremities. Of the arthritic women, 13% were unable to …

Engineeringmedicine.medical_specialtymedicine.diagnostic_testbusiness.industryMechanical Engineering05 social sciencesUsabilityGeneral ChemistryElectromyographymedicine.diseaseScrew cap0506 political sciencePillRheumatoid arthritis0502 economics and businessHealth care050602 political science & public administrationPhysical therapymedicineGeneral Materials ScienceOperations managementbusinessRange of motionPharmaceutical packaging050203 business & managementPackaging Technology and Science
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Dietary acrylamide and physical performance tests: A cross-sectional analysis

2021

Background Dietary acrylamide is found in certain foods, such as deep frying, baking and roasting, and is associated with higher inflammatory and oxidative stress parameters. The association between dietary acrylamide and physical performance has not yet been explored. The aim of the study was to investigate the relationship between dietary acrylamide intake and physical performance tests in a large cohort of North American individuals affected by knee osteoarthritis or at high risk for this condition. Methods Dietary acrylamide intake was obtained through a food frequency questionnaire and reported in quartiles and as an increase in deciles. Physical performance was explored using the 20-…

EpidemiologyCross-sectional studyKneeschemistry.chemical_compoundMathematical and Statistical TechniquesSkeletal JointsMedicine and Health SciencesMedicineMusculoskeletal SystemImmune ResponseAcrylamideMultidisciplinaryCancer Risk FactorsStatisticsQConfoundingRMiddle AgedOncologyQuartileAcrylamidePhysical SciencesLegsRegression AnalysisMedicineAnatomyResearch ArticleAdultScienceImmunologyAdult; Aged; Cross-Sectional Studies; Humans; Middle Aged; AcrylamideLinear Regression AnalysisResearch and Analysis MethodsSigns and SymptomsRheumatologyEnvironmental healthOsteoarthritisLinear regressionDietary acrylamideHumansStatistical MethodsRisk factorSkeletonNutritionAgedInflammationbusiness.industryArthritisBiology and Life SciencesCell Biologymedicine.diseaseDietOxidative StressCross-Sectional StudieschemistryFoodBody LimbsMedical Risk FactorsSarcopeniaClinical MedicinebusinessMathematicsFood contaminant
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Exposure to radial extracorporeal shockwaves induces muscle regeneration after muscle injury in a surgical rat model

2019

The leading cause of training interruption in sport is a muscle injury, for which the standard treatment is nonsteroidal anti-inflammatory drugs (NSAIDs). To find alternative treatments, we investigated whether the radial extracorporeal shockwave application (rESWT) could stimulate muscle regeneration. A lesion with complete rupture (grade III muscle tear) was set in the musculus rectus femoris of 12-week-old Wistar rats, and the NSAID diclofenac, rESWT, or a combined therapy were applied on day 0, 3, and 5 directly following the surgery. Rats were euthanized at 2, 4, and 7 days after surgery and the area of muscle lesion was excised for histological and gene expression analysis to determin…

Extracorporeal Shockwave TherapyMalemedicine.medical_specialty0206 medical engineeringMuscle Fibers SkeletalUrologyH&E stain610 MedizinNeovascularization Physiologic02 engineering and technologyMyoDExtracorporealLesion03 medical and health sciences0302 clinical medicineDiclofenacDownregulation and upregulation610 Medical sciencesMyosinmedicineAnimalsPaired Box Transcription FactorsRegenerationOrthopedics and Sports MedicineRats WistarMuscle SkeletalMyoD Protein030203 arthritis & rheumatologyWound Healingbusiness.industryStandard treatmentAnti-Inflammatory Agents Non-Steroidal020601 biomedical engineeringRatsAthletic Injuriesmedicine.symptombusinessmedicine.drug
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Characterization of postural control impairment in women with fibromyalgia

2018

[EN] The main goal of this cross-sectional study was to detect whether women with fibromyalgia syndrome (FMS) have altered postural control and to study the sensory contribution to postural control. We also explored the possibility that self-induced anxiety and lower limb strength may be related to postural control. For this purpose, 129 women within an age range of 40 to 70 years were enrolled. Eighty of the enrolled women had FMS. Postural control variables, such as Ellipse, Root mean square (RMS) and Sample entropy (SampEn), in both directions (i.e. mediolateral and anteroposterior), were calculated under five different conditions. A force plate was used to register the center of pressur…

FibromyalgiaCross-sectional studyEntropyEmotionslcsh:MedicineSocial SciencesIsometric exerciseAnxietyPostural control0302 clinical medicineFibromyalgiaMedicine and Health SciencesMedicinePsychologylcsh:ScienceMusculoskeletal SystemPostural BalanceMultidisciplinaryPhysicsNeuromuscular DiseasesMiddle AgedFoamBiomechanical PhenomenaFibromyalgia syndromeNeurologyLower ExtremityEllipsesPhysical SciencesSensation DisordersAnxietyThermodynamicsSensory PerceptionFemalemedicine.symptomAnatomyResearch ArticleAdultmedicine.medical_specialtyMaterials by StructureCognitive NeuroscienceMaterials ScienceGeometryPelvis03 medical and health sciencesMotor ReactionsPhysical medicine and rehabilitationSensory CuesRheumatologyHumansMuscle StrengthAged030203 arthritis & rheumatologyHipbusiness.industrylcsh:RBiology and Life Sciencesmedicine.diseaseSample entropyPostural ControlCross-Sectional StudiesCase-Control StudiesLean body massCognitive Sciencelcsh:Qbusiness030217 neurology & neurosurgeryMathematicsNeuroscience
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Thermal imaging ruled out as a supplementary assessment in patients with fibromyalgia: A cross-sectional study

2021

Background The diagnosis of fibromyalgia syndrome (FMS) syndrome is often complicated and relies on diagnostic criteria based mostly on the symptoms reported by patients. Implementing objective complementary tests would be desirable to better characterize this population. Objective The purpose of this cross-sectional study was to compare the skin temperature at rest using thermography in women with FMS and healthy women. Methods Eighty-six women with FMS and 92 healthy controls volunteered to participate. The temperature of all participants was measured by infra-red thermography, registering the skin surface temperature (minimum, maximum and average) at rest in different areas: neck, upper…

FibromyalgiaPhysiologyCross-sectional studyKneesSensory PhysiologyBody TemperatureMedical Conditions0302 clinical medicineSkeletal JointsFibromyalgiaMedicine and Health SciencesMedicineMusculoskeletal SystemImmune Responseeducation.field_of_studyMultidisciplinaryQRSkin temperatureNeuromuscular DiseasesResearch AssessmentMiddle AgedSensory SystemsNeurologyPhysiological ParametersSomatosensory SystemThermographyThermographyMedicineLegsFemaleAnatomyResearch Articlemedicine.medical_specialtyScienceSkin surface temperatureImmunologyPopulationPainResearch and Analysis Methods03 medical and health sciencesSigns and SymptomsRheumatologyHumansIn patienteducationSkeletonResearch ErrorsInflammation030203 arthritis & rheumatologybusiness.industryBiology and Life SciencesPain Sensationmedicine.diseaseCross-Sectional StudiesBody LimbsCase-Control StudiesMann–Whitney U testPhysical therapyClinical MedicineSkin TemperaturebusinessNeck030217 neurology & neurosurgeryNeurosciencePLOS ONE
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