Search results for "dication"

showing 10 items of 733 documents

Selective Inhibition of STAT3 with Respect to STAT1: Insights from Molecular Dynamics and Ensemble Docking Simulations

2016

STAT3 protein, which is known to be involved in cancer development, is a promising target for anticancer therapy. Successful inhibitors of STAT3 should not affect an activity of closely related protein STAT1, which makes their development challenging. The mechanisms of selectivity of several existing STAT3 inhibitors are not clear. In this work, we studied molecular mechanisms of selectivity of 13 experimentally tested STAT3 inhibitors by means of extensive molecular dynamics and ensemble docking simulations. It is shown that all studied inhibitors bind to the large part of the protein surface in an unspecific statistical manner. The binding to the dimerization interface of the SH2 domain, …

STAT3 Transcription Factor0301 basic medicine[ SDV.BBM.BP ] Life Sciences [q-bio]/Biochemistry Molecular Biology/BiophysicsStereochemistryGeneral Chemical Engineering[SDV.CAN]Life Sciences [q-bio]/CancerMolecular Dynamics SimulationLibrary and Information SciencesBiologySelective inhibitionSH2 domain01 natural sciencesMolecular Docking SimulationSubstrate Specificity[ SDV.CAN ] Life Sciences [q-bio]/Cancersrc Homology Domains03 medical and health sciencesMolecular dynamics[SDV.SP.MED]Life Sciences [q-bio]/Pharmaceutical sciences/Medication[CHIM]Chemical SciencesSTAT1STAT3ComputingMilieux_MISCELLANEOUS010405 organic chemistry[ SDV.SP.MED ] Life Sciences [q-bio]/Pharmaceutical sciences/MedicationGeneral Chemistry0104 chemical sciences3. Good healthComputer Science ApplicationsMolecular Docking Simulation[SDV.BBM.BP]Life Sciences [q-bio]/Biochemistry Molecular Biology/BiophysicsSTAT1 Transcription Factor030104 developmental biologyDocking (molecular)Biophysicsbiology.proteinSelectivity
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Domestication of a Robotic Medication-Dispensing Service Among Older People in Finnish Lapland

2020

This paper presents a case study on a robotic medication-dispensing service used in the everyday lives of older people in Finnish Lapland through the concept of domestication. The study took an ethnographic approach. A total of 11 service users, practical nurses, and other health-care professionals participated; the service users averaged age 81 years (M= 81.4, SD = 5.4). The data comprised semistructured interviews complemented by observations and photographs at service users’ homes. We concluded that the domestication of the service was successful, although the service users sometimes felt that it limited their lives. The service users stated that learning and subsequently using the servi…

Service (business)harvaan asutut alueetSocial PsychologySocial networkAging in placeehealthbusiness.industryCommunicationApplied psychologyrobotic medication-dispenserCognitiondigital competenceolder peopleHuman-Computer Interactiondomesticationsparsely populated areaEthnographyrobotiteHealthDomesticationbusinessOlder peoplePsychologyikääntyneetHuman Technology
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Semantic traffic applications based on DatexII

2009

In this work we demonstrate a particular use of ontologies based on the European specifications DATEXII. These specifications are designed and developed as a traffic and travel data exchange mechanism by a European task force to set up and standardise the interface between traffic control and information centres. It is the reference for applications that are developed and implemented in Europe.This language describes concepts and structures of data related to traffic, but the description is just syntactic, not semantic. Therefore the objective to be reached in this part of the research has been to develop a semantic description in order to carry out some applications like syndication and a …

Set (abstract data type)Web syndicationSemantic gridInformation retrievalInterface (Java)Computer scienceData exchangeSemantic computingSemantic analyticsSemantic Web StackData miningcomputer.software_genrecomputerProceedings of the 2009 Euro American Conference on Telematics and Information Systems: New Opportunities to increase Digital Citizenship
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Dicationic Organic Salts: our recent journey in their properties and applications

2014

Settore CHIM/06 - Chimica OrganicaDicationic organic salts ionic liquids gel phases self-assembly
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WHY CORPORATES INVEST IN THE SAME START-UP AN EXPLORATIVE ANALYSIS OF CVC SYNDICATIONS

2016

This study investigates why two or more corporates co-invest in the same start-up syndicating their CVC activities. Based on two strands of literature, the CVC and the alliance, we propose a research framework that explores the possible antecedents of CVC syndications. Particularly, grounded on alliance literature, we look at the CVC syndication by combining two dimensions, relational and technological: the relational dimension describes the competitive or cooperative nature of the relationship between partners of CVC syndications, while the technological one represents the exploitative or explorative technological objectives that corporates could pursue when coinvesting in a start-up. We a…

Settore ING-IND/35 - Ingegneria Economico-GestionaleCorporate Venture Capital Co-investment Syndication
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Rendering in corso...

