Search results for "cycle"

showing 10 items of 3119 documents

Aza-isoindolo and isoindolo-azaquinoxaline derivatives with antiproliferative activity

2015

Abstract Three new ring systems, pyrido[2′,3′:3,4]pyrrolo[1,2- a ]quinoxalines, pyrido[3′,2′:3,4]pyrrolo[1,2- a ]quinoxalines and pyrido[2′,3′:5,6]pyrazino[2,1- a ]isoindoles, were synthesized through an aza-substitution on the already active isoindolo-quinoxaline system and in particular in the position 7 or 4 of the isoindole moiety and in position 5 of the quinoxaline portion. All new compounds were screened by the National Cancer Institute (Bethesda, MD) against a panel of 60 human tumor cell lines. Biological results of the most active derivatives, with pGI 50 values between 7.09 and 7.27, confirmed the importance of the presence of methoxy substituents for biological activity. The ant…

QuinoxalineIsoindolesAzaisoindolo-quinoxalinesStereochemistryAntiproliferative activity; Apoptosis; Azaisoindolo-quinoxalines; DNA interaction; Isoindolo-azaquinoxalines; Quinoxalines; Antineoplastic Agents; Apoptosis; Aza Compounds; Cell Line Tumor; Cell Proliferation; Dose-Response Relationship Drug; Drug Screening Assays Antitumor; Humans; Isoindoles; Molecular Structure; Quinoxalines; Structure-Activity Relationship; Drug Discovery3003 Pharmaceutical Science; Organic Chemistry; Pharmacology; Medicine (all)ApoptosisAntineoplastic AgentsAntiproliferative activityIsoindolesRing (chemistry)Drug Screening AssaysCell LineDose-Response Relationshipchemistry.chemical_compoundStructure-Activity RelationshipQuinoxalineCell Line TumorQuinoxalinesDrug DiscoverymedicineMoietyHumansAntiproliferative activity; Apoptosis; Azaisoindolo-quinoxalines; DNA interaction; Isoindolo-azaquinoxalines; Quinoxalines; Drug Discovery3003 Pharmaceutical Science; Organic Chemistry; PharmacologyCell ProliferationPharmacologyAza CompoundsAzaisoindolo-quinoxalineTumorDose-Response Relationship DrugMolecular StructureDrug Discovery3003 Pharmaceutical ScienceMedicine (all)Organic ChemistryApoptosiBiological activityGeneral MedicineAntitumorCell cycleSettore CHIM/08 - Chimica FarmaceuticaDNA interactionSettore ING-IND/22 - Scienza E Tecnologia Dei MaterialiMechanism of actionchemistryIsoindolo-azaquinoxalineDrug Screening Assays Antitumormedicine.symptomDrugIsoindoleIsoindolo-azaquinoxalines
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The endoperoxide ascaridol shows strong differential cytotoxicity in nucleotide excision repair-deficient cells

2011

Targeting synthetic lethality in DNA repair pathways has become a promising anti-cancer strategy. However little is known about such interactions with regard to the nucleotide excision repair (NER) pathway. Therefore, cell lines with a defect in the NER genes ERCC6 or XPC and their normal counterparts were screened with 53 chemically defined phytochemicals isolated from plants used in traditional Chinese medicine for differential cytotoxic effects. The screening revealed 12 drugs that killed NER-deficient cells more efficiently than proficient cells. Five drugs were further analyzed for IC50 values, effects on cell cycle distribution, and induction of DNA damage. Ascaridol was the most effe…

RAD23BDNA RepairDNA repairDNA damageCyclohexane MonoterpenesBiologyToxicologyCell LineInhibitory Concentration 50HumansCytotoxic T cellMedicine Chinese TraditionalPharmacologyDose-Response Relationship DrugCell cycleAntineoplastic Agents PhytogenicMolecular biologyPeroxidesG2 Phase Cell Cycle CheckpointsCell cultureCancer cellMonoterpenesM Phase Cell Cycle CheckpointsReactive Oxygen SpeciesDNA DamageDrugs Chinese HerbalNucleotide excision repairToxicology and Applied Pharmacology
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Progettare città nel tempo della metamorfosi

2013

Metamorfosi è una potente parola-guida della contemporaneità. E’ un impegno di cui numerosi segni ci facevano intravedere la necessità durante gli anni propulsivi della globalizzazione e molteplici indizi tracciavano la strada da percorrere. Ma, anestetizzati dalle aporie dello sviluppo, li abbiamo ignorati, emarginandoli nella ecosofia o reagendo in modo impulsivo con seducenti inni alla decrescita felice. Oggi invece gli anni recessivi di una crisi che non è una semplice stagione di attraversamento ci chiedono la responsabilità di un mutamento di paradigma che conduca alla metamorfosi ecologica, culturale, economica, sociale e politica. Ma il mutamento sarà soprattutto urbano, perché vivi…

RECYCLE URBAN METAMORPHOSIS URBAN REGENERATION CREATIVE CITYSettore ICAR/21 - Urbanistica
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From Buildings' End of Life to Aggregate Recycling under a Circular Economic Perspective: A Comparative Life Cycle Assessment Case Study

