Search results for "growth"

showing 10 items of 5134 documents

New benzothieno[3,2-d]-1,2,3-triazines with antiproliferative activity: synthesis, spectroscopic studies, and biological activity.

2014

New benzothieno[3,2-d]-1,2,3-triazines, together with precursors triazenylbenzo[b]thiophenes, were designed, synthesized and screened as anticancer agents. The structural features of these compounds prompted us to investigate their DNA binding capability through UV–vis absorption titrations, circular dichroism, and viscometry, pointing out the occurrence of groove-binding. The derivative 3-(4-methoxy-phenyl)benzothieno[3,2-d]-1,2,3-triazin-4(3H)-one showed the highest antiproliferative effect against HeLa cells and was also tested in cell cycle perturbation experiments. The obtained results assessed for the first time the anticancer activity of benzothieno[3,2-d]-1,2,3-triazine nucleus, and…

Circular dichroismStereochemistryClinical BiochemistryPharmaceutical ScienceAntineoplastic AgentsThiophenesBiochemistryHeLachemistry.chemical_compoundStructure-Activity RelationshipSettore BIO/10 - BiochimicaDrug DiscoveryStructure–activity relationshipMoleculeHumansMolecular BiologyCell ProliferationbiologyDose-Response Relationship DrugMolecular StructureChemistryCell growthTriazinesViscosityCircular DichroismOrganic ChemistryCell CycleBiological activityCell cyclebiology.organism_classificationSettore CHIM/08 - Chimica FarmaceuticaCombinatorial chemistrySettore CHIM/03 - Chimica Generale E InorganicaMolecular MedicineBenzothienotriazines Antiproliferative activity Spectroscopic studies Cell-cycle analysis VLAKSpectrophotometry UltravioletDrug Screening Assays AntitumorDNAHeLa CellsBioorganicmedicinal chemistry letters
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Antitumor effects of the novel NF-κB inhibitor dehydroxymethyl-epoxyquinomicin on human hepatic cancer cells: analysis of synergy with cisplatin and …

2006

We tested the novel NF-kappaB inhibitor dehydroxymethylepoxyquinomicin (DHMEQ) in the hepatic cancer (HCC) HepG2, HA22T/VGH and HuH-6 cells. The sensitivity to the cell growth inhibitory and apoptotic effects of the agent increased along with the levels of constitutively activated NF-kappaB, which were low in HepG2 and higher in HA22T/VGH and HuH-6. In HA22T/VGH, DHMEQ exhibited synergy with cisplatin. In the same cells, DHMEQ exerted dose-dependent decreases in the nuclear levels of activated NF-kappaB and attenuated NF-kappaB activation by cisplatin. It down-regulated Bcl-XL mRNA in a dose-dependent manner and up-regulated that of Bcl-XS. It also decreased interleukin 6 (IL-6), NAIP and, …

CisplatinCancer Researchmedicine.medical_specialtyOncogeneCell growthmedicine.medical_treatmentBiologyXIAPEndocrinologyCytokineOncologyApoptosisInternal medicineCancer cellmedicineCancer researchAutocrine signallingmedicine.drugInternational Journal of Oncology
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Evaluation of Chemical Composition of Essential Oils Derived from Different Pelargonium Species Leaves

2019

Abstract Plants have been used for their aromatic and medicinal purposes for centuries. The genus Pelargonium contains about 250-280 species and cultivated around the world for the production of essential oils and absolutes. Pelargonium species are remarkable for their odour diversity, from fresh, lemon and minty scent, through floral, rose, fruity up to spicy and camphoreous smell as well as many health beneficial properties, that is why their essential oils are widely used in perfume, cosmetic, food and pharmaceutical industries. The aim of this study was to determine variability in populations of Pelargonium genus by evaluating their differences in quantitative and qualitative essential …

CitronellolPlant growthEnvironmental EngineeringbiologyPelargoniumbiology.organism_classificationlaw.inventionchemistry.chemical_compoundHorticulturechemistrylawEnvironmental ChemistryCultivarChemical compositionGenus PelargoniumEssential oilGeraniolEcological Chemistry and Engineering S
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Transcriptome and metabolome analysis of citrus fruit to elucidate puffing disorder.