2022

Introduzione al libro "Gaming" di Alexander R. Galloway Introduction to Alexander R. Galloway's "Gaming" book

Settore L-ART/06 - Cinema Fotografia E Televisionegaming videogames postmedication algorithmic society digital culturegaming videogame posticnema società algoritmica cultura digitale
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« La prédication seconde : Essai de mise au point »

2009

La revue "Travaux de linguistique" consacre son cinquante-septième numéro au problème de la prédication seconde dans le domaine de la linguistique française. À travers une série de contributions relevant de plusieurs domaines d'analyse (syntaxique, pragmatique, sémantique) et portant sur des constructions parfois très disparates, ce numéro vise à présenter un état de la question en matière de prédication seconde, qui, en adoptant une attitude réaliste, se soucie moins de fournir des réponses assurées que de poser les bonnes questions. L'objet de l'enquête est, en effet, compliqué dès le départ: quoiqu'il soit possible, en principe et selon des critères de nature partiellement différente, de…

Settore L-LIN/04 - Lingua E Traduzione - Lingua Franceseprédicationprédication seconde
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Cardiovascular Management Self-efficacy: Psychometric Properties of a New Scale and Its Usefulness in a Rehabilitation Context.

2015

Self-efficacy beliefs have been shown to affect various effective health-promoting behaviors in patients. Unfortunately, availability of reliable and valid measures of self-efficacy in cardiovascular diseases (CVDs) is still very limited. Background: Self-efficacy beliefs have been shown to affect various effective health-promoting behaviors in patients. Unfortunately, availability of reliable and valid measures of self-efficacy in cardiovascular diseases (CVDs) is still very limited. Purpose: The aims of this study were to present a new scale measuring self-efficacy beliefs in managing CVD and to examine its psychometric properties. Methods: The study involved 172 patients (mean age = 66.4…

Settore M-PSI/01 - Psicologia GeneraleAdultMalePsychometricsPsychometricsPersonality characteristicsmedicine.medical_treatmentAnxiety; Cardiovascular disease severity; Depression; Illness perception; Impairment in daily functioning; Medication adherence; Personality characteristics; Self-efficacy beliefs;Context (language use)Self-efficacy beliefsAnxietyAffect (psychology)Medication AdherencePersonality characteristicIllness perceptionmedicineCardiovascular disease severityHumansPsychological testingProspective StudiesGeneral PsychologyImpairment in daily functioningAgedSelf-efficacy beliefs; Cardiovascular disease severity; Impairment in daily functioning; Medication adherence; Personality characteristics; Anxiety; Depression; Illness perceptionSelf-efficacyAged 80 and overPsychological TestsRehabilitationCardiac RehabilitationDepressionSelf-efficacy beliefMiddle AgedSelf EfficacySelf-efficacy beliefs . Cardiovascular disease severity . Impairment in daily functioning . Medication adherence . Personality characteristics . Anxiety . Depression . Illness perceptionPsychiatry and Mental healthHealth psychologyCardiovascular DiseasesAnxietyFemalemedicine.symptomPsychologyClinical psychologyAnnals of behavioral medicine : a publication of the Society of Behavioral Medicine
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Disease activity states, reasons for discontinuation and adverse events in 1038 Italian children with juvenile idiopathic arthritis treated with etan…

2017

The advent of biologic medications has increased considerably the potential for treatment benefit in juvenile idiopathic arthritis (JIA), with clinical remission being now achievable in a substantial proportion of patients. However, there is a need of data from the real world of clinical practice to evaluate thoroughly the efficacy and safety profile of the biologic agents currently approved.

Settore MED/38 - Pediatria Generale E Specialisticabiologic medications etanerceptjuvenile idiopathic arthritis
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Efficacy of Low-Dose Paroxetine for the Treatment of Hot Flushes in Surgical and Physiological Postmenopausal Women: Systematic Review and Meta-Analy…

2019

Background and Objectives: Hot flushes and sleep disturbances are the most common vasomotor symptoms (VMS) reported by postmenopausal women. Hormonal treatment is to date referred to as the gold standard approach but not suitable for all the patients. Alternative treatments are needed in case of a contraindication to menopausal hormone therapy (MHT), adverse side effects, and poor compliance. Paroxetine salt is the only nonhormonal medication approved by the US Food and Drug Administration for the management of VMS. Nonetheless, few trials with low consensus are available about this topic. In this review, we aimed to evaluate the efficacy of low-dose paroxetine therapy in the treatment of v…

Sleep Wake Disordersmedicine.medical_specialtyMedicine (General)Ovariectomyvasomotor symptomsefficacymenopauseReviewPlacebosleep disturbanceslaw.inventionR5-920Randomized controlled triallawInternal medicinemedicineHumanshot flusheAdverse effectContraindicationRandomized Controlled Trials as TopicVasomotorbusiness.industryGeneral Medicinemedicine.diseasesleep disturbanceParoxetineMenopausePostmenopauseParoxetineMeta-analysisefficacy; hot flushes; menopause; paroxetine; sleep disturbances; vasomotor symptomsHot FlashesFemalehot flushesbusinessSelective Serotonin Reuptake Inhibitorsmedicine.drugMedicina
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