2021

The demolition of buildings, apart from being energy intensive and disruptive, inevitably produces construction and demolition waste (C&Dw). Unfortunately, even today, the majority of this waste ends up underexploited and not considered as valuable resources to be re-circulated into a closed/open loop process under the umbrella of circular economy (CE). Considering the amount of virgin aggregates needed in civil engineering applications, C&Dw can act as sustainable catalyst towards the preservation of natural resources and the shift towards a CE. This study completes current research by presenting a life cycle inventory compilation and life cycle assessment case study of two buildin…

RECYCLINGProcess (engineering)CIRCULAR ECONOMYGeography Planning and Development0211 other engineering and technologiesTJ807-830MATERIAU DE CONSTRUCTION02 engineering and technologyCONSTRUCTION AND DEMOLITION WASTE-010501 environmental sciencesManagement Monitoring Policy and LawTD194-19501 natural sciences7. Clean energyRenewable energy sources12. Responsible consumptionRECYCLAGE (MATER)RECYCLAGE DES MATERIAUXDUREE DE VIE021105 building & construction11. SustainabilityGE1-350Life-cycle assessmentRECYCLED AGGREGATES0105 earth and related environmental sciencesTransportation planningCONSTRUCTION (EXECUTION)LIFE CYCLE ASSESSMENTEnvironmental effects of industries and plantsEND OF LIFERenewable Energy Sustainability and the EnvironmentCircular economyEnvironmental economicsNatural resourceREUTILISATIONEnvironmental sciences[SPI.GCIV]Engineering Sciences [physics]/Civil Engineeringrecycled aggregateRESIDU INDUSTRIELDemolition waste13. Climate actionSustainability[SDE]Environmental SciencesDemolitionGRANULAT RECYCLEGATE-TO-GRAVEBusiness
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p38α deficiency and oxidative stress cause cytokinesis failure in hepatocytes.

2015

Cytokinesis is the last step in mitosis and it implies re-organization of the actin cytoskeleton. Its failure is one of the major mechanisms of polyploidy and binucleation in mammals. Our aims were 1) to assess the role of redox-sensitive p38α MAPK in cytokinesis by studying the liver of wild type mice or liver-specific p38α knock-out mice; 2) to assess the role of oxidative stress associated with hepatocyte isolation on cytokinesis. When p38α was down-regulated in hepatocytes, MK2 phosphorylation on threonine 334 was completely abrogated. Activation of MNK-1, required for abscission of the intercellular bridge, was diminished. Key proteins of the RhoA pathway (phospho-PRK2, nuclear phospho…

RHOAmacromolecular substancesBiologyCell cycleCofilinActin cytoskeletonBiochemistryCell biologyCytosolPhysiology (medical)biology.proteinMitosisCytokinesisActinFree radical biologymedicine
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Photochemistry of Fluorinated Heterocyclic Compounds. An Expedient Route for the Synthesis of Fluorinated 1,3,4-Oxadiazoles and 1,2,4-Triazoles

2004

The photochemistry of some 3-N-alkylamino-5-perfluoroalkyl-1,2,4-oxadiazoles in the presence of nitrogen nucleophiles such as ammonia and primary and secondary aliphatic amines has been investigated. The primary photolytic intermediate from the cleavage of the ring O-N bond follows two distinct and competing pathways leading to (i). 5-perfluoroalkyl-1,3,4-oxadiazoles, through the ring contraction-ring expansion photoisomerization route favored by the presence of the base or (ii). 5-perfluoroalkyl-1,2,4-triazoles, through the intervention, as an internal nucleophile, of the exocyclic N-alkylamino moiety of the oxadiazole followed by the attack of the external nitrogen nucleophile and subsequ…

RING-PHOTOISOMERIZATIONPrimary (chemistry)PhotoisomerizationFLUORO HETEROCYCLESChemistryOrganic ChemistryOxadiazoleContext (language use)Settore CHIM/06 - Chimica OrganicaRing (chemistry)Photochemistrychemistry.chemical_compoundNucleophile124-OXADIAZOLE DERIVATIVESMoiety5-MEMBERED HETEROCYCLESAliphatic compoundPHOTOINDUCED MOLECULAR-REARRANGEMENTSThe Journal of Organic Chemistry
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Using deep learning to generate synthetic B-mode musculoskeletal ultrasound images

2020

Background and objective\ud Deep learning approaches are common in image processing, but often rely on supervised learning, which requires a large volume of training images, usually accompanied by hand-crafted labels. As labelled data are often not available, it would be desirable to develop methods that allow such data to be compiled automatically. In this study, we used a Generative Adversarial Network (GAN) to generate realistic B-mode musculoskeletal ultrasound images, and tested the suitability of two automated labelling approaches.\ud \ud Methods\ud We used a model including two GANs each trained to transfer an image from one domain to another. The two inputs were a set of 100 longitu…