2014

a b s t r a c t A systems-level analysis reveals details of molecular mechanisms underlying puffing disorder in Citrus fruit. Flavedo, albedo and juice sac tissues of normal fruits and fruits displaying symptoms of puffing disorder were studied using metabolomics at three developmental stages. Microarrays were used to compare normal and puffed fruits for each of the three tissues. A protein-protein interaction network inferred from previous work on Arabidopsis identified hub proteins whose transcripts show significant changes in expression. Glycolysis, the backbone of primary metabolism, appeared to be severely affected by the disorder, based on both transcriptomic and metabolomic results. …

CitrusPlant ScienceBiologyTranscriptomechemistry.chemical_compoundMetabolomicsPlant Growth RegulatorsArabidopsisGeneticsMetabolomeBrassinosteroidMetabolomicsProtein Interaction MapsAbscisic acidOligonucleotide Array Sequence AnalysisPlant DiseasesAlbedo breakdown Citrus Fruit disorder Metabolomics Puffing TranscriptomicsGene Expression Profilingfood and beveragesGeneral Medicinebiology.organism_classificationchemistryBiochemistryFruitGibberellinCitric acidAgronomy and Crop ScienceSignal TransductionTranscription FactorsPlant science : an international journal of experimental plant biology
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Transcriptome profiling of citrus fruit response to huanglongbing disease.

2010

Huanglongbing (HLB) or "citrus greening" is the most destructive citrus disease worldwide. In this work, we studied host responses of citrus to infection with Candidatus Liberibacter asiaticus (CaLas) using next-generation sequencing technologies. A deep mRNA profile was obtained from peel of healthy and HLB- affected fruit. It was followed by pathway and protein-protein network analysis and quantitative real time PCR analysis of highly regulated genes. We identified differentially regulated pathways and constructed networks that provide a deep insight into the metabolism of affected fruit. Data mining revealed that HLB enhanced transcription of genes involved in the light reactions of phot…

CitrusProtein FoldingGene Identification and Analysislcsh:MedicinePlant ScienceTranscriptomechemistry.chemical_compoundRNA interferencePlant Growth RegulatorsGene Expression Regulation PlantModelsGene expressionPlant Genomics2.1 Biological and endogenous factorsPhotosynthesisAetiologylcsh:SciencePlant Growth and DevelopmentPlant PestsMultidisciplinaryProtein StabilityJasmonic acidfood and beveragesHigh-Throughput Nucleotide SequencingAgriculturePlantsCell biologyCarbohydrate MetabolismResearch ArticleSignal TransductionGeneral Science & TechnologyPlant PathogensProtein degradationBiologyModels BiologicalFruitsMolecular GeneticsRhizobiaceaeSettore AGR/07 - Genetica AgrariaHeat shock proteinBotanyGeneticsGene RegulationGene NetworksBiologyTranscription factorPlant DiseasesAnalysis of VarianceGene Expression Profilinglcsh:RCitrus HLB next-generation sequencing candidatus liberibacterComputational BiologyPlantPlant PathologyBiologicalWRKY protein domainGene expression profilingchemistryGene Expression Regulationlcsh:QGene expressionGene FunctionTranscriptomeTranscription Factors
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New Arrivals, Old Places: Demographic Changes and New Planning Challenges in Palermo and Naples

2008

If we look at the demographic changes in the largest cities in Southern Italy, the most significant trend is a balance between population growth and decline, affecting in particular inner urban areas, which is due to the predominance of new ethnic inhabitants. After having described these demographic changes in Naples and Palermo, the paper will include some considerations on the ‘institutional’ landscape of planning and the related policies. How do planning policies and practices face this quick change in such peripheral contexts, which are new to the phenomenon? Can the plural composition of the local society be viewed as an opportunity, and not just as a threat? The paper will use some a…

