Search results for "butanediacetals"

showing 2 items of 2 documents

Synthesis of the aggregation pheromone of the Colorado potato beetle from its degradation product

2015

Incubation of the Colorado potato beetle aggregation pheromone, (S)-1,3-dihydroxy-3,7-dimethyl-6-octen-2-one, with antennal or leg extracts from this beetle gave 6-methyl-5-hepten-2-one as the major product. This ketone was used as a substrate in a stereoselective synthesis of the pheromone. It was attached to the butanediacetal of glycolic acid with good stereoselectivity and the desired isomer was further enriched by purification of the product of this reaction on silica gel.

ColoradoKetoneClinical BiochemistryPharmaceutical ScienceBiochemistryPheromoneschemistry.chemical_compoundbutanediacetalsDrug DiscoveryColorado potato beetleAnimalsOrganic chemistryMolecular BiologyGlycolic acidSolanum tuberosumchemistry.chemical_classificationbiologyChemistrySilica gelOrganic ChemistryColorado potato beetleSubstrate (chemistry)StereoisomerismKetonesbiology.organism_classificationColeopteraBiochemistrySex pheromoneMolecular MedicinePheromoneStereoselectivitypheromone inactivationaggregation pheromoneBioorganic & Medicinal Chemistry Letters
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Selective isomerization of a trans -butanediacetal derivative of tartaric acid with differentiating substituents at C-2 and C-3

2017

Abstract A trans-disubstituted butanediacetal derivative with two different substituents (ester and thioester) – methyl (2R,3R,5R,6R)-3-ethylsulfanylcarbonyl-5,6-dimethoxy-5,6-dimethyl-1,4-dioxane-2-carboxylate, was selectively converted to the cis derivative – methyl (2S,3R,5R,6R)-3-ethylsulfanylcarbonyl-5,6-dimethoxy-5,6-dimethyl-1,4-dioxane-2-carboxylate in high yield on a multigram scale. The product of this reaction offers the possibility for selective modification of one of the substituents, which was demonstrated by Fukuyama reduction of the thioester group.

chemistry.chemical_classification010405 organic chemistryStereochemistryOrganic Chemistryenolateselective isomerization010402 general chemistryThioester01 natural sciencesBiochemistry0104 chemical scienceschemistry.chemical_compoundFukuyama reductionbutanediacetalschemistryYield (chemistry)Drug DiscoveryTartaric acidFukuyama reductionIsomerizationDerivative (chemistry)Tetrahedron Letters
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