Search results for "computer"

showing 10 items of 30657 documents

Synthesis, antiproliferative activity, and in silico insights of new 3-benzoylamino-benzo[ b ]thiophene derivatives

2014

A new series of 3-benzoylamino-5-imidazol-5-yl-benzo[b]thiophenes and the parent amino derivatives were synthesized and screened as antitumor agents. All tested compounds showed concentration-dependent antiproliferative activity profile against HeLa cell line, exhibiting GI50 values in the low micromolar range. The most active compounds were tested in cell cycle perturbation experiments. A rapid accumulation of cells in the G2/M phase, with a concomitant reduction of cells in both the S and G0/G1 phases, was observed, suggesting that cell exposure to selected derivatives produces mitotic failure. To rationalize the biological results, the 3-benzoylamino-benzo[b]thiophenes were analyzed thro…

thiopheneVLAK protocolStereochemistryIn silicoCellAntineoplastic AgentsMechanism of actionHeLa CellHeLaAntineoplastic AgentStructure-Activity Relationship3-Benzoylamino-5-imidazol-4-yl-benzo[b]Settore BIO/10 - BiochimicaDrug DiscoverymedicineHumansMoietyComputer SimulationMitosisCell ProliferationPharmacologyAntitumor agentsbiologyDose-Response Relationship DrugMolecular StructureChemistryDrug Discovery3003 Pharmaceutical ScienceMedicine (all)Cell CycleOrganic ChemistryAntitumor agentG2/M phaseGeneral MedicineSettore CHIM/06 - Chimica OrganicaHeLa cell linebiology.organism_classificationSettore CHIM/08 - Chimica Farmaceuticamedicine.anatomical_structureCell cultureSettore CHIM/03 - Chimica Generale E InorganicathiophenesAntimitotic AgentTopoisomerase-II InhibitorDrug Screening Assays AntitumorHeLa CellsHuman
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Overview of Power Electronic Switches: A Summary of the Past, State-of-the-Art and Illumination of the Future.

2020

As the need for green and effective utilization of energy continues to grow, the advancements in the energy and power electronics industry are constantly driven by this need, as both industries are intertwined for obvious reasons. The developments in the power electronics industry has over the years hinged on the progress of the semiconductor device industry. The semiconductor device industry could be said to be on the edge of a turn into a new era, a paradigm shift from the conventional silicon devices to the wide band gap semiconductor technologies. While a lot of work is being done in research and manufacturing sectors, it is important to look back at the past, evaluate the current progr…

thyristorsEngineeringinsulated gate bipolar transistorslcsh:Mechanical engineering and machinery02 engineering and technologyReviewbipolar transistors01 natural sciencesElectronic switchpower semiconductor devicesPower electronics0103 physical sciences0202 electrical engineering electronic engineering information engineeringPower semiconductor devicelcsh:TJ1-1570Electrical and Electronic Engineering010302 applied physicsbusiness.industrypower semiconductor switchesMechanical Engineering020208 electrical & electronic engineeringThyristorSemiconductor deviceVDP::Teknologi: 500Work (electrical)Control and Systems EngineeringParadigm shiftState (computer science)businessTelecommunicationspower transistorsMicromachines
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Can we automate expert-based journal rankings? Analysis of the Finnish publication indicator

2020

The publication indicator of the Finnish research funding system is based on a manual ranking of scholarly publication channels. These ranks, which represent the evaluated quality of the channels, are continuously kept up to date and thoroughly reevaluated every four years by groups of nominated scholars belonging to different disciplinary panels. This expert-based decision-making process is informed by available citation-based metrics and other relevant metadata characterizing the publication channels. The purpose of this paper is to introduce various approaches that can explain the basis and evolution of the quality of publication channels, i.e., ranks. This is important for the academic …

tiedelehdetfeature importanceComputer scienceProcess (engineering)rankinglistatjulkaisutmedia_common.quotation_subjectLibrary and Information Sciences050905 science studiestutkimusrahoitusautomaatioperformance-based research funding systemFeature (machine learning)Quality (business)automationmedia_commonbusiness.industry05 social sciencesData scienceAutomationComputer Science ApplicationsMetadatamachine learningkoneoppiminenRanking0509 other social sciences050904 information & library sciencesbusinessCitationarviointiDisciplinetieteellinen julkaisutoimintaJournal of Informetrics
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External Assessors as “Reviewers” for Quality Assurance of Open Access Journals

