Search results for "design."

showing 10 items of 5715 documents

A biphasic calcium phosphate coating for potential drug delivery affects early osseointegration of titanium implants.

2016

Background Calcium phosphate (CaP) surface coatings may accelerate osseointegration and serve as a drug delivery system for mineral-binding biomolecules. In a pilot study, the impact of a commercially available, thin CaP coating on early osseous bone remodeling was compared with a modern, subtractive-treated rough surface (SLA-like) in an animal trial. Methods In 16 rabbits, 32 endosseous implants (CaP; n = 16, SLA-like; n = 16) were bilaterally inserted in the proximal tibia after randomization. After 2 and 4 weeks, bone-implant contact (BIC;%) in the cortical (cBIC) and the trabecular bone (sBIC) as well as volume of bone within the screw thread with the highest amount of new-formed bone …

Calcium PhosphatesCancer Researchchemistry.chemical_elementDentistry02 engineering and technologyengineering.materialCalciumOsseointegrationPathology and Forensic MedicineBone remodeling03 medical and health sciencesRandom Allocation0302 clinical medicineDrug Delivery SystemsCoatingOsseointegrationAnimalsDental ImplantsTitaniumChemistrybusiness.industryfungiDental Implantation Endosseous030206 dentistry021001 nanoscience & nanotechnologyBiphasic calcium phosphateTrabecular boneOtorhinolaryngologyDental Prosthesis DesignDrug deliveryModels AnimalengineeringPeriodonticsRabbitsOral Surgery0210 nano-technologyNuclear medicinebusinessTitaniumJournal of oral pathologymedicine : official publication of the International Association of Oral Pathologists and the American Academy of Oral Pathology
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Inhibition of HSP70: a challenging anti-cancer strategy.

2012

HSP70 is a chaperone that accumulates in the cells after many different stresses promoting cell survival in response to the adverse conditions. In contrast to normal cells, most cancer cells abundantly express HSP70 at the basal level to resist to various insults at different stages of tumorigenesis and during anti-cancer treatment. This cancer cells addiction for HSP70 is the rational for its targeting in cancer therapy. Much effort has been dedicated in the last years for the active search of HSP70 inhibitors. Additionally, the recent clinical trials on highly promising inhibitors of another stress protein, HSP90, showed compensatory increase in HSP70 levels and raised the question of nec…

Cancer ResearchAntineoplastic AgentsApoptosismedicine.disease_cause03 medical and health sciences0302 clinical medicineImmune systemStress PhysiologicalHeat shock proteinNeoplasmsmedicineAutophagyAnimalsHumansHSP70 Heat-Shock ProteinsHSP90 Heat-Shock ProteinsMolecular Targeted Therapy030304 developmental biology0303 health sciencesbiologyHsp903. Good healthNeoplasm ProteinsProtein Structure TertiaryClinical trialOncologyApoptosisDrug Resistance Neoplasm030220 oncology & carcinogenesisChaperone (protein)Drug DesignCancer cellImmunologybiology.proteinCancer researchDrug Screening Assays AntitumorCarcinogenesisMolecular ChaperonesCancer letters
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From a Better Understanding of the Mechanisms of Action of Histone Deacetylases Inhibitors to the Progress of the Treatment of Malignant Lymphomas an…

2017

Background Notable progress has been made in chemo- and immunotherapy of B-cell lymphomas, but less in the treatment of T-cell lymphomas. Objective Histone deacetylases inhibitors are a potentially useful therapeutic mean, as an epigenetic dysregulation is present in lymphomas, and especially in T-cell types. We aimed to study the progress made in this area. Method A mini-review was achieved using the articles published in PubMed in the last two years and the new patents made in this field. Results Histone deacetylases inhibitors are involved in the derepression of tumor suppressor genes through a histone deacetylase-mediated transcriptional process. Their inhibition is followed by cell cyc…

Cancer ResearchDrug exportmedicine.medical_treatmentCellular differentiationAntineoplastic Agents010402 general chemistryLymphoma T-Cell01 natural sciencesHistone DeacetylasesRomidepsinPatents as TopicDrug DiscoveryPlasma Cell MyelomamedicineAnimalsHumansPharmacology (medical)Epigeneticsbiology010405 organic chemistrybusiness.industryDrug SynergismGeneral MedicineImmunotherapymedicine.diseasePeripheral T-cell lymphoma0104 chemical sciencesHistone Deacetylase InhibitorsHistoneOncologyDrug DesignImmunologyCancer researchbiology.proteinbusinessMultiple Myelomamedicine.drugRecent patents on anti-cancer drug discovery
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Cathepsin D expression levels in nongynecological solid tumors: clinical and therapeutic implications.

2004

Cathepsin D is a lysosomal acid proteinase which is involved in the malignant progression of breast cancer and other gynecological tumors. Clinical investigations have shown that in breast cancer patients cathepsin D overexpression was significantly correlated with a shorter free-time disease and overall survival, whereas in patients with ovarian or endometrial cancer this phenomenon was associated with tumor aggressiveness and a degree of chemoresistance to various antitumor drugs such as anthracyclines, cis-platinum and vinca alkaloids. Therefore, a lot of research has been undertaken to evaluate the role and the prognostic value of cathepsin D also in other solid neoplasms. However, conf…

Cancer ResearchPathologymedicine.medical_specialtyLung NeoplasmsSkin NeoplasmsCathepsin DAntineoplastic AgentsBiologyDigestive System NeoplasmsCathepsin DMetastasisCentral Nervous System NeoplasmsBreast cancerSurgical oncologyNeoplasmsmedicineBiomarkers TumorNeoplasmHumansClinical significanceThyroid NeoplasmsMelanomaEndometrial cancerGeneral Medicinecathepsin D lysosomal proteinases matrix-metalloproteinases metastasis neoplasm plasminogen activator prognosis tumor progressionmedicine.diseaseNeoplasm ProteinsOncologyTumor progressionHead and Neck NeoplasmsDrug DesignCancer researchDisease ProgressionLysosomesUrogenital NeoplasmsClinicalexperimental metastasis
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Association study of 44 candidate genes with depressive and anxiety symptoms in post-partum women.