RM695_Physicalultrasoundmusclegenerative adversarial networkmedical imagingdeep learningsynthetic imagelihaksetQPQA76koneoppiminenkuvantaminenultraäänitutkimuscycleGAN
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Vertical transmission of naturally occurring Bunyamwera and insect-specific flavivirus infections in mosquitoes from islands and mainland shores of L…

2018

Background Many arboviruses transmitted by mosquitoes have been implicated as causative agents of both human and animal illnesses in East Africa. Although epidemics of arboviral emerging infectious diseases have risen in frequency in recent years, the extent to which mosquitoes maintain pathogens in circulation during inter-epidemic periods is still poorly understood. This study aimed to investigate whether arboviruses may be maintained by vertical transmission via immature life stages of different mosquito vector species. Methodology We collected immature mosquitoes (egg, larva, pupa) on the shores and islands of Lake Baringo and Lake Victoria in western Kenya and reared them to adults. Mo…

RNA virusesMale0301 basic medicineViral DiseasesAnopheles GambiaevirusesAnopheles gambiaeRC955-962Marine and Aquatic SciencesDisease VectorsPathology and Laboratory MedicineMosquitoes0302 clinical medicineAedesArctic medicine. Tropical medicineMedicine and Health SciencesChikungunya VirusbiologyPupaAnophelesEukaryotavirus diseasesGene PoolInsectsCulexInfectious DiseasesArboviral InfectionsMedical MicrobiologyViral PathogensLarvaVirusesFemalePublic aspects of medicineRA1-1270PathogensResearch ArticleFreshwater EnvironmentsArthropodaAlphaviruses030231 tropical medicineZoologyMosquito VectorsAedes aegyptiAedes AegyptiMicrobiologyArbovirusTogaviruses03 medical and health sciencesAedes luteocephalusSpecies SpecificityAnophelesparasitic diseasesCulex pipiensGeneticsmedicineAnimalsBunyamwera virusMicrobial PathogensAedesEvolutionary BiologyLife Cycle StagesPopulation BiologyFlavivirusEcology and Environmental SciencesfungiOrganismsPublic Health Environmental and Occupational HealthBiology and Life SciencesAquatic EnvironmentsBodies of Watermedicine.diseasebiology.organism_classificationInvertebratesKenyaInsect VectorsSpecies InteractionsLakes030104 developmental biologyVector (epidemiology)Earth SciencesArbovirusesPopulation GeneticsPLOS Neglected Tropical Diseases
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The radiosensitization effect of titanate nanotubes as a new tool in radiation therapy for glioblastoma: A proof-of-concept

2013

Abstract Background and purpose One of the new challenges to improve radiotherapy is to increase the ionizing effect by using nanoparticles. The interest of titanate nanotubes (TiONts) associated with radiotherapy was evaluated in two human glioblastoma cell lines (SNB-19 and U87MG). Materials and methods Titanate nanotubes were synthetized by the hydrothermal treatment of titanium dioxide powder in a strongly basic NaOH solution. The cytotoxicity of TiONts was evaluated on SNB-19 and U87MG cell lines by cell proliferation assay. The internalization of TiONts was studied using Transmission Electron Microscopy (TEM). Finally, the effect of TiONts on cell radiosensitivity was evaluated using …

Radiation-Sensitizing AgentsCell SurvivalDNA repairCellApoptosisFlow cytometryCell Line TumormedicineHumansRadiology Nuclear Medicine and imagingRadiosensitivityClonogenic assayCytotoxicityTitaniumNanotubesmedicine.diagnostic_testBrain NeoplasmsChemistryCell growthCell CycleHematologyCell cyclemedicine.anatomical_structureOncologyBiophysicsGlioblastomaReactive Oxygen SpeciesDNA DamageRadiotherapy and Oncology
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A radiosensitizing effect of artesunate in glioblastoma cells is associated with a diminished expression of the inhibitor of apoptosis protein surviv…

2011

Abstract Background and purpose Novel strategies to overcome an irradiation resistant phenotype may help to increase therapeutic efficacy in glioblastoma multiforme. The present study aimed to elucidate radiation sensitizing properties of artesunate, a semi synthetic derivate of artemisinin and to assess factors involved in this effect. Materials and methods LN229 and U87MG cells were treated with various concentrations of artesunate and radiation response was determined by a colony forming assay. Cell numbers, apoptosis induction, cell cycle distribution, and DNA repair following combined modality treatment were monitored by MTT-, caspase 3/7 assay, cytofluorometry, and γ-H2AX foci formati…

Radiation-Sensitizing AgentsDNA RepairCell SurvivalSurvivinArtesunateDown-RegulationCaspase 3ApoptosisInhibitor of apoptosisInhibitor of Apoptosis Proteinschemistry.chemical_compoundCell Line TumorSurvivinHumansRadiology Nuclear Medicine and imagingClonogenic assayDose-Response Relationship DrugBrain NeoplasmsCell CycleHematologyCell cycleArtemisininsXIAPNeoplasm ProteinsOncologychemistryArtesunateApoptosisCancer researchGlioblastomaRadiotherapy and oncology : journal of the European Society for Therapeutic Radiology and Oncology
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