Città multietnica Interetnia Politiche urbanebusiness.industrymedia_common.quotation_subjectGeography Planning and DevelopmentImmigrationEthnic groupDistribution (economics)Face (sociological concept)Context (language use)Settore ICAR/21 - UrbanisticaGeographyEconomyPhenomenonPopulation growthbusinessmedia_commonPluralDemographyInternational Planning Studies
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The Paradox of Effectiveness: Growth, Institutionalisation and Evaluation of Anti-Mafia Policies in Italy

2004

This contribution focuses on Italian policies that have been envisaged and implemented to combat, prevent or contain mafia-type organised crime.1 After having shown that a proper analysis of anti-mafia policies is strangely lacking (section 2), policies directly addressing the mafia are dealt with, hinting at the norms concerning specific criminal offences, vast investigatory powers and penetrating preventive measures, financial transactions and money laundering, collaborators of justice, the peculiarity of mafia trials, judicial attitudes and sanctions (section 3.1). Section 3.2 presents the wide variety of other policies addressing civil society and public administrations, and only indire…

Civil societyEconomic growthInstitutionalisationFinancial transactionEconomicsmedia_common.cataloged_instanceSanctionsLegislationPublic administrationEuropean unionPrinciple of legalityMoney launderingmedia_common
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Institutions, crises, and political confidence in seven contemporary democracies. An elite-mass analysis

2017

There is ample consensus in the literature that institutional confidence by the public is needed in democracies and at the same time elites, particularly political elites, need to share this confidence in their guidance of state institutions, if political stability in established democracies and the consolidation of new democracies are desired. The research takes the form of a quantitative analysis based on the World Values Surveys and the elite surveys (parliamentarians) conducted in 2006 (before the financial crisis) and in 2012–2013 (post the crisis when apparently, the worst of the economic crunch had lessened up) in the 7 countries selected. We explore what lies at the base of politica…

Civil societyEconomic growthLatin AmericansPublic Administration05 social sciencesConfidence intervalCrunch0506 political sciencePoliticsConsolidation (business)0502 economics and businessPolitical Science and International RelationsFinancial crisisDevelopment economicsElite050602 political science & public administrationSociology050207 economicsJournal of Public Affairs
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International development aid and young people's participation in societal development of the global south

2018

International development aid has in recent years sought to strengthen youths’ societal participation by cooperation between international non-governmental organisations (INGOs) and local youth associations. In this paper, we address and conceptualise some of the underlying causes that may enable and/or limit such efforts to support youth participation in the global south. We seek to contribute to the growing literature exploring the multiple scales of young people's political agency. A core argument proposed is that notions of generational relationality, as seen in the case of international development aid targeting youth, must include conceptions of power as a topological relation across …

Civil societyEconomic growthSociology and Political ScienceSocial Psychology05 social sciencesGeography Planning and Development0507 social and economic geographyGlobal South050906 social workPolitical scienceSocietal development0509 other social sciencesInternational development050703 geography
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Rational Foundations of Democratic Politics

2003

1. Introduction Albert Breton, Gianluigi Galeotti, Pierre Salmon and Ronald Wintrobe Part I. Some Problems with Democratic Institutions and Trends in Their Evolution: 2. Demobilization, demoralization and the loosening bonds of electoral politics Michael C. Munger 3. Turning 'citizens' into 'consumers': economic growth and the level of public discourse Stergios Skaperdas 4. Economic and cultural prerequisites for democracy Roger D. Congleton 5. Civil society and the contemporary social order Frederique Chaumont-Chancelier Part II. Morals in Politics: 6. When does altruism overcome the intransitivity of income redistribution? Donald Wittman 7. Democratic resilience and the necessity of virtu…

Civil societymedia_common.quotation_subject05 social sciences050109 social psychologyDemobilization16. Peace & justice[SHS.ECO]Humanities and Social Sciences/Economics and FinanceSolidarityDemocracyPoliticsSocial orderSovereigntyLawPolitical science8. Economic growth0502 economics and business[ SHS.ECO ] Humanities and Social Sciences/Economies and finances0501 psychology and cognitive sciences050207 economics[SHS.ECO] Humanities and Social Sciences/Economics and FinanceSocial capitalLaw and economicsmedia_common
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