2009

The post-partum period is a time of extreme vulnerability for a whole spectrum of psychiatric disorders. Delivery may be considered an important risk factor in genetically susceptible women. Five hundred and eight SNPs in 44 genes at candidate pathways putatively related to mood changes after delivery were genotyped in a multicenter cohort of 1804 women from Spain. Participants completed two scales at 2-3 days, 8 weeks, and 32 weeks post-partum, the Edinburgh Post-partum Depression Scale (EPDS) and the Spielberger State-Trait Anxiety Inventory (STAI). Those women who scored 9 or more on EPDS were evaluated for major depression using the Diagnostic Interview for Genetics Studies (DIGS) adapt…

Candidate genemedicine.medical_specialtyTime FactorsGenotypeAnxietyPolymorphism Single NucleotideWhite PeopleCohort StudiesDepression PostpartumInternal medicinePost-hoc analysisProtein Kinase C betamedicineHumansPsychiatryBiological PsychiatrySerotonin transporterDepression (differential diagnoses)Protein Kinase CRetrospective StudiesPsychiatric Status Rating ScalesSerotonin Plasma Membrane Transport ProteinsbiologyPostpartum PeriodRepeated measures designPsychiatry and Mental healthMoodSpainCohortbiology.proteinDopa DecarboxylaseAnxietyFemalemedicine.symptomPsychologyGenome-Wide Association StudyJournal of psychiatric research
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The mixed capacitated general routing problem with turn penalties

2011

In this paper we deal with the mixed capacitated general routing problem with turn penalties. This problem generalizes many important arc and node routing problems, and it takes into account turn penalties and forbidden turns, which are crucial in many real-life applications, such as mail delivery, waste collection and street maintenance operations. Through a polynomial transformation of the considered problem into a Generalized Vehicle routing problem, we suggest a new approach for solving this new problem by transforming it into an Asymmetric Capacitated Vehicle routing problem. In this way, we can solve the new problem both optimally and heuristically using existing algorithms. A powerfu…

Capacitated vehicle routing problemMathematical optimizationRouting problemsPolynomial transformationReal-life applicationsTurn penaltiesCapacitated general routing problemRouting algorithmsVehicle Routing ProblemsTransformationPolynomial transformationsArtificial IntelligenceVehicle routing problemDestination-Sequenced Distance Vector routingGeneral routing problemMathematicsta113Average deviationStatic routingWaste collectionNode (networking)General EngineeringSolution methodsMaintenance operationsVehicle routingComputer Science ApplicationsMemetic algorithmsBenchmark (computing)Network routingMemetic algorithmRouting (electronic design automation)MATEMATICA APLICADAAlgorithmsExpert Systems with Applications
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Il principio di gerarchia delle resistenze capacity design

2012

The devastating effects generated by earthquakes occurred in different parts of the world have attract at a major interest in Earthquake Engineering. This branch of Structural Engineering studies the response and capacity of structural systems subjected to seismic actions, and develops design and prediction methods aimed at achieving adequate safety standards in presence of seismic events. A strategy used for the seismic prediction of RC structures, based on the capacity design of structural elements is the "hierarchy of strengths" (HS) principle. The paper shows how a proper use of the HS capacity design method can be included within the seismic design of RC structures achieving high level…

Capacity Design Duttilità Cerniere Plastiche Dissipazione di Energia.Settore ICAR/08 - Scienza Delle Costruzioni
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Retrofitting of Existing Steel MR-Frames by Encasing the Columns

2005

Summary The study concerns the behaviour of steel MR-frames subjected to vertical and lateral forces, not properly designed according to capacity design criteria, and upgraded by means of encasing the steel columns with concrete having different grade. The purpose of the paper is to examine if the proposed technique allows one to adequately increase the lateral stiffness and the resistance of the frames. Pushover analyses on multi-storey frames are performed trough a non-linear calculus program, able to take into account of the second order effects. The behaviour of frames with encased columns was compared with those of the bare frames, highlighting that with the proposed technique it is po…

Capacity designEngineeringSteel columnssteel moment resisting frames refurbischement of the columns by encasing.business.industryHingeRetrofittingLateral stiffnessLimit state designStructural engineeringDuctilitybusinessJoint (geology)IABSE Symposium, Lisbon 2005: Structures and Extreme Events
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Approximate Algorithm for Fast Capacity Provisioning in WANs with Trade-Off between Performance and Cost under Budget Constraint

2014

Due to the emergence of Software Defined Networking (SDN) with the idea of centralized control over computer networks, the Capacity and Flow Assignment Problem (CFA) may be approached in a classical non-distributed fashion in real-life scenarios. The question arises whether a heuristical approach to this NP-complete problem is of any use in practice.

Capacity provisioningFlow (mathematics)Computer scienceDistributed computingControl (management)Routing (electronic design automation)Trade-offSoftware-defined networkingAssignment problemBudget constraint
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A critical appraisal of capillary electrochromatography.

2002

Although still in its infancy, CEC promises some advantages over competitive techniques for separating charged analytes including biomolecules.

Capillary electrochromatographyCritical appraisalSpectrometry Mass Electrospray IonizationChemistryElectrophoresis CapillaryProteinsNanotechnologyEquipment DesignPeptidesChromatography High Pressure LiquidAnalytical ChemistryAnalytical chemistry
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