2017

tiedelehdetopen accessexternal assessorsSocial Psychologyscholary researchbusiness.industryCommunicationscientific journalsjournalslaatu030230 surgeryHuman-Computer InteractionWorld Wide Web03 medical and health sciences0302 clinical medicinereviewersqualityopen access journals030212 general & internal medicinevertaisarviointita518businessQuality assurancetieteellinen julkaisutoiminta
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In Pursuit of Measuring Pre-reflective Music Listening Experiences

2022

While the diverse effects and uses of music and sound have been extensively documented within music psychology, relatively little attention has been paid to the process and experience of listening itself. Previous literature have, however, considered different ways of attending to sounds via the concept of listening modes, which highlights the different ways and strategies through which listeners intentionally orientate themselves to the activity of listening and creating the experiential meaning of the sound. In this paper, we continue on these lines by focusing on the very basic attentional dispositions for listening that often remain unconscious. As op posed to more deliberate and intent…

tietoisuushuman computer interaction (HCI)musiikkimusiikkipsykologiapre-reflective experiencesound and music computingkuunteleminenembodied cognitionmodes of listeningkokemuksetmusicääni (fysikaaliset ilmiöt)merkitys (tärkeys)tarkkaavaisuuslisteningimagination
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Applying video games in language learning and teaching : the learner perspective: a case study

2012

Tutkielman tarkoituksena on selvittää oppijoiden näkemyksiä videopelien nykyisistä ja mahdollisista käyttötavoista kieltenopetuksessa ottaen huomioon koehenkilöiden koulutus- ja pelaajataustan. Pelitutkimusta ei ole vielä tehty kauaa, joten ala on hajanainen, mutta tämä tutkimus pohjautuu tietokoneavusteisen oppimisen (CALL) ja videopeleihin perustuvan oppimisen (DGBL) tutkimukseen. CALL ei keskity erikseen pelien käyttöön tai käsittelee enemmän kieltenoppimiseen tehtyjä ohjelmia, kun taas peleihin perustuvassa opetuksessa kielet eivät ole erityisasemassa. Oppimistuloksia ja oppijakokemuksia pelien käytöstä on kerätty lähinnä esikoulu- ja peruskouluikäisiltä, joten lukiolaiskokeilu täydentä…

tietokoneavusteinen opettaminencomputer-assisted learningdigital game-based learningcomputer-assisted teachingpeleihin perustuva opetusVideopelittietokoneavusteinen oppiminenvideo gameslanguage teachingkielen oppiminenlanguage learning
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On the rocky road of reading : effects of computer-assisted reading intervention for at-risk children

2010

tietokoneavusteinen opetusEkapeliPitkittäistutkimuslukeminencomputer-assisted instructionchildrenat risk populationsriskiryhmäterityisopetuslukutaitotietokoneavusteinen oppiminenremedial readinglukihäiriötreading educationlapsetreading disabilities
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A Study on the Assessment of Introductory Computational Thinking via Scratch Programming in Primary Schools

2018

Computational thinking (CT), a transversal intellectual foundation integral to computer science, is making its way into compulsory comprehensive education worldwide. Students are expected to attain skills and knowledge in such interdisciplinary CT principles as Algorithmic thinking, Data representation, and Debugging. Problem-solving by designing and manipulating interactive media with Scratch, a graphical programming tool, is popular especially at the primary school level. However, there has been confusion regarding how introductory CT can be operationalized for educational practice. Teachers and students need research-based knowledge for setting appropriate learning goals in addition to i…

tietokoneavusteinen opetusgraphical programmingComputer scienceassessment02 engineering and technologyalakouluprimary schoolFormative assessmentcomputational thinking020204 information systemsComputingMilieux_COMPUTERSANDEDUCATION0202 electrical engineering electronic engineering information engineeringMathematics educationta516computer.programming_languageVisual programming languageta113educationOperationalizationConceptualizationbusiness.industryComputational thinking05 social sciences050301 educationScratchAssessment for learningScratchohjelmointiongelmanratkaisubusiness0503 educationcomputerInteractive media
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EFL teachers talking about their use of computers at work : a discourse-analytic study

2003

tietokoneavusteinen opetusinterviewsqualitativecomputer usediscursive researchEFL teachersdiskurssianalyysi
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The effect of using computer literate game in the teaching of reading literacy skills in Zambia

2008

tietokoneavusteinen opetuslukutaitokirjoitustaitoSambiacurriculumZambiacomputer gamesliteracyliterate gameopetusphonemeopetussuunnitelmat
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